DK145610C - 3-oximer af 17alfa-ethynyl-19-nortestosteronestere til anvendelse til undertrykkelse af fertilitet - Google Patents

3-oximer af 17alfa-ethynyl-19-nortestosteronestere til anvendelse til undertrykkelse af fertilitet

Info

Publication number: DK145610C
Authority: DK; Denmark
Prior art keywords: nortestoster; 17alfa; oximes; fertility; ethynyl
Prior art date: 1975-07-24

Application number

DK335876A

Other languages

English (en)

Other versions

DK335876A (da

DK145610B (da

Inventor

Arvin Pranlal Shroff

Original Assignee

Ortho Pharma Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1975-07-24

Filing date

1976-07-23

Publication date

1983-08-01

1976-07-23 Application filed by Ortho Pharma Corp filed Critical Ortho Pharma Corp

1977-01-25 Publication of DK335876A publication Critical patent/DK335876A/da

1982-12-27 Publication of DK145610B publication Critical patent/DK145610B/da

1983-08-01 Application granted granted Critical

1983-08-01 Publication of DK145610C publication Critical patent/DK145610C/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0005—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring the nitrogen atom being directly linked to the cyclopenta(a)hydro phenanthrene skeleton
- C07J41/0016—Oximes
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Reproductive Health (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Endocrinology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyridine Compounds (AREA)
Fertilizers (AREA)

DK335876A 1975-07-24 1976-07-23 3-oximer af 17alfa-ethynyl-19-nortestosteronestere til anvendelse til undertrykkelse af fertilitet DK145610C (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US59896675A	1975-07-24	1975-07-24
US59896675		1975-07-24
US05/652,000 US4027019A (en)	1975-07-24	1976-01-23	3-Oximes of D-17α-ethynyl-19-nortestosterone esters and method
US65200076		1976-01-23

Publications (3)

Publication Number	Publication Date
DK335876A DK335876A (da)	1977-01-25
DK145610B DK145610B (da)	1982-12-27
DK145610C true DK145610C (da)	1983-08-01

Family

ID=27083202

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK335876A DK145610C (da)	1975-07-24	1976-07-23	3-oximer af 17alfa-ethynyl-19-nortestosteronestere til anvendelse til undertrykkelse af fertilitet

Country Status (22)

Country	Link
US (1)	US4027019A (da)
JP (1)	JPS5214760A (da)
AT (1)	AT350748B (da)
AU (1)	AU501808B2 (da)
CA (1)	CA1072948A (da)
CH (1)	CH599249A5 (da)
DE (2)	DE2633210C2 (da)
DK (1)	DK145610C (da)
ES (1)	ES450108A1 (da)
FI (1)	FI55036C (da)
FR (1)	FR2318645A1 (da)
GB (1)	GB1557197A (da)
IE (1)	IE43581B1 (da)
IL (1)	IL50103A (da)
MX (1)	MX3417E (da)
NL (1)	NL192206C (da)
NO (1)	NO143350C (da)
NZ (1)	NZ181130A (da)
PH (1)	PH12003A (da)
PT (1)	PT65402B (da)
SE (2)	SE421800B (da)
YU (1)	YU39968B (da)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4507290A (en) *	1981-04-07	1985-03-26	World Health Organization	Esters of 17 α-ethynyl 19-nor-testosterone and 17 α-ethynyl-18-homo-19-nor-testosterone and pharmaceutical compositions containing the same
GB8313921D0 (en) *	1983-05-19	1983-06-22	World Health Org	Contraceptive compositions
WO1993013122A1 (de) *	1991-12-22	1993-07-08	Schering Aktiengesellschaft	3-methylsulfonylhydrazono- und 3-oxyimino-steroide, ein verfahren zu deren herstellung, diese steroide enthaltende pharmazeutische präparate sowie ihre verwendung zur herstellung von arzneimitteln
US7989436B2 (en)	2003-07-23	2011-08-02	Duramed Pharmaceuticals, Inc.	Estrogenic compounds and pharmaceutical formulations comprising the same
US6855703B1 (en)	2000-03-10	2005-02-15	Endeavor Pharmaceuticals	Pharmaceutical compositions of conjugated estrogens and methods of analyzing mixtures containing estrogenic compounds
US7459445B2 (en) *	2000-03-10	2008-12-02	Duramed Pharmaceuticals, Inc.	Estrogenic compounds and topical pharmaceutical formulations of the same
US6660726B2 (en)	2000-03-10	2003-12-09	Endeavor Pharmaceuticals	Estrogenic compounds, pharmaceutical compositions thereof, and methods of using same
US20050143360A1 (en) *	2001-02-02	2005-06-30	Joel Krasnow	Method of using a cyclooxygenase-2 inhibitor and sex steroids as a combination therapy for the treatment and prevention of dismenorrhea
US6992075B2 (en) *	2003-04-04	2006-01-31	Barr Laboratories, Inc.	C(14) estrogenic compounds
MXPA05010871A (es) *	2003-04-11	2005-11-25	Barr Lab Inc	Metodos para administrar estrogenos y progestinas.
AR039733A1 (es) *	2003-06-25	2005-03-09	Gador Sa	Proceso para la obtencion de norelgestromin en distintas relaciones de los isomeros e y z
HUP0301981A2 (hu) *	2003-06-30	2005-04-28	Richter Gedeon Vegyészeti Gyár Rt.	Tiszta d-(17alfa)-13-etil-17-hidroxi-18,19-dinor-pregn-4-én-20-in-3-on-3E- és 3Z-oxim izomerek, valamint eljárás az izomer keverékek és a tiszta izomerek előállítására
US7816546B2 (en) *	2003-06-30	2010-10-19	Richter Gedeon Vegyeszeti Gyar Rt.	Process for the synthesis of high purity d-(17α)-13-ethyl-17-hydroxy-18,19-dinorpregn-4-ene-20-yn-3-one-oxime
HUP0301982A2 (hu) *	2003-06-30	2005-04-28	Richter Gedeon Vegyészeti Gyár Rt.	Eljárás nagy tisztaságú d-(17alfa)-13-etil-17-hidroxi-18,19-dinor-pregn-4-én-20-in-3-on-oxim előállítására
EP1778716A1 (en) *	2004-08-12	2007-05-02	Sicor Inc.	Process for the preparation of 3-oximino steroids
EP1853272A1 (en) *	2005-02-03	2007-11-14	Duramed Pharmaceuticals, Inc.	Compositions of unconjugated estrogens and methods for their use

