DK164684A - 4-substituerede-2-azetidinon-forbindelser, fremgangsmaade til fremstilling heraf og mellemprodukter til brug herved - Google Patents

4-substituerede-2-azetidinon-forbindelser, fremgangsmaade til fremstilling heraf og mellemprodukter til brug herved Download PDF

Info

Publication number: DK164684A
Authority: DK; Denmark
Prior art keywords: slaughter; stalling; pigs; stalling pigs
Prior art date: 1983-03-25

Application number

DK164684A

Other languages

English (en)

Other versions

DK164684D0 (da

Inventor

Toshinari Tamura

Hidenori Iwamoto

Makoto Yoshida

Minoru Yamamoto

Original Assignee

Yamanouchi Pharma Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-03-25

Filing date

1984-03-23

Publication date

1984-09-26

1983-03-25 Priority claimed from JP58048989A external-priority patent/JPS59225182A/ja

1983-11-25 Priority claimed from JP58221470A external-priority patent/JPS60115578A/ja

1983-11-25 Priority claimed from JP58221469A external-priority patent/JPS60115577A/ja

1984-03-23 Application filed by Yamanouchi Pharma Co Ltd filed Critical Yamanouchi Pharma Co Ltd

1984-03-23 Publication of DK164684D0 publication Critical patent/DK164684D0/da

1984-09-26 Publication of DK164684A publication Critical patent/DK164684A/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
- C07K5/06147—Dipeptides with the first amino acid being heterocyclic and His-amino acid; Derivatives thereof

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Genetics & Genomics (AREA)
Biochemistry (AREA)
Biophysics (AREA)
General Health & Medical Sciences (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)

DK164684A 1983-03-25 1984-03-23 4-substituerede-2-azetidinon-forbindelser, fremgangsmaade til fremstilling heraf og mellemprodukter til brug herved DK164684A (da)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP58048989A JPS59225182A (ja)	1983-03-25	1983-03-25	２−アゼチジノン−４−カルボン酸の誘導体
JP58221470A JPS60115578A (ja)	1983-11-25	1983-11-25	２−アゼチジノン−４−置換化合物
JP58221469A JPS60115577A (ja)	1983-11-25	1983-11-25	２−アゼチジノン−４−置換体

Publications (2)

Publication Number	Publication Date
DK164684D0 DK164684D0 (da)	1984-03-23
DK164684A true DK164684A (da)	1984-09-26

Family

ID=27293483

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK164684A DK164684A (da)	1983-03-25	1984-03-23	4-substituerede-2-azetidinon-forbindelser, fremgangsmaade til fremstilling heraf og mellemprodukter til brug herved

Country Status (8)

