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BRPI0312547B8 - uso de derivados de imidazo [4,5-c]piridina como inibidores virais - Google Patents

uso de derivados de imidazo [4,5-c]piridina como inibidores virais

Info

Publication number
BRPI0312547B8
BRPI0312547B8 BRPI0312547A BR0312547A BRPI0312547B8 BR PI0312547 B8 BRPI0312547 B8 BR PI0312547B8 BR PI0312547 A BRPI0312547 A BR PI0312547A BR 0312547 A BR0312547 A BR 0312547A BR PI0312547 B8 BRPI0312547 B8 BR PI0312547B8
Authority
BR
Brazil
Prior art keywords
imidazo
pyridine derivatives
viral inhibitors
virus
class
Prior art date
Application number
BRPI0312547A
Other languages
English (en)
Other versions
BR0312547A (pt
BRPI0312547B1 (pt
Inventor
De Clercq Erik
Pürstinger Gerhard
Neyts Johan
Original Assignee
Gerhard Puerstinger
Gilead Sciences Inc
K U Leuven Res & Development
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0313251A external-priority patent/GB0313251D0/en
Application filed by Gerhard Puerstinger, Gilead Sciences Inc, K U Leuven Res & Development filed Critical Gerhard Puerstinger
Publication of BR0312547A publication Critical patent/BR0312547A/pt
Publication of BRPI0312547B1 publication Critical patent/BRPI0312547B1/pt
Publication of BRPI0312547B8 publication Critical patent/BRPI0312547B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/20—Antivirals for DNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Investigating Or Analysing Biological Materials (AREA)

Abstract

inibidores virais. a presente invenção refere-se a uma composição farmacêutica para o tratamento ou prevenção de infecções virais compreendendo como um princípio ativo pelo menos um derivado de imidazo[4,5-c]piridina tendo a fórmula geral (z): a invenção também refere-se aos processos para a preparação de compostos de acordo com a invenção tendo a fórmula geral mencionada acima e seu uso como um medicamento ou para tratar ou prevenir infecções virais.
BRPI0312547A 2002-07-03 2003-07-03 uso de derivados de imidazo [4,5-c]piridina como inibidores virais BRPI0312547B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0215293.2A GB0215293D0 (en) 2002-07-03 2002-07-03 Viral inhibitors
GB0313251A GB0313251D0 (en) 2003-06-10 2003-06-10 Viral inhibitors
PCT/BE2003/000117 WO2004005286A2 (en) 2002-07-03 2003-07-03 Viral inhibitors

Publications (3)

Publication Number Publication Date
BR0312547A BR0312547A (pt) 2005-04-26
BRPI0312547B1 BRPI0312547B1 (pt) 2020-01-21
BRPI0312547B8 true BRPI0312547B8 (pt) 2021-05-25

Family

ID=30117086

Family Applications (2)

Application Number Title Priority Date Filing Date
BR122018077110-0A BR122018077110B1 (pt) 2002-07-03 2003-07-03 derivados de imidazo [4,5-c]piridina, seus compostos e respectivas composições farmacêuticas
BRPI0312547A BRPI0312547B8 (pt) 2002-07-03 2003-07-03 uso de derivados de imidazo [4,5-c]piridina como inibidores virais

Family Applications Before (1)

Application Number Title Priority Date Filing Date
BR122018077110-0A BR122018077110B1 (pt) 2002-07-03 2003-07-03 derivados de imidazo [4,5-c]piridina, seus compostos e respectivas composições farmacêuticas

Country Status (21)

Country Link
US (2) US7737162B2 (pt)
EP (2) EP1521754B1 (pt)
JP (2) JP4907082B2 (pt)
KR (2) KR101184032B1 (pt)
CN (1) CN1328279C (pt)
AT (1) ATE522528T1 (pt)
AU (2) AU2003243846B9 (pt)
BR (2) BR122018077110B1 (pt)
CA (1) CA2491243C (pt)
CY (1) CY1112042T1 (pt)
DK (1) DK1521754T3 (pt)
EA (1) EA013562B1 (pt)
ES (2) ES2372277T3 (pt)
GB (1) GB0215293D0 (pt)
IL (1) IL166055A (pt)
MX (1) MXPA04012965A (pt)
NO (1) NO330766B1 (pt)
NZ (1) NZ537473A (pt)
PT (2) PT1521754E (pt)
SI (1) SI1521754T1 (pt)
WO (1) WO2004005286A2 (pt)

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