HK1118291A1 - Benzothiazole cyclobutyl amine derivatives and their use as histamine-3 receptors ligands - Google Patents
Benzothiazole cyclobutyl amine derivatives and their use as histamine-3 receptors ligandsInfo
- Publication number
- HK1118291A1 HK1118291A1 HK08109754.9A HK08109754A HK1118291A1 HK 1118291 A1 HK1118291 A1 HK 1118291A1 HK 08109754 A HK08109754 A HK 08109754A HK 1118291 A1 HK1118291 A1 HK 1118291A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- histamine
- amine derivatives
- cyclobutyl amine
- receptors ligands
- benzothiazole
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/64—Benzothiazoles with only hydrocarbon or substituted hydrocarbon radicals attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A61P25/00—Drugs for disorders of the nervous system
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- A61P35/00—Antineoplastic agents
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- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/08—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing alicyclic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Reproductive Health (AREA)
- Addiction (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Pregnancy & Childbirth (AREA)
- Rheumatology (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Anesthesiology (AREA)
- Gynecology & Obstetrics (AREA)
- Psychology (AREA)
- Vascular Medicine (AREA)
- Emergency Medicine (AREA)
- Epidemiology (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US71951605P | 2005-09-22 | 2005-09-22 | |
US11/518,132 US7576110B2 (en) | 2005-09-22 | 2006-09-08 | Benzothiazole cyclobutyl amine derivatives |
PCT/US2006/036422 WO2007038074A1 (en) | 2005-09-22 | 2006-09-19 | Benzothiazole cyclobutyl amine derivatives and their use as histamine-3 receptors ligands |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1118291A1 true HK1118291A1 (en) | 2009-02-06 |
Family
ID=37885027
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK08109754.9A HK1118291A1 (en) | 2005-09-22 | 2008-09-02 | Benzothiazole cyclobutyl amine derivatives and their use as histamine-3 receptors ligands |
Country Status (26)
Country | Link |
---|---|
US (2) | US7576110B2 (es) |
EP (2) | EP1926729B1 (es) |
JP (1) | JP2009508957A (es) |
KR (1) | KR20080050628A (es) |
AT (1) | ATE538119T1 (es) |
AU (1) | AU2006295065C1 (es) |
BR (1) | BRPI0616146A2 (es) |
CA (1) | CA2623252A1 (es) |
CR (1) | CR9822A (es) |
CY (1) | CY1112727T1 (es) |
DK (1) | DK1926729T3 (es) |
EC (1) | ECSP088326A (es) |
ES (1) | ES2378197T3 (es) |
HK (1) | HK1118291A1 (es) |
HR (2) | HRP20080174A2 (es) |
IL (1) | IL190350A (es) |
MY (2) | MY150990A (es) |
NO (1) | NO20081905L (es) |
NZ (1) | NZ566834A (es) |
PL (1) | PL1926729T3 (es) |
PT (1) | PT1926729E (es) |
RS (1) | RS52231B (es) |
SI (1) | SI1926729T1 (es) |
TW (1) | TWI393717B (es) |
WO (1) | WO2007038074A1 (es) |
ZA (1) | ZA200802508B (es) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7576110B2 (en) * | 2005-09-22 | 2009-08-18 | Abbott Laboratories | Benzothiazole cyclobutyl amine derivatives |
US9108948B2 (en) * | 2006-06-23 | 2015-08-18 | Abbvie Inc. | Cyclopropyl amine derivatives |
ES2533009T3 (es) * | 2006-06-23 | 2015-04-06 | Abbvie Bahamas Ltd. | Derivados de ciclopropilamina como moduladores del receptor histamina H3 |
JP2010524881A (ja) * | 2007-04-19 | 2010-07-22 | ユセベ ファルマ ソシエテ アノニム | シクロブトキシ基を含むヒスタミンh3受容体リガンド |
US8153813B2 (en) * | 2007-12-20 | 2012-04-10 | Abbott Laboratories | Benzothiazole and benzooxazole derivatives and methods of use |
US20090221648A1 (en) * | 2007-12-21 | 2009-09-03 | Abbott Laboratories | Compositions for treatment of cognitive disorders |
US8383657B2 (en) * | 2007-12-21 | 2013-02-26 | Abbott Laboratories | Thiazolylidine urea and amide derivatives and methods of use thereof |
PE20091883A1 (es) * | 2008-01-24 | 2010-01-07 | Ucb Pharma Sa | Compuestos que comprenden un grupo ciclobutoxi |
KR100986433B1 (ko) | 2008-05-30 | 2010-10-08 | 현대자동차주식회사 | 전동식 파워스티어링 시스템 |
US9186353B2 (en) * | 2009-04-27 | 2015-11-17 | Abbvie Inc. | Treatment of osteoarthritis pain |
WO2012037258A1 (en) | 2010-09-16 | 2012-03-22 | Abbott Laboratories | Processes for preparing 1,2-substituted cyclopropyl derivatives |
JP2016526538A (ja) | 2013-06-20 | 2016-09-05 | バイエル・クロップサイエンス・アクチェンゲゼルシャフト | 殺ダニ剤及び殺虫剤としてのアリールスルフィド誘導体及びアリールスルホキシド誘導体 |