Country	Link
US (3)	US4564609A (da)
EP (1)	EP0123444B1 (da)
KR (3)	KR870000357B1 (da)
CA (1)	CA1256650A (da)
DE (1)	DE3476399D1 (da)
DK (1)	DK164684A (da)
ES (4)	ES530960A0 (da)
NO (1)	NO158740C (da)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4719207A (en) *	1984-06-25	1988-01-12	Yamanouchi Pharmaceutical Co., Ltd.	CNS active substituted azetidinone compounds
JPS6253994A (ja)	1985-05-09	1987-03-09	Yamanouchi Pharmaceut Co Ltd	１−置換シリル−４−オキソ−２−アゼチジンカルボン酸低級アルキルエステル
ZA868957B (en) *	1985-12-06	1987-07-29	Yamanouchi Pharma Co Ltd	Crystals of nalpha-(((s)-4-oxo-2-azetidinyl)carbonyl)-l-histidyl-l-prolinamide and process for producing the crystals
US5686420A (en) *	1987-06-05	1997-11-11	Georgetown University	Thyrotropin-releasing hormone analogs and method of use
US5151497A (en) *	1989-02-21	1992-09-29	Japan Tobacco Inc.	Histidyl peptide derivatives
DK437289D0 (da) *	1989-09-04	1989-09-04	Hans Bundgaard	Prodrug derivatives of thyrotropin-releasing hormone (trh)
IT1249728B (it) *	1991-11-06	1995-03-09	Sigma Tau Ind Farmaceuti	Derivati delle prolinammide quali attivatori della memoria e dei processi di apprendimento e composizioni farmaceutiche che li contengono
CA2288986A1 (en) *	1997-05-09	1998-11-12	Smithkline Beecham Corporation	Beta-lactam inhibitors of coa-it
US20020151502A1 (en) *	1997-10-09	2002-10-17	Albert Sattin	Tri-peptides for neurological and neurobehavior applications
US7202279B1 (en) *	1998-02-11	2007-04-10	Georgetown University	Cyclic dipeptides and azetidinone compounds and their use in treating CNS injury and neurodegenerative disorders
WO2002004016A1 (fr) *	2000-07-11	2002-01-17	Shionogi & Co., Ltd.	Preparations enteriques contenant des peptides physiologiquement actifs
JP4817281B2 (ja)	2000-08-31	2011-11-16	塩野義製薬株式会社	パーキンソン病治療剤
US6982251B2 (en) *	2000-12-20	2006-01-03	Schering Corporation	Substituted 2-azetidinones useful as hypocholesterolemic agents
US20060287254A1 (en) *	2001-01-26	2006-12-21	Schering Corporation	Use of substituted azetidinone compounds for the treatment of sitosterolemia
NZ545332A (en) *	2001-01-26	2007-09-28	Schering Corp	Combinations of sterol absorption inhibitor(s) with cardiovascular agent(s) for the treatment of vascular conditions
US20030053981A1 (en) *	2001-01-26	2003-03-20	Schering Corporation	Combinations of bile acid sequestrant(s) and sterol absorption inhibitor(s) and treatments for vascular indications
SK9502003A3 (en) *	2001-01-26	2003-12-02	Schering Corp	Combinations of sterol absorption inhibitor(s) with blood modifier(s) for treating vascular conditions
AR034204A1 (es) *	2001-01-26	2004-02-04	Schering Corp	Composiciones y combinaciones de acido nicotinico y derivados del mismo con inhibidor(es) de la absorcion de los esteroles, y el uso de los mismos para preparar medicamentos para el tratamiento para indicaciones vasculares
WO2002058732A2 (en) *	2001-01-26	2002-08-01	Schering Corporation	Combinations of peroxisome proliferator-activated receptor (ppar) activator(s) and sterol absorption inhibitor(s) and treatments for vascular indications
RS50406B (sr) *	2001-01-26	2009-12-31	Schering Corporation,	Upotreba supstituisanih jedinjenja azetidinona za lečenje sitosterolemije
US7071181B2 (en) *	2001-01-26	2006-07-04	Schering Corporation	Methods and therapeutic combinations for the treatment of diabetes using sterol absorption inhibitors
US20030013699A1 (en) *	2001-05-25	2003-01-16	Davis Harry R.	Methods for treating alzheimer's disease and/or regulating levels of amyloid beta peptides in a subject
US7053080B2 (en) *	2001-09-21	2006-05-30	Schering Corporation	Methods and therapeutic combinations for the treatment of obesity using sterol absorption inhibitors
DE60216300T2 (de) *	2001-09-21	2007-06-28	Schering Corp.	Behandlung von xanthom mittels azetidinon-derivate als hemmer der sterol absorption
PT1427409E (pt) *	2001-09-21	2008-11-27	Schering Corp	Métodos para tratar ou para impedir a inflamação vascular utilizando inibidor(es) de absorção de esteróis
US7056906B2 (en) *	2001-09-21	2006-06-06	Schering Corporation	Combinations of hormone replacement therapy composition(s) and sterol absorption inhibitor(s) and treatments for vascular conditions in post-menopausal women
US20030119808A1 (en) *	2001-09-21	2003-06-26	Schering Corporation	Methods of treating or preventing cardiovascular conditions while preventing or minimizing muscular degeneration side effects
AU2003291719A1 (en) *	2002-11-06	2004-06-03	Schering Corporation	Cholesterol absorptions inhibitors for the treatment of autoimmune disorders
JP4589919B2 (ja) *	2003-03-07	2010-12-01	シェーリングコーポレイション	高コレステロール血症の処置のための、置換アゼチジノン化合物、これらの処方物および使用
WO2004081002A1 (en) *	2003-03-07	2004-09-23	Schering Corporation	Substituted azetidinone compounds, formulations and uses thereof for the treatment of hypercholesterolemia
JP2006519869A (ja) *	2003-03-07	2006-08-31	シェーリング　コーポレイション	置換アゼチジノン化合物、置換アゼチジノン化合物を調製するためのプロセス、それらの処方物および使用
US7459442B2 (en) *	2003-03-07	2008-12-02	Schering Corporation	Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
JP2007510659A (ja) *	2003-11-05	2007-04-26	シェーリング　コーポレイション	脂質調節剤および置換アゼチジノンの組み合わせならびに血管状態の処置
US7462595B2 (en) *	2004-09-17	2008-12-09	Prange Jr Arthur Jergen	Methods for treating cancer-related fatigue
KR101137503B1 (ko) *	2009-07-14	2012-04-20	웰이앤씨 주식회사	고분자 고체 지지체를 이용한 히스티딜-프롤린아미드 유도체의 제조 방법
NZ629709A (en)	2013-08-16	2018-04-27	Univ Maine System	Compounds and methods for improving plant performance

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3959248A (en) *	1974-04-03	1976-05-25	Merck & Co., Inc.	Analogs of thyrotropin-releasing hormone
GB1523598A (en) *	1975-03-08	1978-09-06	Reckitt & Colmann Prod Ltd	Tripeptides
US4271164A (en) *	1979-04-16	1981-06-02	Warner-Lambert Company	6-Substituted-arylpyrido[2,3-d]pyrimidin-7-amines and derivatives
HU180926B (en) *	1979-06-28	1983-05-30	Richter Gedeon Vegyeszet	Process for preparing trh analogues,tripeptide amides infectives on the central nerve sysrhem
US4328134A (en) *	1980-05-06	1982-05-04	Schally Andrew Victor	Anorexigenic peptides
US4426378A (en) *	1981-04-09	1984-01-17	The United States Of America As Represented By The Secretary Of The Army	Thyrotropin releasing hormone in therapy of shock and as a central nervous system stimulant

