BRPI0418135B8 - Processo para a preparação de triazolpirimidinas, bem como seu uso - Google Patents
Processo para a preparação de triazolpirimidinas, bem como seu usoInfo
- Publication number
- BRPI0418135B8 BRPI0418135B8 BRPI0418135A BRPI0418135A BRPI0418135B8 BR PI0418135 B8 BRPI0418135 B8 BR PI0418135B8 BR PI0418135 A BRPI0418135 A BR PI0418135A BR PI0418135 A BRPI0418135 A BR PI0418135A BR PI0418135 B8 BRPI0418135 B8 BR PI0418135B8
- Authority
- BR
- Brazil
- Prior art keywords
- triazolpyrimidines
- preparation
- well
- amino
- alkyloxycarbonyl
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 3
- AVXURJPOCDRRFD-UHFFFAOYSA-N Hydroxylamine Chemical class ON AVXURJPOCDRRFD-UHFFFAOYSA-N 0.000 abstract 1
- -1 alkyloxycarbonyl isothiocyanate Chemical class 0.000 abstract 1
- 125000005161 aryl oxy carbonyl group Chemical group 0.000 abstract 1
- 239000003960 organic solvent Substances 0.000 abstract 1
- LJXQPZWIHJMPQQ-UHFFFAOYSA-N pyrimidin-2-amine Chemical compound NC1=NC=CC=N1 LJXQPZWIHJMPQQ-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
"PROCESSO PARA A PREPARAÇÃO DE TRIAZOLPIRIMIDINAS". A presente invenção refere-se a um processo para a preparação de 2-amino-[1,2,4]triazolpirimidinas substituídas ou não-substituídas que compreende combinar A) 2-amino-pirimidina ou seus derivados com isotiocianato de alquiloxicarbonila ou isotiocianato de ariloxicarbonila com B) sal de hidroxil amônio e uma base em que a reação é realizada em um solvente orgânico aprótico polar na faixa de temperatura de 40 a 150<198>C.
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US53161303P | 2003-12-23 | 2003-12-23 | |
US60/531,613 | 2003-12-23 | ||
EP03029728.7 | 2003-12-23 | ||
EP03029728 | 2003-12-23 | ||
EP2005063753 | 2005-07-14 |
Publications (3)
Publication Number | Publication Date |
---|---|
BRPI0418135A BRPI0418135A (pt) | 2007-04-27 |
BRPI0418135B1 BRPI0418135B1 (pt) | 2014-05-27 |
BRPI0418135B8 true BRPI0418135B8 (pt) | 2022-06-28 |
Family
ID=34923924
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0418135A BRPI0418135B8 (pt) | 2003-12-23 | 2004-12-22 | Processo para a preparação de triazolpirimidinas, bem como seu uso |
Country Status (17)
Country | Link |
---|---|
US (1) | US7781582B2 (pt) |
EP (1) | EP1699794B1 (pt) |
JP (1) | JP4838146B2 (pt) |
KR (1) | KR101142649B1 (pt) |
CN (1) | CN1898245B (pt) |
AR (1) | AR046987A1 (pt) |
AT (1) | ATE382622T1 (pt) |
AU (1) | AU2004309056B2 (pt) |
BR (1) | BRPI0418135B8 (pt) |
CA (1) | CA2550874C (pt) |
DE (1) | DE602004011113T2 (pt) |
DK (1) | DK1699794T3 (pt) |
ES (1) | ES2295960T3 (pt) |
IL (1) | IL176471A (pt) |
PL (1) | PL1699794T3 (pt) |
WO (1) | WO2005063753A1 (pt) |
ZA (1) | ZA200605472B (pt) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
BR102012002852B1 (pt) * | 2011-02-09 | 2018-05-29 | Dow Agrosciences Llc | Composições pesticidas e processos relacionados das mesmas |
CN104768954B (zh) * | 2012-09-14 | 2017-11-17 | 美国陶氏益农公司 | 由4‑氨基‑2,5‑二甲氧基嘧啶制备2‑氨基‑5,8‑二甲氧基[1,2,4]三唑并[1,5‑c]嘧啶的改善方法 |
