[go: up one dir, main page]
More Web Proxy on the site http://driver.im/

ES8702423A1 - Un procedimiento para la preparacion de tiazol y tiazin-ben-cimidazoles - Google Patents

Un procedimiento para la preparacion de tiazol y tiazin-ben-cimidazoles

Info

Publication number
ES8702423A1
ES8702423A1 ES545233A ES545233A ES8702423A1 ES 8702423 A1 ES8702423 A1 ES 8702423A1 ES 545233 A ES545233 A ES 545233A ES 545233 A ES545233 A ES 545233A ES 8702423 A1 ES8702423 A1 ES 8702423A1
Authority
ES
Spain
Prior art keywords
formula
chr
independently represent
heteroaryl
ring
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES545233A
Other languages
English (en)
Other versions
ES545233A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
John Wyeth and Brother Ltd
Original Assignee
John Wyeth and Brother Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB838316645A external-priority patent/GB8316645D0/en
Priority claimed from GB838333231A external-priority patent/GB8333231D0/en
Application filed by John Wyeth and Brother Ltd filed Critical John Wyeth and Brother Ltd
Publication of ES8702423A1 publication Critical patent/ES8702423A1/es
Publication of ES545233A0 publication Critical patent/ES545233A0/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

PROCEDIMIENTO PARA LA OBTENCION DE TIAZOL Y TIAZIN-BENZIMIDAZOLES, DE FORMULA (I), Y DE SUS SALES. COMPRENDE LA REACCION DE CICLIZACION DE UN COMPUESTO DE FORMULA (II), PARA FORMAR UN COMPUESTO DE FORMULA (I), EN LA QUE -B-B1- ES UNA CADENA RADICAL DE 1 O 2 ATOMOS DE CARBONO QUE PUEDEN ESTAR SUSTITUIDOS POR VARIOS TIPOS DE RADICALES, R Y R1-R4 REPRESENTAN HIDROGENO O VARIOS SUSTITUYENTES, Y UNO DE A Y B2 ES SH Y EL OTRO ES UN GRUPO PARTIENTE. LA REACCION SE LLEVA A CABO POR CALENTAMIENTO, EN PRESENCIA DE UNA BASE O DE UN ACIDO. ESTOS COMPUESTOS TIENEN APLICACIONES FARMACOLOGICAS POR SU ACTIVIDAD ANTIBACTERIANA Y ANTIFUNGAL.
ES545233A 1983-06-18 1985-07-16 Un procedimiento para la preparacion de tiazol y tiazin-ben-cimidazoles Expired ES8702423A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB838316645A GB8316645D0 (en) 1983-06-18 1983-06-18 Heterocyclic compounds
GB838333231A GB8333231D0 (en) 1983-12-13 1983-12-13 Heterocyclic compounds

Publications (2)

Publication Number Publication Date
ES8702423A1 true ES8702423A1 (es) 1987-01-01
ES545233A0 ES545233A0 (es) 1987-01-01

Family

ID=26286415

Family Applications (3)

Application Number Title Priority Date Filing Date
ES533496A Expired ES8607323A1 (es) 1983-06-18 1984-06-16 Un procedimiento para la preparacion de tiazol y tiazin-bencimidazoles
ES545233A Expired ES8702423A1 (es) 1983-06-18 1985-07-16 Un procedimiento para la preparacion de tiazol y tiazin-ben-cimidazoles
ES545234A Expired ES8702424A1 (es) 1983-06-18 1985-07-16 Un procedimiento para la preparacion de tiazol y tiazin-ben-cimidazoles

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES533496A Expired ES8607323A1 (es) 1983-06-18 1984-06-16 Un procedimiento para la preparacion de tiazol y tiazin-bencimidazoles

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES545234A Expired ES8702424A1 (es) 1983-06-18 1985-07-16 Un procedimiento para la preparacion de tiazol y tiazin-ben-cimidazoles

Country Status (14)

Country Link
EP (1) EP0129409B1 (es)
JP (1) JPS6013794A (es)
KR (1) KR910009212B1 (es)
AR (2) AR243895A1 (es)
AT (1) ATE96441T1 (es)
AU (1) AU569519B2 (es)
DE (1) DE3486233T2 (es)
DK (1) DK296084A (es)
ES (3) ES8607323A1 (es)
FI (1) FI80458C (es)
GB (1) GB2141429B (es)
GR (1) GR81595B (es)
IE (1) IE57723B1 (es)
PT (1) PT78734B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1341314C (en) 1984-07-06 2001-11-06 David Cox Derivatives of benzimidazole, benzothiazole and benzoxazole
GB8506657D0 (en) * 1985-03-14 1985-04-17 Wyeth John & Brother Ltd Heterocyclic compounds
PT859612E (pt) * 1995-09-21 2003-10-31 Pharma Pass Ii Llc Composicao farmaceutica contendo um omeprazol acid-labil e um processo para a sua preparacao
US20060024362A1 (en) 2004-07-29 2006-02-02 Pawan Seth Composition comprising a benzimidazole and process for its manufacture

