ES2134563T3 - Cianofenilsulfenil halogenuro y su utilizacion en el procedimiento de preparacion de benzoisotiazol 3-sustituido. - Google Patents
Cianofenilsulfenil halogenuro y su utilizacion en el procedimiento de preparacion de benzoisotiazol 3-sustituido.Info
- Publication number
- ES2134563T3 ES2134563T3 ES96302851T ES96302851T ES2134563T3 ES 2134563 T3 ES2134563 T3 ES 2134563T3 ES 96302851 T ES96302851 T ES 96302851T ES 96302851 T ES96302851 T ES 96302851T ES 2134563 T3 ES2134563 T3 ES 2134563T3
- Authority
- ES
- Spain
- Prior art keywords
- substituted
- halogenuro
- cyanofenilsulfenil
- benzoisotiazole
- preparation procedure
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C255/00—Carboxylic acid nitriles
- C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
- C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C313/08—Sulfenic acids; Derivatives thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C313/00—Sulfinic acids; Sulfenic acids; Halides, esters or anhydrides thereof; Amides of sulfinic or sulfenic acids, i.e. compounds having singly-bound oxygen atoms of sulfinic or sulfenic groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C313/08—Sulfenic acids; Derivatives thereof
- C07C313/10—Sulfenic acids; Esters thereof
- C07C313/16—Sulfenic acids; Esters thereof having sulfur atoms of sulfenic groups bound to carbon atoms of six-membered aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
UN COMPUESTO DE 2-CIANOBENCENOSULFENIL ESTA REPRESENTADO POR LA FORMULA GENERAL (I): EN DONDE X REPRESENTA CL O BR Y PUEDE SER UTILIZADO PARA LA PREPARACION DE BENCISOTIAZOL 3-SUBSTITUIDO POR LA REACCION DEL COMPUESTO (I) CON UN COMPUESTO DE PIPERAZINA. EL COMPUESTO (I) PUEDE SER PREPARADO POR HALOGENACION DE UN DERIVADO DE 2-CIANOFENILTIO DE LA FORMULA (II): EN DONDE R REPRESENTA H, METAL ALCALINO, 2-CIANOFENILTIO O ALQUILO C{SUB,1-4}.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP09838795A JP3701044B2 (ja) | 1995-04-24 | 1995-04-24 | シアノベンゼンスルフェニルハライドおよびそれを用いる3−置換ベンゾイソチアゾールの製造方法 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES2134563T3 true ES2134563T3 (es) | 1999-10-01 |
Family
ID=14218454
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES96302851T Expired - Lifetime ES2134563T3 (es) | 1995-04-24 | 1996-04-24 | Cianofenilsulfenil halogenuro y su utilizacion en el procedimiento de preparacion de benzoisotiazol 3-sustituido. |
Country Status (9)
Country | Link |
---|---|
US (2) | US5679827A (es) |
EP (1) | EP0741129B1 (es) |
JP (1) | JP3701044B2 (es) |
KR (1) | KR100387538B1 (es) |
CN (2) | CN1061975C (es) |
CA (1) | CA2174797C (es) |
DE (1) | DE69602802T2 (es) |
ES (1) | ES2134563T3 (es) |
TW (1) | TW326033B (es) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN1071324C (zh) * | 1995-11-07 | 2001-09-19 | 辉瑞大药厂 | 制备3-(1-哌嗪基)-1,2-苯并异噻唑的方法和中间体 |
JP3996228B2 (ja) * | 1996-10-11 | 2007-10-24 | 住友精化株式会社 | 3−ピペラジニルベンズイソチアゾール類の製造法 |
TWI232214B (en) * | 1998-04-16 | 2005-05-11 | Shionogi & Co | Preparation of aryl sulfenyl halide |