EA202092001A1 (ru) | 2018-03-27 | 2021-01-29 | ПиТиСи ТЕРАПЬЮТИКС, ИНК. | Соединения для лечения болезни гентингтона |
WO2021222366A1 (en) * | 2020-04-28 | 2021-11-04 | Kymera Therapeutics, Inc. | Irak inhibitors and uses thereof |
Family Cites Families (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US78133A (en) * | 1868-05-19 | Improvement in heuometebs | ||
US224952A (en) * | 1880-02-24 | Nventor | ||
US171181A (en) * | 1875-12-14 | Improvement in fence-posts | ||
DE491224C (de) | 1923-05-20 | 1930-02-22 | Leopold Cassella & Co G M B H | Verfahren zur Darstellung von Arylaminosubstitutionsprodukten von o-Aminoarylmercaptanen |
GB8621790D0 (en) | 1986-09-10 | 1986-10-15 | Ici Plc | Tertiary amine compounds |
GB9300194D0 (en) | 1993-01-06 | 1993-03-03 | Wyeth John & Brother Ltd | Piperazine derivatives |
UA71945C2 (en) | 1999-01-27 | 2005-01-17 | Pfizer Prod Inc | Substituted bicyclic derivatives being used as anticancer agents |
RU2174505C1 (ru) | 2000-02-18 | 2001-10-10 | Открытое акционерное общество "Всероссийский научно-исследовательский институт органического синтеза" | Способ получения функционально замещенного метиленциклобутана |
DE10155202A1 (de) * | 2001-11-09 | 2003-07-31 | Boehringer Ingelheim Int | Herstellung und Verwendung von substituierten Imidazolen |
US20030131975A1 (en) * | 2002-01-11 | 2003-07-17 | Sabina Houle | Integrated heat spreader with mechanical interlock designs |
PL376751A1 (pl) | 2002-11-12 | 2006-01-09 | Abbott Laboratories | Bicykliczne podstawione aminy jako ligandy receptora histaminowego-3 |
US20040224952A1 (en) * | 2003-05-07 | 2004-11-11 | Cowart Marlon D. | Fused bicyclic-substituted amines as histamine-3 receptor ligands |
CA2555071A1 (en) * | 2004-02-02 | 2005-09-01 | Pfizer Products Inc. | Histamine-3 receptor modulators |
US7553964B2 (en) | 2005-06-03 | 2009-06-30 | Abbott Laboratories | Cyclobutyl amine derivatives |
US7576110B2 (en) * | 2005-09-22 | 2009-08-18 | Abbott Laboratories | Benzothiazole cyclobutyl amine derivatives |
-
2006
- 2006-09-08 US US11/518,132 patent/US7576110B2/en active Active
- 2006-09-19 EP EP06814914A patent/EP1926729B1/en active Active
- 2006-09-19 MY MYPI20114346 patent/MY150990A/en unknown
- 2006-09-19 RS RS20120112A patent/RS52231B/en unknown
- 2006-09-19 AU AU2006295065A patent/AU2006295065C1/en not_active Ceased
- 2006-09-19 AT AT06814914T patent/ATE538119T1/de active
- 2006-09-19 CA CA002623252A patent/CA2623252A1/en not_active Abandoned
- 2006-09-19 MY MYPI20080763A patent/MY146028A/en unknown
- 2006-09-19 NZ NZ566834A patent/NZ566834A/en not_active IP Right Cessation
- 2006-09-19 KR KR1020087009662A patent/KR20080050628A/ko not_active Application Discontinuation
- 2006-09-19 WO PCT/US2006/036422 patent/WO2007038074A1/en active Application Filing
- 2006-09-19 DK DK06814914.5T patent/DK1926729T3/da active
- 2006-09-19 ES ES06814914T patent/ES2378197T3/es active Active
- 2006-09-19 PL PL06814914T patent/PL1926729T3/pl unknown
- 2006-09-19 SI SI200631280T patent/SI1926729T1/sl unknown
- 2006-09-19 EP EP11165455.4A patent/EP2386556B1/en active Active
- 2006-09-19 PT PT06814914T patent/PT1926729E/pt unknown
- 2006-09-19 BR BRPI0616146-4A patent/BRPI0616146A2/pt not_active IP Right Cessation
- 2006-09-19 JP JP2008532313A patent/JP2009508957A/ja not_active Ceased
- 2006-09-21 TW TW095135007A patent/TWI393717B/zh not_active IP Right Cessation
-
2008
- 2008-03-18 ZA ZA2008/02508A patent/ZA200802508B/en unknown
- 2008-03-20 IL IL190350A patent/IL190350A/en not_active IP Right Cessation
- 2008-03-24 CR CR9822A patent/CR9822A/es unknown
- 2008-03-28 EC EC2008008326A patent/ECSP088326A/es unknown
- 2008-04-15 HR HR20080174A patent/HRP20080174A2/xx not_active Application Discontinuation
- 2008-04-22 NO NO20081905A patent/NO20081905L/no not_active Application Discontinuation
- 2008-09-02 HK HK08109754.9A patent/HK1118291A1/xx not_active IP Right Cessation
-
2009
- 2009-06-22 US US12/489,269 patent/US8592467B2/en active Active
-
2012
- 2012-03-16 CY CY20121100283T patent/CY1112727T1/el unknown
- 2012-03-19 HR HRP20120251TT patent/HRP20120251T1/hr unknown
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PC | Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee) |
Effective date: 20150919 |