BR9711842A - Derivatives of n- (benzothiazol-2-yl) piperidine-1-ethanamine its preparation and its application in therapeutics - Google Patents

Derivatives of n- (benzothiazol-2-yl) piperidine-1-ethanamine its preparation and its application in therapeutics

Info

Publication number: BR9711842A
Authority: BR; Brazil
Prior art keywords: ethanamine; benzothiazol; therapeutics; piperidine; derivatives
Prior art date: 1996-10-01

Application number

BR9711842A

Other languages

Portuguese (pt)

Inventor

Gihad Dargazanli

Pascal George

Patrick Lardenois

Jonathan Frost

Johannes Schoemaker

Maria-Carmen Renones

Pascale Magat

Original Assignee

Synthelabo

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-10-01

Filing date

1997-09-26

Publication date

1999-08-24

1997-09-26 Application filed by Synthelabo filed Critical Synthelabo

1999-08-24 Publication of BR9711842A publication Critical patent/BR9711842A/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Medicinal Chemistry (AREA)
Neurosurgery (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)

BR9711842A 1996-10-01 1997-09-26 Derivatives of n- (benzothiazol-2-yl) piperidine-1-ethanamine its preparation and its application in therapeutics BR9711842A (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR9611925A FR2753970B1 (en)	1996-10-01	1996-10-01	N- (BENZOTHIAZOL-2-YL) PIPERIDINE-1-ETHANAMINE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION
PCT/FR1997/001692 WO1998014444A1 (en)	1996-10-01	1997-09-26	N-(benzothiazol-2-yl) piperidine-1-ethanamine derivatives, their preparation and application in therapeutics

Publications (1)

Publication Number	Publication Date
BR9711842A true BR9711842A (en)	1999-08-24

Family

ID=9496217

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BR9711842A BR9711842A (en)	1996-10-01	1997-09-26	Derivatives of n- (benzothiazol-2-yl) piperidine-1-ethanamine its preparation and its application in therapeutics

Country Status (23)

Country	Link
EP (1)	EP0929550A1 (en)
JP (1)	JP2001501217A (en)
KR (1)	KR20000048767A (en)
CN (1)	CN1230959A (en)
AR (1)	AR009105A1 (en)
AU (1)	AU722147B2 (en)
BG (1)	BG103271A (en)
BR (1)	BR9711842A (en)
CA (1)	CA2266510A1 (en)
CO (1)	CO4650030A1 (en)
CZ (1)	CZ112699A3 (en)
EE (1)	EE9900135A (en)
FR (1)	FR2753970B1 (en)
HU (1)	HUP9904091A3 (en)
IL (1)	IL128902A (en)
NO (1)	NO991581L (en)
NZ (1)	NZ334553A (en)
PL (1)	PL332648A1 (en)
SK (1)	SK42299A3 (en)
TR (1)	TR199900634T2 (en)
TW (1)	TW438800B (en)
WO (1)	WO1998014444A1 (en)
ZA (1)	ZA978772B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9725541D0 (en) *	1997-12-02	1998-02-04	Pharmacia & Upjohn Spa	Amino-benzothiazole derivatives
US6107313A (en) *	1998-10-02	2000-08-22	Combichem, Inc.	Dopamine receptor antagonists
HUP0301315A3 (en) *	2000-06-21	2007-10-29	Hoffmann La Roche	Benzothiazole derivatives, process for their preparation, their use and pharmaceutical compositions containing them
US7087761B2 (en)	2003-01-07	2006-08-08	Hoffmann-La Roche Inc.	Cyclization process for substituted benzothiazole derivatives
WO2005040129A2 (en) *	2003-10-24	2005-05-06	F. Hoffmann-La Roche Ag	Ccr3 receptor antagonists
EA011279B1 (en)	2004-05-24	2009-02-27	Ф. Хоффманн-Ля Рош Аг	4-hydroxy-4-methyl-piperidine-1-carboxylic acid (4-methoxy-7-morpholin-4-yl-benzothiazol-2yl)-amide
DE602005008095D1 (en)	2004-11-05	2008-08-21	Hoffmann La Roche	PROCESS FOR THE PREPARATION OF ISONICOTINIC ACID DERIVATIVES
JP4801724B2 (en)	2005-03-23	2011-10-26	エフ．ホフマン−ラロシュアーゲー	Acetylenyl-pyrazolo-pyrimidine derivatives as mGluR2 antagonists
CN101273040B (en)	2005-09-27	2011-11-09	弗·哈夫曼-拉罗切有限公司	Oxadiazolyl pyrazolo-pyrimidines as MGLUR2 antagonists

