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BR0009465A - Formulação farmacêutica na forma de uma cápsula par administração oral, uso de undecanoato de testosterona, e, método de tratamento compreendendo a administração de undecanoato de testosterona a um homem em necessidade de suplementação de andrógeno - Google Patents

Formulação farmacêutica na forma de uma cápsula par administração oral, uso de undecanoato de testosterona, e, método de tratamento compreendendo a administração de undecanoato de testosterona a um homem em necessidade de suplementação de andrógeno

Info

Publication number
BR0009465A
BR0009465A BR0009465-0A BR0009465A BR0009465A BR 0009465 A BR0009465 A BR 0009465A BR 0009465 A BR0009465 A BR 0009465A BR 0009465 A BR0009465 A BR 0009465A
Authority
BR
Brazil
Prior art keywords
testosterone undecanoate
administration
oral administration
capsule
man
Prior art date
Application number
BR0009465-0A
Other languages
English (en)
Inventor
Henrik De Nijs
Susan Chandler
Elizabeth Anne Perry
Josephine Joan Chri Ferdinando
Original Assignee
Akzo Nobel Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv
Publication of BR0009465A publication Critical patent/BR0009465A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/568Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/16Masculine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Reproductive Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Fats And Perfumes (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Steroid Compounds (AREA)

Abstract

"FORMULAçãO FARMACêUTICA NA FORMA DE UMA CáPSULA PARA ADMINISTRAçãO ORAL, USO DE UNDECANOATO DE TESTOSTERONA, E, MéTODO DE TRATAMENTO COMPREENDENDO A ADMINISTRAçãO DE UNDECANOATO DE TESTOSTERONA A UM HOMEM EM NECESSIDADE DE SUPLEMENTAçãO DE ANDRóGENO" Divulgada é uma formulação farmacêutica na forma de uma cápsula para administração oral compreendendo undecanoato de testosterona como um ingrediente ativo dissolvido em um veiculo liquido farmaceuticamente aceitável, caracterizado em que o veículo liquido compreende pelo menos 50% em peso de óleo de ricino. A escolha de óleo de rícino como o veiculo liquido, em conjunção com a escolha de undecanoato de testosterona como o andrógeno, produz uma solução que compreende cerca de 200 a 250 mg/ml de TU. Esta é uma nova conquista para qualquer solução oralmente administrável de testosterona. A solução pode também conter um tensoativo lipofílico tal como lauroglicol.
BR0009465-0A 1999-04-01 2000-03-27 Formulação farmacêutica na forma de uma cápsula par administração oral, uso de undecanoato de testosterona, e, método de tratamento compreendendo a administração de undecanoato de testosterona a um homem em necessidade de suplementação de andrógeno BR0009465A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP99302581 1999-04-01
PCT/EP2000/002677 WO2000059512A1 (en) 1999-04-01 2000-03-27 Formulation comprising testosteron undecanoate and castor oil

Publications (1)

Publication Number Publication Date
BR0009465A true BR0009465A (pt) 2002-01-08

Family

ID=8241306

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0009465-0A BR0009465A (pt) 1999-04-01 2000-03-27 Formulação farmacêutica na forma de uma cápsula par administração oral, uso de undecanoato de testosterona, e, método de tratamento compreendendo a administração de undecanoato de testosterona a um homem em necessidade de suplementação de andrógeno

Country Status (27)

