EE04748B1 - Bitsüklilised heterotsüklilised ühendid, neid ühendeid sisaldavad ravimid, nende kasutamine ja meetodid nende valmistamiseks - Google Patents

Bitsüklilised heterotsüklilised ühendid, neid ühendeid sisaldavad ravimid, nende kasutamine ja meetodid nende valmistamiseks

Info

Publication number: EE04748B1
Authority: EE; Estonia
Prior art keywords: compounds; preparation; methods; bicyclic heterocyclic; drugs containing
Prior art date: 1999-06-21

Application number

EEP200100695A

Other languages

English (en)

Estonian (et)

Inventor

Himmelsbach Frank

Langkopf Elke

Metz Thomas

Solca Flavio

Jung Birgit

Baum Anke

Original Assignee

Boehringer Ingelheim Pharma Kg

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-06-21

Filing date

2000-06-16

Publication date

2006-12-15

1999-06-21 Priority claimed from DE1999128281 external-priority patent/DE19928281A1/de

2000-05-11 Priority claimed from DE2000123085 external-priority patent/DE10023085A1/de

2000-06-16 Application filed by Boehringer Ingelheim Pharma Kg filed Critical Boehringer Ingelheim Pharma Kg

2003-02-17 Publication of EE200100695A publication Critical patent/EE200100695A/xx

2006-12-15 Publication of EE04748B1 publication Critical patent/EE04748B1/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
- C07D239/72—Quinazolines; Hydrogenated quinazolines
- C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
- C07D239/94—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Gastroenterology & Hepatology (AREA)
Pulmonology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

EEP200100695A 1999-06-21 2000-06-16 Bitsüklilised heterotsüklilised ühendid, neid ühendeid sisaldavad ravimid, nende kasutamine ja meetodid nende valmistamiseks EE04748B1 (et)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
DE1999128281 DE19928281A1 (de)	1999-06-21	1999-06-21	Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
US14664499P	1999-07-30	1999-07-30
DE2000123085 DE10023085A1 (de)	2000-05-11	2000-05-11	Bicyclische Heterocyclen, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung
PCT/EP2000/005547 WO2000078735A1 (de)	1999-06-21	2000-06-16	Bicyclische heterocyclen, diese verbindungen enthaltende arzneimittel, deren verwendung und verfahren zu ihrer herstellung

Publications (2)

Publication Number	Publication Date
EE200100695A EE200100695A (et)	2003-02-17
EE04748B1 true EE04748B1 (et)	2006-12-15

Family

ID=27213849

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200100695A EE04748B1 (et)	1999-06-21	2000-06-16	Bitsüklilised heterotsüklilised ühendid, neid ühendeid sisaldavad ravimid, nende kasutamine ja meetodid nende valmistamiseks

Country Status (26)

Country	Link
US (4)	US7220750B2 (pt)
EP (2)	EP1194418A1 (pt)
JP (1)	JP3686610B2 (pt)
KR (1)	KR100709909B1 (pt)
CN (1)	CN1166645C (pt)
AU (1)	AU775285B2 (pt)
BG (1)	BG65890B1 (pt)
CA (1)	CA2375259C (pt)
CZ (1)	CZ302365B6 (pt)
DK (1)	DK1731511T3 (pt)
EA (1)	EA004981B1 (pt)
EE (1)	EE04748B1 (pt)
ES (1)	ES2552813T3 (pt)
HK (1)	HK1044769B (pt)
HU (1)	HUP0201900A3 (pt)
IL (2)	IL147133A0 (pt)
ME (1)	MEP45508A (pt)
MX (1)	MXPA01012899A (pt)
NO (1)	NO322094B1 (pt)
NZ (1)	NZ516633A (pt)
PT (1)	PT1731511E (pt)
SK (1)	SK287010B6 (pt)
TR (1)	TR200103692T2 (pt)
UA (1)	UA71976C2 (pt)
WO (1)	WO2000078735A1 (pt)
YU (1)	YU90901A (pt)

Families Citing this family (101)