1984
- 1984-03-15 CA CA000449641A patent/CA1256650A/en not_active Expired
- 1984-03-23 KR KR1019840001506A patent/KR870000357B1/ko not_active IP Right Cessation
- 1984-03-23 DK DK164684A patent/DK164684A/da not_active Application Discontinuation
- 1984-03-23 NO NO841158A patent/NO158740C/no unknown
- 1984-03-23 ES ES530960A patent/ES530960A0/es active Granted
- 1984-03-23 US US06/592,866 patent/US4564609A/en not_active Expired - Fee Related
- 1984-03-26 DE DE8484302016T patent/DE3476399D1/de not_active Expired
- 1984-03-26 EP EP84302016A patent/EP0123444B1/en not_active Expired
1985
- 1985-06-14 ES ES544235A patent/ES8604208A1/es not_active Expired
- 1985-06-14 ES ES544236A patent/ES8604136A1/es not_active Expired
- 1985-06-14 ES ES85544234A patent/ES8604209A1/es not_active Expired
- 1985-10-07 US US06/785,169 patent/US4636567A/en not_active Expired - Fee Related
- 1985-10-07 US US06/785,168 patent/US4610821A/en not_active Expired - Fee Related
1987
- 1987-01-20 KR KR1019870000408A patent/KR890002104B1/ko not_active IP Right Cessation
- 1987-01-20 KR KR1019870000409A patent/KR890002105B1/ko not_active IP Right Cessation

Also Published As

Publication number	Publication date
NO158740B (no)	1988-07-18
ES8604208A1 (es)	1986-01-16
ES544235A0 (es)	1986-01-16
US4610821A (en)	1986-09-09
ES8604209A1 (es)	1986-01-16
KR840008021A (ko)	1984-12-12
NO841158L (no)	1984-09-26
US4636567A (en)	1987-01-13
ES544236A0 (es)	1986-01-16
KR880009549A (ko)	1988-09-15
EP0123444A1 (en)	1984-10-31
CA1256650A (en)	1989-06-27
EP0123444B1 (en)	1989-01-25
NO158740C (no)	1988-10-26
US4564609A (en)	1986-01-14
ES8604136A1 (es)	1986-01-16
DK164684D0 (da)	1984-03-23
KR880009550A (ko)	1988-09-15
DE3476399D1 (en)	1989-03-02
KR870000357B1 (ko)	1987-03-05
ES544234A0 (es)	1986-01-16
KR890002105B1 (ko)	1989-06-19
ES8600279A1 (es)	1985-10-01
KR890002104B1 (ko)	1989-06-19
ES530960A0 (es)	1985-10-01

Publication	Publication Date	Title
DK164684A (da)	1984-09-26	4-substituerede-2-azetidinon-forbindelser, fremgangsmaade til fremstilling heraf og mellemprodukter til brug herved
GB2138926B (en)	1986-07-09	Muzzle reference system
ZA845680B (en)	1985-03-27	Wear-parts system
GB8422613D0 (en)	1984-10-10	Conveyor system
DE3480054D1 (en)	1989-11-16	Pump-actuated sequencing system
GB2143667B (en)	1987-02-11	Instruction system topic-interpreting method
GB8304384D0 (en)	1983-03-23	Photobleach system
GB8402153D0 (en)	1984-02-29	Conveyor system
GB2137718B (en)	1986-07-02	Flow-stopping system
GB2169809B (en)	1987-06-10	Combined insufflation-irrigation system for an endoscope
GB2140366B (en)	1986-06-04	Side-support system for crawler-driven units
ZA852292B (en)	1985-11-27	Apparatus for decapitating fish
GB2152004B (en)	1988-04-20	Conveyor system
GB2143886B (en)	1986-11-19	Formwok system
GB8314968D0 (en)	1983-07-06	Apparatus for slaughtering animals
GB8315232D0 (en)	1983-07-06	Conveyor system
GB8423721D0 (en)	1984-10-24	Anti-icing system
IE820194L (en)	1982-08-06	Rearing unit for pigs
EP0138701A3 (en)	1985-06-19	Goniostelemeter system
CS337083A1 (en)	1985-08-31	Vyfukovy system turbodmychadlem preplnovaneho spalovaciho motoru
GB2140647B (en)	1986-05-08	3d-television system
DE3563298D1 (en)	1988-07-21	Storage system for carcasses
PL236859A1 (en)	1983-12-19	Swine slaughtering method
GB8413444D0 (en)	1984-07-04	Conveyor system
GB8329609D0 (en)	1983-12-07	Cattle flooring system

Legal Events

Date	Code	Title	Description
1993-11-15	AHS	Application shelved for other reasons than non-payment