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GT199700104BA - Procedimientos e intermedios para preparar derivados de cromanol sustituidos - Google Patents

Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Info

Publication number
GT199700104BA
GT199700104BA GT199700104BL GT199700104L GT199700104BA GT 199700104B A GT199700104B A GT 199700104BA GT 199700104B L GT199700104B L GT 199700104BL GT 199700104 L GT199700104 L GT 199700104L GT 199700104B A GT199700104B A GT 199700104BA
Authority
GT
Guatemala
Prior art keywords
intermediates
procedures
chromanol derivatives
substituted chromanol
prepare substituted
Prior art date
Application number
GT199700104BL
Other languages
English (en)
Inventor
Anthony Piscopio
Joel M Hawkins
Stephane Caron
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of GT199700104BA publication Critical patent/GT199700104BA/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C33/00Unsaturated compounds having hydroxy or O-metal groups bound to acyclic carbon atoms
    • C07C33/40Halogenated unsaturated alcohols
    • C07C33/50Halogenated unsaturated alcohols containing six-membered aromatic rings and other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/04Benzo[b]pyrans, not hydrogenated in the carbocyclic ring
    • C07D311/22Benzo[b]pyrans, not hydrogenated in the carbocyclic ring with oxygen or sulfur atoms directly attached in position 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

ESTA INVENCION SE REFIERE A LA PREPARACION DE DERIVADOS DE CROMANOL SUSTITUIDOS Y A INTERMEDIOS UTILES EN DICHA PREPARACION. LOS DERIVADOS DE CROMANOL SUSTITUIDOS QUE SE PREPARAN DE ACUERDO CON LA PRESENTE INVENCION, INHIBEN LA ACCION DE LTB4. ESTOS COMPUESTOS TIENEN LA ESTRUCTURA QUIMICA(XIII), EN LA QUE R3,R4,R7, SON GRUPOS FUNCIONALES DESCRITOS EN EL EXPEDIENTE.
GT199700104BL 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos GT199700104BA (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US2637296P 1996-09-16 1996-09-16

Publications (1)

Publication Number Publication Date
GT199700104BA true GT199700104BA (es) 1999-03-28

Family

ID=21831429

Family Applications (3)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.
GT199700104AK GT199700104AA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos
GT199700104BL GT199700104BA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Family Applications Before (2)

Application Number Title Priority Date Filing Date
GT199700104A GT199700104A (es) 1996-09-16 1997-09-08 Procedimientos e intermedios para preparar derivados de cromanol sustituidos.
GT199700104AK GT199700104AA (es) 1996-09-16 1997-10-04 Procedimientos e intermedios para preparar derivados de cromanol sustituidos

Country Status (39)

Country Link
US (4) US6096906A (es)
EP (1) EP0925292B1 (es)
JP (1) JP3117730B2 (es)
KR (1) KR100339164B1 (es)
CN (1) CN1108298C (es)
AP (1) AP726A (es)
AT (1) ATE249452T1 (es)
AU (1) AU713701B2 (es)
BG (1) BG63542B1 (es)
BR (1) BR9711482A (es)
CA (1) CA2265043C (es)
CO (1) CO4600635A1 (es)
DE (1) DE69724801T2 (es)
DK (1) DK0925292T3 (es)
DZ (1) DZ2308A1 (es)
EA (1) EA002204B1 (es)
ES (1) ES2206738T3 (es)
GT (3) GT199700104A (es)
HN (1) HN1997000127A (es)
HR (1) HRP970497B1 (es)
ID (1) ID19613A (es)
IL (1) IL128732A0 (es)
IS (1) IS4980A (es)
MA (1) MA24319A1 (es)
NO (1) NO991254L (es)
NZ (1) NZ334214A (es)
OA (1) OA10995A (es)
PA (1) PA8437901A1 (es)
PE (1) PE109798A1 (es)
PL (1) PL332351A1 (es)
PT (1) PT925292E (es)
SK (1) SK31399A3 (es)
TN (1) TNSN97155A1 (es)
TR (1) TR199900592T2 (es)
TW (1) TW449579B (es)
UA (1) UA58520C2 (es)
WO (1) WO1998011085A1 (es)
YU (1) YU13299A (es)
ZA (1) ZA978291B (es)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6436987B1 (en) * 2000-06-08 2002-08-20 Pfizer Inc. Crystalline forms of (3S-trans)-2-[3,4-dihydro-4-hydroxy-3-(phenylmethyl)-2H-1-benzopyran-7-yl]-4-(trifluoromethyl)-benzoic acid
BR0206771A (pt) * 2001-01-30 2004-02-25 Pfizer Prod Inc Processos para a preparação de cidos cromanilbenzóicos
AU4239302A (en) * 2001-06-28 2003-01-02 Pfizer Products Inc. Benzoic acid substituted benzopyrans for the treatment of atherosclerosis
CA2694068C (en) * 2007-07-23 2016-08-30 The Board Of Trustees Of The University Of Illinois System for controlling the reactivity of boronic acids
US8338601B2 (en) 2008-09-26 2012-12-25 Board Of Trustees Of The University Of Illinois Slow release of organoboronic acids in cross-coupling reactions
US8304513B2 (en) * 2009-09-02 2012-11-06 E I Du Pont De Nemours And Company Polyesters comprising fluorovinylether functionalized aromatic moieties
MX2012002588A (es) * 2009-09-02 2012-04-02 Du Pont Peliculas de poliester con repelencia al aceite mejorada.
US20110218319A1 (en) * 2009-09-02 2011-09-08 E. I. Du Pont De Nemours And Company Polyaramid films comprising fluorovinylether functionalized aromatic moieties
CN102597060B (zh) * 2009-09-02 2014-05-07 纳幕尔杜邦公司 包含氟乙烯基醚官能化芳族部分的芳族聚酰胺
EP2473474A4 (en) 2009-09-02 2012-10-24 Du Pont FUNCTIONALIZED AROMATIC DIESTERS OF FLUOROETHER AND DERIVATIVES THEREOF
WO2011028766A2 (en) * 2009-09-02 2011-03-10 E. I. Du Pont De Nemours And Company Fluorinated 4-oxo-chroman-carboxylates
US8557980B2 (en) 2010-02-18 2013-10-15 The Board Of Trustees Of The University Of Illinois Methods for forming protected organoboronic acids
WO2016149126A1 (en) 2015-03-13 2016-09-22 The Board Of Trustees Of The Leland Stanford Junior University Ltb4 inhibition to prevent and treat human lymphedema
KR102807066B1 (ko) * 2019-09-30 2025-05-15 주식회사 엘지화학 아민계 화합물 제조방법

