EG24137A - Tropane derivatives useful in therapy - Google Patents

Tropane derivatives useful in therapy

Info

Publication number: EG24137A
Authority: EG; Egypt
Prior art keywords: therapy; derivatives useful; tropane derivatives; tropane; useful
Prior art date: 2000-05-26

Application number

EG20010535A

Other languages

English (en)

Inventor

Perros Manoussos

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-26

Filing date

2001-05-22

Publication date

2008-08-06

2000-05-26 Priority claimed from GB0014046A external-priority patent/GB0014046D0/en

2000-06-27 Priority claimed from GB0015835A external-priority patent/GB0015835D0/en

2001-05-22 Application filed by Pfizer filed Critical Pfizer

2008-08-06 Application granted granted Critical

2008-08-06 Publication of EG24137A publication Critical patent/EG24137A/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4196—1,2,4-Triazoles
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
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- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/12—Antidiarrhoeals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
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- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
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- A61P19/00—Drugs for skeletal disorders
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A—HUMAN NECESSITIES
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- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
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- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
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- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Immunology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Cardiology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Virology (AREA)
Obesity (AREA)
Hospice & Palliative Care (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Hematology (AREA)
Endocrinology (AREA)
Physical Education & Sports Medicine (AREA)
Urology & Nephrology (AREA)
Heart & Thoracic Surgery (AREA)
Rheumatology (AREA)
Molecular Biology (AREA)
Orthopedic Medicine & Surgery (AREA)
AIDS & HIV (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Emergency Medicine (AREA)
Transplantation (AREA)

EG20010535A 2000-05-26 2001-05-22 Tropane derivatives useful in therapy EG24137A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB0014046A GB0014046D0 (en)	2000-05-26	2000-05-26	Compounds useful in therapy
GB0015835A GB0015835D0 (en)	2000-06-27	2000-06-27	Compounds useful in therapy

Publications (1)

Publication Number	Publication Date
EG24137A true EG24137A (en)	2008-08-06

Family

ID=26244452

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EG20010535A EG24137A (en)	2000-05-26	2001-05-22	Tropane derivatives useful in therapy

Country Status (51)

Country	Link
EP (3)	EP1284974B1 (de)
JP (2)	JP3693957B2 (de)
KR (2)	KR100523501B1 (de)
CN (2)	CN100355753C (de)
AP (1)	AP1965A (de)
AR (2)	AR028622A1 (de)
AT (2)	ATE260914T1 (de)
AU (2)	AU2001252482B2 (de)
BG (1)	BG65966B1 (de)
BR (1)	BRPI0110955B8 (de)
CA (1)	CA2408909C (de)
CR (1)	CR10145A (de)
CU (1)	CU23288B7 (de)
CY (3)	CY2008006I1 (de)
CZ (1)	CZ299102B6 (de)
DE (3)	DE60102233T2 (de)
DK (2)	DK1526134T3 (de)
DZ (1)	DZ3464A1 (de)
EA (2)	EA007580B1 (de)
EE (1)	EE05110B1 (de)
EG (1)	EG24137A (de)
ES (3)	ES2311126T3 (de)
FR (1)	FR08C0007I2 (de)
GE (1)	GEP20063799B (de)
HK (3)	HK1054927A1 (de)
HR (1)	HRP20020938B1 (de)
HU (1)	HU225810B1 (de)
IL (2)	IL152531A0 (de)
IS (1)	IS2511B (de)
LT (1)	LTC1284974I2 (de)
LU (1)	LU91417I2 (de)
MA (1)	MA26902A1 (de)
ME (1)	ME00555A (de)
MX (1)	MXPA02011631A (de)
MY (3)	MY156920A (de)
NL (1)	NL300338I2 (de)
NO (3)	NO327892B1 (de)
NZ (1)	NZ521477A (de)
OA (1)	OA12264A (de)
PA (1)	PA8517101A1 (de)
PE (1)	PE20011371A1 (de)
PL (1)	PL200551B1 (de)
PT (2)	PT1284974E (de)
RS (2)	RS50904B (de)
SI (2)	SI1526134T1 (de)
SK (1)	SK286129B6 (de)
TN (1)	TNSN01077A1 (de)
TR (1)	TR200400541T4 (de)
TW (1)	TWI230160B (de)
UY (1)	UY26727A1 (de)
WO (1)	WO2001090106A2 (de)

