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HK1213891A1 - 製備伏立康唑及其類似物的方法 - Google Patents

製備伏立康唑及其類似物的方法

Info

Publication number
HK1213891A1
HK1213891A1 HK16101881.2A HK16101881A HK1213891A1 HK 1213891 A1 HK1213891 A1 HK 1213891A1 HK 16101881 A HK16101881 A HK 16101881A HK 1213891 A1 HK1213891 A1 HK 1213891A1
Authority
HK
Hong Kong
Prior art keywords
voriconazole
analogues
preparation
Prior art date
Application number
HK16101881.2A
Other languages
English (en)
Inventor
．伯里爾
．奧尼爾
．派特曼
Original Assignee
Pfizer Ireland Pharmaceuticals
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Ireland Pharmaceuticals filed Critical Pfizer Ireland Pharmaceuticals
Publication of HK1213891A1 publication Critical patent/HK1213891A1/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/30—Halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK16101881.2A 2012-10-15 2016-02-19 製備伏立康唑及其類似物的方法 HK1213891A1 (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261713761P 2012-10-15 2012-10-15
PCT/IB2013/059202 WO2014060900A1 (en) 2012-10-15 2013-10-08 Process for the preparation of voriconazole and analogues thereof

Publications (1)

Publication Number Publication Date
HK1213891A1 true HK1213891A1 (zh) 2016-07-15

Family

ID=49641810

Family Applications (1)

Application Number Title Priority Date Filing Date
HK16101881.2A HK1213891A1 (zh) 2012-10-15 2016-02-19 製備伏立康唑及其類似物的方法

Country Status (24)

Country Link
US (2) US9388167B2 (zh)
EP (1) EP2906555B1 (zh)
JP (1) JP6180533B2 (zh)
KR (1) KR101706488B1 (zh)
CN (1) CN104884450B (zh)
AU (1) AU2013333534B2 (zh)
BR (1) BR112015007821B1 (zh)
CA (1) CA2888127A1 (zh)
CY (1) CY1118451T1 (zh)
DK (1) DK2906555T3 (zh)
ES (1) ES2615743T3 (zh)
HK (1) HK1213891A1 (zh)
HU (1) HUE031877T2 (zh)
IL (1) IL238209A (zh)
IN (1) IN2015DN02877A (zh)
MX (1) MX358245B (zh)
NZ (1) NZ706764A (zh)
PL (1) PL2906555T3 (zh)
PT (1) PT2906555T (zh)
RU (1) RU2619928C2 (zh)
SG (1) SG11201502237RA (zh)
SI (1) SI2906555T1 (zh)
WO (1) WO2014060900A1 (zh)
ZA (1) ZA201501904B (zh)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101706488B1 (ko) * 2012-10-15 2017-02-13 화이자 아일랜드 파마슈티컬즈 보리코나졸 및 그의 유사체의 제조 방법
CN106432198B (zh) * 2016-09-08 2022-10-21 浙江华海药业股份有限公司 一种制备伏立康唑拆分中间体的方法
CN112898273B (zh) * 2021-03-30 2022-05-31 海南锦瑞制药有限公司 伏立康唑的合成方法及应用
CN113185465B (zh) * 2021-05-26 2022-09-27 无锡捷化医药科技有限公司 一种4-乙基-5-氨基嘧啶的制备方法

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8819308D0 (en) 1988-08-13 1988-09-14 Pfizer Ltd Triazole antifungal agents
GB9002375D0 (en) * 1990-02-02 1990-04-04 Pfizer Ltd Triazole antifungal agents
GB9516121D0 (en) 1995-08-05 1995-10-04 Pfizer Ltd Organometallic addition to ketones
CA2590687C (en) * 2004-12-14 2013-09-10 Dr. Reddy's Laboratories Ltd. Process for preparing voriconazole
BRPI0518509A2 (pt) * 2005-01-10 2008-11-25 Pfizer pirrolopirazàis, inibidores de cinase potentes
KR100889937B1 (ko) * 2007-08-06 2009-03-20 한미약품 주식회사 보리코나졸의 제조방법
WO2011045807A2 (en) * 2009-10-14 2011-04-21 Neuland Laboratories Ltd. A novel process to manufacture (2r,3s)-2-(2,4-difluorophenyl)-3-(5-fluoropyrimidin-4-yl)-1-(1h-1,2,4-triazol-1-yl)butan-2-ol
CN102827073A (zh) * 2011-06-17 2012-12-19 安吉奥斯医药品有限公司 治疗活性组合物和它们的使用方法
CN103814020B (zh) * 2011-06-17 2017-07-14 安吉奥斯医药品有限公司 治疗活性组合物和它们的使用方法
WO2014048065A1 (en) * 2012-09-28 2014-04-03 Merck Sharp & Dohme Corp. Triazolyl derivatives as syk inhibitors
KR101706488B1 (ko) * 2012-10-15 2017-02-13 화이자 아일랜드 파마슈티컬즈 보리코나졸 및 그의 유사체의 제조 방법
JO3383B1 (ar) * 2013-03-14 2019-03-13 Lilly Co Eli مثبطات cdc7

Also Published As

Publication number Publication date
IN2015DN02877A (zh) 2015-09-11
JP2015536305A (ja) 2015-12-21
MX358245B (es) 2018-08-10
US9388167B2 (en) 2016-07-12
US20150239867A1 (en) 2015-08-27
BR112015007821B1 (pt) 2022-02-15
US9499520B2 (en) 2016-11-22
US20160229842A1 (en) 2016-08-11
CA2888127A1 (en) 2014-04-24
CN104884450B (zh) 2017-03-29
AU2013333534B2 (en) 2016-04-14
HUE031877T2 (en) 2017-08-28
CN104884450A (zh) 2015-09-02
MX2015004450A (es) 2015-06-24
PL2906555T3 (pl) 2017-07-31
PT2906555T (pt) 2017-02-15
EP2906555A1 (en) 2015-08-19
RU2619928C2 (ru) 2017-05-22
WO2014060900A1 (en) 2014-04-24
AU2013333534A1 (en) 2015-04-09
BR112015007821A2 (pt) 2017-07-04
SG11201502237RA (en) 2015-05-28
IL238209A0 (en) 2015-06-30
RU2015113741A (ru) 2016-12-10
JP6180533B2 (ja) 2017-08-16
IL238209A (en) 2017-07-31
DK2906555T3 (en) 2017-02-06
KR20150055009A (ko) 2015-05-20
KR101706488B1 (ko) 2017-02-13
CY1118451T1 (el) 2017-07-12
ZA201501904B (en) 2017-01-25
NZ706764A (en) 2017-11-24
ES2615743T3 (es) 2017-06-08
SI2906555T1 (sl) 2017-02-28
EP2906555B1 (en) 2016-12-14

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20231006