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9119920D0 (en) * 1991-09-18 1991-10-30 Glaxo Group Ltd Chemical compounds
AU2773392A (en) * 1992-01-23 1993-09-01 Pfizer Inc. Benzopyran and related LTB4 antagonists
MX9300312A (es) * 1992-01-23 1993-07-31 Pfizer Antagonistas benzopiranicos y relacionado de ltb.
PL308474A1 (en) * 1992-10-21 1995-08-07 Pfizer Sulphonamidic derivatives of hydroxy substituted cycloalkylic and heterocyclic compounds with condensed benzene ring
WO1994008986A1 (en) * 1992-10-21 1994-04-28 Pfizer, Inc. Enantiomeric cis-3-(4,6-dihydroxychroman-3-yl-methyl)benzoic acids
WO1996011925A1 (en) * 1994-10-13 1996-04-25 Pfizer Inc. Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene b4' (ltb4) antagonists
PL319688A1 (en) * 1994-10-13 1997-08-18 Pfizer Benzopyrane and benzo-condensed compounds, method of obtaining them and their application as antagosists of leucotriene b4 (ltb4)
US5539128A (en) * 1994-11-30 1996-07-23 Pfizer Inc. Processes and intermediates for preparing cis(+)3-[4,6-dihydroxy chroman-3-ylmethyl]-4-methoxyaniline

Also Published As

Publication number Publication date
TW449579B (en) 2001-08-11
DE69724801D1 (de) 2003-10-16
SK31399A3 (en) 2000-05-16
CA2265043C (en) 2003-01-14
PL332351A1 (en) 1999-09-13
KR100339164B1 (ko) 2002-06-01
CA2265043A1 (en) 1998-03-19
US6444826B1 (en) 2002-09-03
MA24319A1 (fr) 1998-04-01
US6355825B1 (en) 2002-03-12
DE69724801T2 (de) 2004-06-17
IS4980A (is) 1999-02-16
HN1997000127A (es) 1997-12-20
WO1998011085A1 (en) 1998-03-19
GT199700104A (es) 1999-03-02
ZA978291B (en) 1999-03-15
PT925292E (pt) 2004-01-30
PA8437901A1 (es) 2000-05-24
BG63542B1 (bg) 2002-04-30
BG103231A (en) 1999-12-30
BR9711482A (pt) 1999-08-24
NO991254D0 (no) 1999-03-15
ATE249452T1 (de) 2003-09-15
CO4600635A1 (es) 1998-05-08
YU13299A (sh) 2001-03-07
EP0925292A1 (en) 1999-06-30
ID19613A (id) 1998-07-23
JP2000502726A (ja) 2000-03-07
TNSN97155A1 (fr) 2005-03-15
DZ2308A1 (fr) 2002-12-28
EA002204B1 (ru) 2002-02-28
UA58520C2 (uk) 2003-08-15
US6096906A (en) 2000-08-01
CN1230954A (zh) 1999-10-06
AP726A (en) 1999-01-29
US6288242B1 (en) 2001-09-11
US20020099227A1 (en) 2002-07-25
NO991254L (no) 1999-05-14
AU713701B2 (en) 1999-12-09
HRP970497B1 (en) 2002-06-30
JP3117730B2 (ja) 2000-12-18
CN1108298C (zh) 2003-05-14
ES2206738T3 (es) 2004-05-16
US20020042526A1 (en) 2002-04-11
HRP970497A2 (en) 1998-08-31
AU3781497A (en) 1998-04-02
NZ334214A (en) 2000-09-29
OA10995A (en) 2001-11-06
TR199900592T2 (xx) 1999-06-21
EP0925292B1 (en) 2003-09-10
DK0925292T3 (da) 2004-01-12
KR20000036136A (ko) 2000-06-26
GT199700104AA (es) 1999-03-28
AP9701083A0 (en) 1997-10-31
IL128732A0 (en) 2000-01-31
EA199900204A1 (ru) 1999-08-26
PE109798A1 (es) 1999-01-13

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