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA1260474A (en) *	1984-12-03	1989-09-26	Raymond A. Stokbroekx	Benzoxazol- and benzothiazolamine derivatives
KR930005004B1 (en) *	1985-04-15	1993-06-11	쟈안센 파아마슈우티카 엔. 부이.	Process for preparing substituted n-\|(4-piperidinyl) alkyl¨ bicycle condensed oxazole and thiazolamines

1996
- 1996-10-01 FR FR9611925A patent/FR2753970B1/en not_active Expired - Fee Related
1997
- 1997-09-26 HU HU9904091A patent/HUP9904091A3/en unknown
- 1997-09-26 AU AU44638/97A patent/AU722147B2/en not_active Ceased
- 1997-09-26 PL PL97332648A patent/PL332648A1/en unknown
- 1997-09-26 JP JP10516272A patent/JP2001501217A/en active Pending
- 1997-09-26 IL IL12890297A patent/IL128902A/en not_active IP Right Cessation
- 1997-09-26 CA CA002266510A patent/CA2266510A1/en not_active Abandoned
- 1997-09-26 CZ CZ991126A patent/CZ112699A3/en unknown
- 1997-09-26 EP EP97943001A patent/EP0929550A1/en not_active Ceased
- 1997-09-26 BR BR9711842A patent/BR9711842A/en not_active Application Discontinuation
- 1997-09-26 KR KR1019990702753A patent/KR20000048767A/en not_active Application Discontinuation
- 1997-09-26 EE EEP199900135A patent/EE9900135A/en unknown
- 1997-09-26 CN CN97198112A patent/CN1230959A/en active Pending
- 1997-09-26 CO CO97056315A patent/CO4650030A1/en unknown
- 1997-09-26 TR TR1999/00634T patent/TR199900634T2/en unknown
- 1997-09-26 WO PCT/FR1997/001692 patent/WO1998014444A1/en not_active Application Discontinuation
- 1997-09-26 NZ NZ334553A patent/NZ334553A/en unknown
- 1997-09-26 SK SK422-99A patent/SK42299A3/en unknown
- 1997-09-30 TW TW086114229A patent/TW438800B/en active
- 1997-09-30 ZA ZA9708772A patent/ZA978772B/en unknown
- 1997-09-30 AR ARP970104493A patent/AR009105A1/en not_active Application Discontinuation
1999
- 1999-03-22 BG BG103271A patent/BG103271A/en unknown
- 1999-03-30 NO NO991581A patent/NO991581L/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
CN1230959A (en)	1999-10-06
HUP9904091A2 (en)	2000-05-28
AR009105A1 (en)	2000-03-08
SK42299A3 (en)	1999-12-10
CZ112699A3 (en)	1999-06-16
WO1998014444A1 (en)	1998-04-09
FR2753970B1 (en)	1998-10-30
NZ334553A (en)	2000-11-24
CA2266510A1 (en)	1998-04-09
IL128902A (en)	2001-07-24
KR20000048767A (en)	2000-07-25
BG103271A (en)	2000-05-31
NO991581L (en)	1999-06-01
TW438800B (en)	2001-06-07
HUP9904091A3 (en)	2000-07-28
JP2001501217A (en)	2001-01-30
AU722147B2 (en)	2000-07-20
PL332648A1 (en)	1999-09-27
CO4650030A1 (en)	1998-09-03
AU4463897A (en)	1998-04-24
IL128902A0 (en)	2000-02-17
ZA978772B (en)	1998-03-27
FR2753970A1 (en)	1998-04-03
TR199900634T2 (en)	1999-06-21
EE9900135A (en)	1999-12-15
NO991581D0 (en)	1999-03-30
EP0929550A1 (en)	1999-07-21

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Legal Events

Date	Code	Title	Description
2001-02-06	PC	Transfer	Free format text: SANOFI-SYNTHELABO (FR)
2006-12-19	B07A	Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
2007-11-06	B09B	Patent application refused [chapter 9.2 patent gazette]	Free format text: INDEFIRO O PRESENTE PEDIDO DE PATENTE, DE ACORDO COM ART. 36 DA LPI (LEI 9279/96).