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE242226C (es) *
US3704239A (en) * 1971-03-17 1972-11-28 American Home Prod Certain thiazole(3,2-a)benzimidazole compounds
DE2155415A1 (de) * 1971-11-08 1973-05-17 Jose Rosan Verfahren und vorrichtung zur gewinnung eines extrakts aus einer nahrungsmittelsubstanz
HU169255B (es) * 1973-06-20 1976-10-28
GB1601335A (en) * 1978-05-26 1981-10-28 Ruskin B E S Methods and apparatus for packaging and preparing beverages
US4214089A (en) * 1978-07-18 1980-07-22 American Home Products Corporation Thiazolo[3,2-a]benzimidazoles, imidazo [2,1-b]thiazoles, and related compounds as antineoplastic agents, and enhancers of the immune response
JPS6038396B2 (ja) * 1979-07-26 1985-08-31 エスエス製薬株式会社 イミダゾ−ル誘導体及びその製造法
JPS579787A (en) * 1980-06-20 1982-01-19 Ss Pharmaceut Co Ltd Thiazinobenzimidazole derivative and its preparation
US4293696A (en) * 1980-12-22 1981-10-06 American Home Products Corporation 3-Substituted phenylthiazolo[3'2':1,2]imidazo[4,5-b]pyridine-2-alkanoic acids
US4376769A (en) * 1981-06-19 1983-03-15 Schering Corporation Substituted imidazo thiazoles thiazines, thiazepines and thiazocines

Also Published As

Publication number Publication date
ATE96441T1 (de) 1993-11-15
GB2141429B (en) 1986-12-10
FI80458B (fi) 1990-02-28
KR910009212B1 (ko) 1991-11-05
EP0129409A2 (en) 1984-12-27
EP0129409B1 (en) 1993-10-27
PT78734B (en) 1986-06-03
AU2917784A (en) 1984-12-20
FI842353A0 (fi) 1984-06-11
DE3486233T2 (de) 1994-03-03
DK296084A (da) 1984-12-19
AR242214A1 (es) 1993-03-31
JPS6013794A (ja) 1985-01-24
FI80458C (fi) 1990-06-11
ES533496A0 (es) 1986-06-01
EP0129409A3 (en) 1985-12-18
DK296084D0 (da) 1984-06-15
DE3486233D1 (de) 1993-12-02
GB8415173D0 (en) 1984-07-18
GR81595B (es) 1984-12-11
KR850000461A (ko) 1985-02-27
ES545234A0 (es) 1987-01-01
ES8607323A1 (es) 1986-06-01
ES545233A0 (es) 1987-01-01
IE841399L (en) 1984-12-18
AR243895A1 (es) 1993-09-30
GB2141429A (en) 1984-12-19
PT78734A (pt) 1985-01-01
ES8702424A1 (es) 1987-01-01
FI842353A (fi) 1984-12-19
JPH0564155B2 (es) 1993-09-14
IE57723B1 (en) 1993-03-24
AU569519B2 (en) 1988-02-04

Similar Documents

Publication Publication Date Title
KR940007270B1 (en) Quinazoline derivatives
EP1035123A4 (en) NEW HETEROCYCLIC COMPOUNDS
MY109737A (en) Treatment and compounds.
ES8801651A1 (es) Un procedimiento para preparar fenixialquil(substituido con heterociclo)-isozazoles y furanos
NZ335388A (en) New benzothiophene, benzofuran and indole compounds, a process for their preparation and pharmaceutical compositions containing them for treatment of thrombosis
DK457286A (da) Fluorenforbindelse og farmaceutisk praeparat indeholdende en saadan forbindelse
DK519985D0 (da) Quinoloncarboxylsyrederivater, fremgangsmaade til fremstilling deraf og antibakterielt middel indeholdende saadanne derivater
DK322588A (da) Cycloalkylamider af 6-substituerede (8beta)-1-alkylergoliner og fremgangsmaade til fremstilling af saadanne forbindelser
ES8702424A1 (es) Un procedimiento para la preparacion de tiazol y tiazin-ben-cimidazoles
DE69001111D1 (de) Antikrebs-zusammensetzung.
ATE55057T1 (de) Zentralwirkende muskelrelaxante.
HUP9904594A2 (hu) Piperazinoszármazékok, ezeket tartalmazó gyógyszerkészítmények és alkalmazásuk
DE69007356D1 (de) Zyklisches Tetrapeptid und Verfahren zu dessen Herstellung.
ES8404980A1 (es) Un procedimiento para preparar guanidino-fenilamidinas heterociclicas sustituidas.
ES8304940A1 (es) "procedimiento para la preparacion de heteroariloxipropanolaminas".
HU913293D0 (en) Process for the production of pierazine derivatives and medical preparations containing them
CY1742A (en) Mitomycin analogs a process for preparing them and pharmaceutical compositions
GR3026006T3 (en) Pyridazinone derivatives, processes for production thereof and use thereof.
MY104164A (en) Heterocyclic compounds.