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CO6351783A2 - Derivados de indazoles sustituidos con fenilo o piridinilo - Google Patents

Derivados de indazoles sustituidos con fenilo o piridinilo

Info

Publication number
CO6351783A2
CO6351783A2 CO10137241A CO10137241A CO6351783A2 CO 6351783 A2 CO6351783 A2 CO 6351783A2 CO 10137241 A CO10137241 A CO 10137241A CO 10137241 A CO10137241 A CO 10137241A CO 6351783 A2 CO6351783 A2 CO 6351783A2
Authority
CO
Colombia
Prior art keywords
derivatives
indazols
piridinyl
phenyll
replaced
Prior art date
Application number
CO10137241A
Other languages
English (en)
Inventor
Markus Berger
Jan Dahmen
Hartmut Rehwinkel
Stinabritt Nilsson
Matti Lepisto
Henrik Johansson
Nafizal Hossain
Martin Hemmerling
Thomas Hansson
Karl Edman
Original Assignee
Astrazeneca Ab
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41340347&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO6351783(A2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab, Bayer Schering Pharma Ag filed Critical Astrazeneca Ab
Publication of CO6351783A2 publication Critical patent/CO6351783A2/es

Links

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    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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Abstract

Un compuesto de fórmula la:La presente invención se refiere a nuevos derivados de indazolilo, a composiciones farmacéuticas que comprenden tales derivados, a procesos para preparar dichos nuevos derivados y al uso de tales derivados como medicamentos.
CO10137241A 2008-05-20 2010-11-04 Derivados de indazoles sustituidos con fenilo o piridinilo CO6351783A2 (es)

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CO10137238A CO6331310A2 (es) 2008-05-20 2010-11-04 Derivados de indazol sustituidos con fenilo y benzodioxinilo

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PE20091925A1 (es) 2010-01-24
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DOP2010000359A (es) 2010-12-15
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ECSP10010619A (es) 2010-12-30
PT2291369E (pt) 2016-03-11
SV2010003738A (es) 2011-03-15
EP2291359A1 (en) 2011-03-09
EA201001682A1 (ru) 2011-06-30
CL2009001247A1 (es) 2010-07-23
DOP2010000357A (es) 2010-12-15
EA018629B1 (ru) 2013-09-30
MX2010012529A (es) 2011-03-29
KR101593253B1 (ko) 2016-02-11
CA2724508C (en) 2016-10-25
IL209121A0 (en) 2011-01-31
AU2009249874B2 (en) 2012-08-16
PA8827001A1 (es) 2009-12-16
CN102099355A (zh) 2011-06-15
NZ588994A (en) 2012-08-31
US20100080786A1 (en) 2010-04-01
UY31831A (es) 2010-01-05
CN102112449A (zh) 2011-06-29
JP2014185188A (ja) 2014-10-02
WO2009142571A1 (en) 2009-11-26
ME02455B (me) 2017-02-20
EA018629B8 (ru) 2013-12-30
CL2009001248A1 (es) 2010-06-11
PL2291369T3 (pl) 2016-04-29
AU2009249874A1 (en) 2009-11-26
IL209122A0 (en) 2011-01-31

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