CN104910165A (zh) * | 2015-06-02 | 2015-09-16 | 安徽兴东化工有限公司 | 一种2-氨基-5,7-二甲氧基-三嗪并嘧啶的制备方法 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5571775A (en) * | 1994-07-11 | 1996-11-05 | Dowelanco | N-aryl[1,2,4]triazolo[1,5-a]pyridine-2-sulfonamide herbicides |
CN1159297C (zh) * | 1996-09-24 | 2004-07-28 | 道农业科学公司 | N-([1,2,4]三唑并吖嗪基)苯磺酰胺和吡啶磺酰胺化合物和它们作为除草剂的用途 |
SK286484B6 (sk) * | 2000-11-03 | 2008-11-06 | Dow Agrosciences Llc | N-(5,7-Dimetoxy[1,2,4]-triazol[1,5-a]pyrimidin-2-yl)arylsulfónamidové zlúčeniny, spôsob ich výrobya ich použitie |
-
2004
- 2004-12-22 DE DE602004011113T patent/DE602004011113T2/de active Active
- 2004-12-22 AT AT04804192T patent/ATE382622T1/de not_active IP Right Cessation
- 2004-12-22 ZA ZA200605472A patent/ZA200605472B/en unknown
- 2004-12-22 ES ES04804192T patent/ES2295960T3/es active Active
- 2004-12-22 DK DK04804192T patent/DK1699794T3/da active
- 2004-12-22 AU AU2004309056A patent/AU2004309056B2/en active Active
- 2004-12-22 JP JP2006546054A patent/JP4838146B2/ja active Active
- 2004-12-22 CA CA2550874A patent/CA2550874C/en active Active
- 2004-12-22 WO PCT/EP2004/014596 patent/WO2005063753A1/en active IP Right Grant
- 2004-12-22 US US10/584,720 patent/US7781582B2/en active Active
- 2004-12-22 BR BRPI0418135A patent/BRPI0418135B8/pt active IP Right Grant
- 2004-12-22 KR KR1020067012499A patent/KR101142649B1/ko active IP Right Grant
- 2004-12-22 AR ARP040104853A patent/AR046987A1/es active IP Right Grant
- 2004-12-22 CN CN200480038604XA patent/CN1898245B/zh active Active
- 2004-12-22 PL PL04804192T patent/PL1699794T3/pl unknown
- 2004-12-22 EP EP04804192A patent/EP1699794B1/en active Active
-
2006
- 2006-06-21 IL IL176471A patent/IL176471A/en active IP Right Grant
Also Published As
Publication number | Publication date |
---|---|
BRPI0418135B1 (pt) | 2014-05-27 |
IL176471A (en) | 2011-08-31 |
EP1699794B1 (en) | 2008-01-02 |
KR101142649B1 (ko) | 2012-05-11 |
ATE382622T1 (de) | 2008-01-15 |
AU2004309056B2 (en) | 2009-11-19 |
JP2007515449A (ja) | 2007-06-14 |
CN1898245A (zh) | 2007-01-17 |
CA2550874A1 (en) | 2005-07-14 |
PL1699794T3 (pl) | 2008-06-30 |
AU2004309056A1 (en) | 2005-07-14 |
JP4838146B2 (ja) | 2011-12-14 |
US20070238873A1 (en) | 2007-10-11 |
KR20060110333A (ko) | 2006-10-24 |
CN1898245B (zh) | 2011-07-20 |
US7781582B2 (en) | 2010-08-24 |
ES2295960T3 (es) | 2008-04-16 |
AR046987A1 (es) | 2006-01-04 |
DE602004011113D1 (de) | 2008-02-14 |
EP1699794A1 (en) | 2006-09-13 |
DE602004011113T2 (de) | 2008-04-30 |
IL176471A0 (en) | 2006-10-05 |
ZA200605472B (en) | 2007-11-28 |
CA2550874C (en) | 2012-04-10 |
DK1699794T3 (da) | 2008-05-19 |
WO2005063753A1 (en) | 2005-07-14 |
BRPI0418135A (pt) | 2007-04-27 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B06F | Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette] | ||
B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
B09A | Decision: intention to grant [chapter 9.1 patent gazette] | ||
B16A | Patent or certificate of addition of invention granted [chapter 16.1 patent gazette] |
Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 22/12/2004, OBSERVADAS AS CONDICOES LEGAIS. |
|
B25D | Requested change of name of applicant approved |