WO2001012594A1 (fr) * | 1999-08-12 | 2001-02-22 | Nippon Finechemical Co., Ltd. | Procede de preparation de chlorures de sulfenyle aromatiques et autres |
WO2004002950A1 (ja) * | 2002-06-28 | 2004-01-08 | Shimadzu Corporation | スルフェニル化合物、ラベル化試薬、及びペプチドの解析方法 |
US8981095B2 (en) | 2011-07-28 | 2015-03-17 | Mapi Pharma Ltd. | Intermediate compounds and process for the preparation of lurasidone and salts thereof |
CN105669588B (zh) * | 2016-03-16 | 2017-11-07 | 天津大学 | 苯并异噻唑类衍生物的制备方法 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2609864C2 (de) * | 1976-03-10 | 1984-02-16 | Basf Ag, 6700 Ludwigshafen | Verfahren zur Herstellung von 3-Amino-1,2-benzisothiazolen |
EP0053652A1 (de) * | 1980-11-10 | 1982-06-16 | Klaus Arlt | Energie-Erzeuger: Maschinelle Vorrichtung zur Erzeugung von Energie durch Schwerkraftwirkung |
US4590196A (en) * | 1984-08-23 | 1986-05-20 | Bristol-Myers Company | Analgesic 1,2-benzisothiazol-3-ylpiperazine derivatives |
JPH0625181B2 (ja) * | 1985-03-27 | 1994-04-06 | 住友製薬株式会社 | 新規なイミド誘導体 |
JPS6383067A (ja) * | 1986-09-26 | 1988-04-13 | Sumitomo Pharmaceut Co Ltd | 新規コハク酸イミド誘導体 |
JPS6383085A (ja) * | 1986-09-26 | 1988-04-13 | Sumitomo Pharmaceut Co Ltd | 新規なイミド誘導体 |
TW241263B (es) * | 1991-08-22 | 1995-02-21 | Hoechst Roussel Pharma | |
US5359068A (en) * | 1993-06-28 | 1994-10-25 | Pfizer Inc. | Processes and intermediates for the preparation of 5-[2-(4-(benzoisothiazol-3-yl)-piperazin-1-yl)ethyl]-6-chloro-1,3-dihydro-indol-2-one |
-
1995
- 1995-04-24 JP JP09838795A patent/JP3701044B2/ja not_active Expired - Fee Related
-
1996
- 1996-04-10 US US08/630,730 patent/US5679827A/en not_active Expired - Lifetime
- 1996-04-12 TW TW085104333A patent/TW326033B/zh not_active IP Right Cessation
- 1996-04-23 CA CA002174797A patent/CA2174797C/en not_active Expired - Fee Related
- 1996-04-23 KR KR1019960012366A patent/KR100387538B1/ko not_active IP Right Cessation
- 1996-04-24 EP EP96302851A patent/EP0741129B1/en not_active Expired - Lifetime
- 1996-04-24 ES ES96302851T patent/ES2134563T3/es not_active Expired - Lifetime
- 1996-04-24 CN CN96106019A patent/CN1061975C/zh not_active Expired - Fee Related
- 1996-04-24 CN CNB001086383A patent/CN1187346C/zh not_active Expired - Fee Related
- 1996-04-24 DE DE69602802T patent/DE69602802T2/de not_active Expired - Lifetime
-
1997
- 1997-05-21 US US08/861,426 patent/US5756806A/en not_active Expired - Lifetime
Also Published As
Publication number | Publication date |
---|---|
JP3701044B2 (ja) | 2005-09-28 |
CA2174797A1 (en) | 1996-10-25 |
TW326033B (en) | 1998-02-01 |
KR960037647A (ko) | 1996-11-19 |
EP0741129A3 (en) | 1997-05-07 |
DE69602802D1 (de) | 1999-07-15 |
CA2174797C (en) | 2007-01-09 |
CN1289770A (zh) | 2001-04-04 |
EP0741129A2 (en) | 1996-11-06 |
US5679827A (en) | 1997-10-21 |
CN1138032A (zh) | 1996-12-18 |
CN1061975C (zh) | 2001-02-14 |
JPH08291134A (ja) | 1996-11-05 |
DE69602802T2 (de) | 1999-10-21 |
CN1187346C (zh) | 2005-02-02 |
US5756806A (en) | 1998-05-26 |
EP0741129B1 (en) | 1999-06-09 |
KR100387538B1 (ko) | 2003-11-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FG2A | Definitive protection |
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