* Cited by examiner, † Cited by third party
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JP4703183B2 (ja)	2002-07-15	2011-06-15	シンフォニーエボルーション，インク．	受容体型キナーゼモジュレーターおよびその使用方法
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2000
- 2000-06-16 MX MXPA01012899A patent/MXPA01012899A/es active IP Right Grant
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- 2000-06-16 JP JP2001504901A patent/JP3686610B2/ja not_active Expired - Lifetime
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- 2000-06-16 EP EP00936888A patent/EP1194418A1/de not_active Ceased
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- 2000-06-16 KR KR1020017016457A patent/KR100709909B1/ko active Protection Beyond IP Right Term
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- 2000-06-16 WO PCT/EP2000/005547 patent/WO2000078735A1/de active IP Right Grant
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- 2001-12-10 US US10/016,280 patent/US7220750B2/en not_active Expired - Lifetime
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2002
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2007
- 2007-04-12 US US11/734,350 patent/US20070185091A1/en not_active Abandoned
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Publication number	Publication date
PT1731511E (pt)	2015-11-13
NZ516633A (en)	2004-09-24
NO322094B1 (no)	2006-08-14
IL147133A (en)	2006-09-05
SK18452001A3 (sk)	2002-04-04
EP1194418A1 (de)	2002-04-10
EP1731511B1 (de)	2015-08-12
CA2375259C (en)	2009-04-28
HK1044769A1 (en)	2002-11-01
DK1731511T3 (en)	2015-10-26
HUP0201900A2 (hu)	2002-12-28
NO20016185D0 (no)	2001-12-18
CA2375259A1 (en)	2000-12-28
KR100709909B1 (ko)	2007-04-24
CN1356990A (zh)	2002-07-03
JP3686610B2 (ja)	2005-08-24
US20120329778A1 (en)	2012-12-27
US8722694B2 (en)	2014-05-13
IL147133A0 (en)	2002-08-14
US20070185091A1 (en)	2007-08-09
BG65890B1 (bg)	2010-04-30
EA004981B1 (ru)	2004-10-28
EA200200008A1 (ru)	2002-06-27
JP2003502410A (ja)	2003-01-21
EP1731511A1 (de)	2006-12-13
UA71976C2 (en)	2005-01-17
CZ20014497A3 (cs)	2002-03-13
ES2552813T3 (es)	2015-12-02
AU775285B2 (en)	2004-07-29
SK287010B6 (sk)	2009-09-07
US7220750B2 (en)	2007-05-22
TR200103692T2 (tr)	2002-10-21
US20100069414A1 (en)	2010-03-18
YU90901A (sh)	2004-07-15
KR20020012290A (ko)	2002-02-15
BG106189A (bg)	2002-08-30
CZ302365B6 (cs)	2011-04-13
AU5221400A (en)	2001-01-09
MXPA01012899A (es)	2002-07-30
US20020169180A1 (en)	2002-11-14
MEP45508A (en)	2011-02-10
EE200100695A (et)	2003-02-17
NO20016185L (no)	2001-12-18
HK1044769B (zh)	2005-02-25
WO2000078735A1 (de)	2000-12-28
HUP0201900A3 (en)	2003-02-28
CN1166645C (zh)	2004-09-15

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NO20011216L (no)	2001-05-09	Azetidinderivater, deres fremstilling og medikamenter inneholdende forbindelsene
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EE200200041A (et)	2003-04-15	Karboksüülhappeamiidid, neid ühendeid sisaldavad ravimid, nende kasutamine ja valmistamine
EE200300167A (et)	2003-08-15	Amidoalküülpiperidiini ja -piperasiini derivaadid, neid sisaldav farmatseutiline kompositsioon ningühendite kasutamine närvisüsteemi häirete raviks
IL146104A0 (en)	2002-07-25	Substituted bicyclic heterocyclic compounds, processes for their preparation and pharmaceutical compositions containing the same
EE200100027A (et)	2002-06-17	Fosfororgaanilised ühendid, neid sisaldav farmatseutiline preparaat ja nende kasutamine
EE05004B1 (et)	2008-04-15	Aminotiasooli derivaadid, nende valmistamine ja neid sisaldavad farmatseutilised kompositsioonid
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