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1493161B2 (de) *	1951-01-28	1973-08-30		17alpha-aethinyl-18-methyl-19nortestosteronester, verfahren zu ihrer herstellung und diese enthaltendes mittel
US3780073A (en) *	1966-07-06	1973-12-18	Ortho Pharma Corp	3-oximes of 19-nortestosterone esters
US3532689A (en) *	1967-04-20	1970-10-06	Ortho Pharma Corp	3-oxime and 3-oxime esters of 19-nortestosterone
NL7306609A (da) *	1972-05-26	1973-11-28
US3912768A (en) *	1972-09-26	1975-10-14	Warner Lambert Co	Norethindrone O-alkyloximes

1976
- 1976-01-23 US US05/652,000 patent/US4027019A/en not_active Expired - Lifetime
- 1976-06-11 NZ NZ181130A patent/NZ181130A/en unknown
- 1976-06-14 PH PH18572A patent/PH12003A/en unknown
- 1976-06-14 FR FR7617973A patent/FR2318645A1/fr active Granted
- 1976-06-15 GB GB24769/76A patent/GB1557197A/en not_active Expired
- 1976-06-28 AU AU15357/76A patent/AU501808B2/en not_active Expired
- 1976-07-06 CA CA256,343A patent/CA1072948A/en not_active Expired
- 1976-07-13 YU YU1733/76A patent/YU39968B/xx unknown
- 1976-07-22 CH CH940376A patent/CH599249A5/xx not_active IP Right Cessation
- 1976-07-22 IL IL50103A patent/IL50103A/xx unknown
- 1976-07-22 JP JP51086661A patent/JPS5214760A/ja active Granted
- 1976-07-22 MX MX001792U patent/MX3417E/es unknown
- 1976-07-23 NL NL7608210A patent/NL192206C/nl not_active IP Right Cessation
- 1976-07-23 AT AT543976A patent/AT350748B/de not_active IP Right Cessation
- 1976-07-23 ES ES450108A patent/ES450108A1/es not_active Expired
- 1976-07-23 DE DE2633210A patent/DE2633210C2/de not_active Expired
- 1976-07-23 IE IE1636/76A patent/IE43581B1/en unknown
- 1976-07-23 SE SE7608407A patent/SE421800B/xx not_active IP Right Cessation
- 1976-07-23 FI FI762116A patent/FI55036C/fi not_active IP Right Cessation
- 1976-07-23 DK DK335876A patent/DK145610C/da not_active IP Right Cessation
- 1976-07-23 PT PT65402A patent/PT65402B/pt unknown
- 1976-07-23 NO NO762583A patent/NO143350C/no unknown
- 1976-07-23 DE DE2661002A patent/DE2661002C2/de not_active Expired
1979
- 1979-12-14 SE SE7910336A patent/SE445458B/sv not_active IP Right Cessation