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Also Published As

Publication number	Publication date
IL152531A (en)	2010-05-17
AU5248201A (en)	2001-12-03
ME00555B (me)	2011-12-20
NO2010007I2 (no)	2013-09-09
MXPA02011631A (es)	2003-03-27
ME00555A (en)	2011-12-20
NO327892B1 (no)	2009-10-12
DK1284974T3 (da)	2004-06-07
ES2311126T3 (es)	2009-02-01
AU2001252482B2 (en)	2006-01-19
YU82202A (sh)	2005-11-28
BRPI0110955B1 (pt)	2016-06-28
LTPA2008004I1 (lt)	2020-07-27
CY2008006I2 (el)	2009-11-04
MA26902A1 (fr)	2004-12-20
AP2002002663A0 (en)	2002-12-31
LTC1284974I2 (lt)	2020-11-10
CY2008006I1 (el)	2009-11-04
HUP0302474A2 (hu)	2003-11-28
TR200400541T4 (tr)	2004-04-21
CU23288B7 (es)	2008-06-30
AR060159A2 (es)	2008-05-28
PT1526134E (pt)	2008-10-28
CY1108451T1 (el)	2014-04-09
ES2401812T3 (es)	2013-04-24
PE20011371A1 (es)	2002-01-18
HU225810B1 (en)	2007-10-29
SK16432002A3 (sk)	2004-01-08
LU91417I9 (de)	2019-01-02
CZ20023806A3 (cs)	2004-01-14
ATE260914T1 (de)	2004-03-15
EP1526134B1 (de)	2008-09-03
LU91417I2 (fr)	2008-04-22
FR08C0007I2 (fr)	2009-01-15
MY131019A (en)	2007-07-31
EP1284974B1 (de)	2004-03-03
FR08C0007I1 (de)	2008-04-25
DE60135685D1 (de)	2008-10-16
CA2408909A1 (en)	2001-11-29
CY2022009I2 (el)	2022-05-27
HK1078573A1 (en)	2006-03-17
KR100523501B1 (ko)	2005-10-25
NO20025227L (no)	2002-10-31
ATE407134T1 (de)	2008-09-15
EP1526134A2 (de)	2005-04-27
CN1437599A (zh)	2003-08-20
CN100355753C (zh)	2007-12-19
TNSN01077A1 (fr)	2005-11-10
NL300338I2 (nl)	2008-06-02
CR10145A (es)	2008-08-19
JP3693957B2 (ja)	2005-09-14
ES2215129T3 (es)	2004-10-01
SK286129B6 (sk)	2008-04-07
AU2001252482C1 (en)	2001-12-03
CY2022009I1 (el)	2022-05-27
EP1990341A1 (de)	2008-11-12
DE122008000011I1 (de)	2008-06-05
RS50904B (sr)	2010-08-31
NO2010007I1 (no)	2010-04-08
GEP20063799B (en)	2006-04-25
EE200200656A (et)	2004-06-15
IL152531A0 (en)	2003-05-29
JP4854970B2 (ja)	2012-01-18
UY26727A1 (es)	2001-12-28
PT1284974E (pt)	2004-06-30
OA12264A (en)	2003-11-10
BG107140A (bg)	2003-05-30
HRP20020938B1 (en)	2011-05-31
NL300338I1 (nl)	2008-05-01
HK1090836A1 (en)	2007-01-05
MY156920A (en)	2016-04-15
CZ299102B6 (cs)	2008-04-23
PL359267A1 (en)	2004-08-23
MY153023A (en)	2014-12-31
EP1990341B1 (de)	2013-01-23
CN1680371A (zh)	2005-10-12
EA200201141A1 (ru)	2003-04-24
WO2001090106A3 (en)	2002-03-28
IS6565A (is)	2002-09-24
SI1526134T1 (sl)	2008-12-31
KR20030004417A (ko)	2003-01-14
KR20050046743A (ko)	2005-05-18
PL200551B1 (pl)	2009-01-30
EA005382B1 (ru)	2005-02-24
EP1284974A2 (de)	2003-02-26
BR0110955A (pt)	2003-06-03
HUP0302474A3 (en)	2007-05-29
CN1279040C (zh)	2006-10-11
AP1965A (en)	2009-03-04
KR100548854B1 (ko)	2006-02-02
PA8517101A1 (es)	2002-10-24
BRPI0110955B8 (pt)	2021-05-25
DK1526134T3 (da)	2008-11-17
JP2003534343A (ja)	2003-11-18
AR028622A1 (es)	2003-05-14
EP1526134A3 (de)	2006-11-29
NO2020019I1 (no)	2020-06-30
BG65966B1 (bg)	2010-07-30
SI1284974T1 (en)	2004-08-31
HK1054927A1 (en)	2003-12-19
WO2001090106A2 (en)	2001-11-29
RS20090438A (en)	2010-05-07
RS51436B (en)	2011-04-30
NZ521477A (en)	2004-07-30
HRP20020938A2 (en)	2005-02-28
IS2511B (is)	2009-05-15
EA200401056A1 (ru)	2005-04-28
DE60102233T2 (de)	2005-01-27
TWI230160B (en)	2005-04-01
CA2408909C (en)	2006-06-27
EE05110B1 (et)	2008-12-15
DE60102233D1 (de)	2004-04-08
JP2005194283A (ja)	2005-07-21
DZ3464A1 (de)	2001-11-29
NO20025227D0 (no)	2002-10-31
EA007580B1 (ru)	2006-12-29