Also Published As

Publication number	Publication date
IE43581B1 (en)	1981-04-08
PT65402A (en)	1976-08-01
FI55036C (fi)	1979-05-10
ES450108A1 (es)	1977-11-16
IE43581L (en)	1977-01-24
CA1072948A (en)	1980-03-04
SE7608407L (sv)	1977-01-25
NO143350C (no)	1981-01-28
DK335876A (da)	1977-01-25
DE2661002C2 (da)	1988-03-17
NL7608210A (nl)	1977-01-26
IL50103A0 (en)	1976-09-30
US4027019A (en)	1977-05-31
JPS5214760A (en)	1977-02-03
DE2633210A1 (de)	1977-02-17
DK145610B (da)	1982-12-27
PH12003A (en)	1978-10-06
IL50103A (en)	1979-11-30
CH599249A5 (da)	1978-05-31
AU1535776A (en)	1978-01-05
NZ181130A (en)	1984-07-06
NO762583L (da)	1977-01-25
SE445458B (sv)	1986-06-23
PT65402B (en)	1979-06-09
YU39968B (en)	1985-06-30
NL192206C (nl)	1997-03-04
DE2633210C2 (de)	1987-04-09
FI55036B (fi)	1979-01-31
NL192206B (nl)	1996-11-01
NO143350B (no)	1980-10-13
FR2318645A1 (fr)	1977-02-18
JPS624400B2 (da)	1987-01-30
YU173376A (en)	1982-08-31
SE7910336L (sv)	1979-12-14
DE2661002A1 (da)	1985-05-02
FR2318645B1 (da)	1978-11-17
SE421800B (sv)	1982-02-01
MX3417E (es)	1980-11-13
FI762116A (da)	1977-01-25
AT350748B (de)	1979-06-11
AU501808B2 (en)	1979-06-28
ATA543976A (de)	1978-11-15
GB1557197A (en)	1979-12-05

Publication	Publication Date	Title
DK153228C (da)	1988-11-07	Fremgangsmaade til afgummiering af triglyceridolier
DK49676A (da)	1976-08-13	Fremgangsmade til fremstilling af hypolipidemiske midler
DK143044C (da)	1981-10-19	Sprededybel af formstof
DK145610C (da)	1983-08-01	3-oximer af 17alfa-ethynyl-19-nortestosteronestere til anvendelse til undertrykkelse af fertilitet
DK339876A (da)	1977-02-01	Fremgangsmade til desoxygenering af sekundere alkoholer
DK145859C (da)	1983-10-03	Analogifremgangsmaade til fremstilling af estre af 3-hydroxy-5beta-oestran-17-on
DK107876A (da)	1976-09-15	Fremgangsmade til fremstilling af thiocarbamider
DK141458C (da)	1980-09-08	Sprededybel af formstof
DK535476A (da)	1977-05-29	Fremgangsmade til fremstilling af 7-methoxycephalosporiner
DK150676A (da)	1976-10-12	Fremgangsmade til fremstilling af krystallinsk natrium-o-formyl-cefamandol
DK438976A (da)	1977-04-17	Fremgangsmade til fremstilling af cyclohexylphenylderivater
DK399976A (da)	1977-03-05	Fremgangsmade til fremstilling af aralkylamider
DK415576A (da)	1977-04-02	Fremgangsmade til fremstilling af krystallinsk dipilocarpiniumpamoat
DK9876A (da)	1976-07-14	Fremgangsmade til ojeblikkelig indledning af skarring
DK366676A (da)	1977-02-15	Fremgangsmade til fremstilling af slagseje polyvinylaromater
DK526676A (da)	1977-05-25	Fremgangsmade til fremstilling af 4-chlor-2-butynyl-m-chlorcarbanilat
DK480676A (da)	1977-04-24	Fremgangsmade til fremstilling af s-alkylphosphordihalogeniddithioater
DK424676A (da)	1977-03-27	Fremgangsmade til fremstilling af 2-alkylindan
DK246976A (da)	1976-12-14	Fremgangsmade til fremstilling af isoquinoliner
DK46476A (da)	1976-08-14	Fremgangsmade til fremstilling af 5-nitrothiazolylimidazolidiner
TR19384A (tr)	1979-02-20	Sukros esterlerinin tasfiyesi
DK415376A (da)	1977-03-31	Fremgangsmade til fremstilling af acylcyanoguanidiner
DK537476A (da)	1977-06-02	Fremgangsmade til fremstilling af et eburnanpreparat
DK55476A (da)	1976-08-13	Fremgangsmade til fremstilling af dinitronaphthalener
DK238776A (da)	1976-12-03	Fremgangsmade til fremstilling af 3-brombenzaldehyd

Legal Events

Date	Code	Title	Description
1996-08-26	PUP	Patent expired