Publication	Publication Date	Title
EG24137A (en)	2008-08-06	Tropane derivatives useful in therapy
GB0016787D0 (en)	2000-08-30	Compounds useful in therapy
AP2004003147A0 (en)	2004-09-30	Tropane derivatives useful in therapy
GB9912411D0 (en)	1999-07-28	Compounds useful in therapy
IL151919A0 (en)	2003-04-10	Imidazopyridine derivatives and triazolpyrimidine derivatives
GB9912413D0 (en)	1999-07-28	Compounds useful in therapy
PT1296974E (pt)	2009-11-03	Derivados 2-cianopirrolidina e sua utilização como medicamentos
EP1296698A4 (de)	2005-02-16	Therapeutische verbindungen
GB0009606D0 (en)	2000-06-07	Therapeutic combinations
GB0004167D0 (en)	2000-04-12	1-piperidinyl-propan-2-ol derivatives and their use as therapeutic agents
GB9912410D0 (en)	1999-07-28	Compounds useful in therapy
PL363048A1 (en)	2004-11-15	Azabicyclic derivatives and their therapeutic use
GB9912415D0 (en)	1999-07-28	Compounds useful in therapy
GB9912416D0 (en)	1999-07-28	Compounds useful in therapy
SI1330453T1 (sl)	2006-08-31	Derivati indolilpiperidina kot antihistaminicna in antialergijska sredstva
GB0014046D0 (en)	2000-08-02	Compounds useful in therapy
GB9906130D0 (en)	1999-05-12	Compounds for use in therapy
GB0208071D0 (en)	2002-05-22	Tropane derivatives useful in therapy
GB0014866D0 (en)	2000-08-09	Compounds useful in therapy
GB0015835D0 (en)	2000-08-23	Compounds useful in therapy
GB9921314D0 (en)	1999-11-10	Compounds useful in therapy
GB9910765D0 (en)	1999-07-07	Compounds useful in therapy
GB9910772D0 (en)	1999-07-07	Compounds useful in therapy
GB9910769D0 (en)	1999-07-07	Compounds useful in therapy
GB9910767D0 (en)	1999-07-07	Compounds useful in therapy