Country Link
EP (1) EP1189620B1 (pt)
JP (1) JP2002541111A (pt)
KR (1) KR100666016B1 (pt)
CN (1) CN1155385C (pt)
AT (1) ATE269708T1 (pt)
AU (1) AU768537B2 (pt)
BR (1) BR0009465A (pt)
CA (1) CA2366856C (pt)
CZ (1) CZ298573B6 (pt)
DE (1) DE60011771T2 (pt)
DK (1) DK1189620T3 (pt)
ES (1) ES2222199T3 (pt)
HK (1) HK1043544A1 (pt)
HU (1) HU229455B1 (pt)
ID (1) ID30481A (pt)
IL (2) IL145524A0 (pt)
MX (1) MXPA01009919A (pt)
NO (1) NO329420B1 (pt)
NZ (1) NZ514290A (pt)
PL (1) PL195163B1 (pt)
PT (1) PT1189620E (pt)
RU (1) RU2246296C2 (pt)
SK (1) SK286071B6 (pt)
TR (1) TR200102769T2 (pt)
TW (1) TWI280124B (pt)
WO (1) WO2000059512A1 (pt)
ZA (1) ZA200107781B (pt)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6652880B1 (en) 1999-04-01 2003-11-25 R.P. Scherer Technologies, Inc. Oral pharmaceutical compositions containing long-chain triglycerides and liphophilic surfactants
GB9907715D0 (en) * 1999-04-01 1999-05-26 Scherer Corp R P Pharmaceutical compositions
JO2505B1 (en) * 2003-03-14 2009-10-05 باير شيرنغ فارما اكتنجيسيلشافت Pharmacy methods and formulations for obtaining acceptable serum testosterone levels
DK1530965T3 (da) 2003-11-11 2006-07-17 Mattern Udo Kontrolleret frigivelsesleveringssystem til nasal applikation
US8784869B2 (en) 2003-11-11 2014-07-22 Mattern Pharma Ag Controlled release delivery system for nasal applications and methods of treatment
US20060140820A1 (en) 2004-12-28 2006-06-29 Udo Mattern Use of a container of an inorganic additive containing plastic material
US8492369B2 (en) 2010-04-12 2013-07-23 Clarus Therapeutics Inc Oral testosterone ester formulations and methods of treating testosterone deficiency comprising same
WO2006113505A2 (en) * 2005-04-15 2006-10-26 Clarus Therapeutics, Inc. Pharmaceutical delivery systems for hydrophobic drugs and compositions comprising same
CA2664427C (en) 2006-10-04 2012-06-05 M & P Patent Aktiengesellschaft Controlled release delivery system for nasal application of neurotransmitters
GB0818473D0 (en) 2008-10-08 2008-11-12 Probio Nutraceuticals As Composition
US11304960B2 (en) 2009-01-08 2022-04-19 Chandrashekar Giliyar Steroidal compositions
CA2795908C (en) * 2010-04-12 2015-10-13 Clarus Therapeutics, Inc. Oral testosterone ester formulations and methods of treating testoterone deficiency comprising same
GB201006200D0 (en) * 2010-04-14 2010-06-02 Ayanda As Composition
US9358241B2 (en) 2010-11-30 2016-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US20180153904A1 (en) 2010-11-30 2018-06-07 Lipocine Inc. High-strength testosterone undecanoate compositions
US9034858B2 (en) 2010-11-30 2015-05-19 Lipocine Inc. High-strength testosterone undecanoate compositions
US20120148675A1 (en) 2010-12-10 2012-06-14 Basawaraj Chickmath Testosterone undecanoate compositions
BR112013019257B1 (pt) * 2011-01-26 2019-09-03 Allergan Inc composição de androgênio para tratar uma condição oftálmica
US20130045958A1 (en) 2011-05-13 2013-02-21 Trimel Pharmaceuticals Corporation Intranasal 0.15% and 0.24% testosterone gel formulations and use thereof for treating anorgasmia or hypoactive sexual desire disorder
US9757388B2 (en) 2011-05-13 2017-09-12 Acerus Pharmaceuticals Srl Intranasal methods of treating women for anorgasmia with 0.6% and 0.72% testosterone gels
AR086400A1 (es) 2011-05-13 2013-12-11 Trimel Pharmaceuticals Corp Formulaciones en gel intranasal de testosterona en dosis de menor potencia y uso de las mismas para el tratamiento de la anorgasmia o el trastorno de deseo sexual hipoactivo
US11744838B2 (en) 2013-03-15 2023-09-05 Acerus Biopharma Inc. Methods of treating hypogonadism with transnasal testosterone bio-adhesive gel formulations in male with allergic rhinitis, and methods for preventing an allergic rhinitis event
CA2950670A1 (en) 2014-06-17 2015-12-23 Merck Sharp & Dohme B.V. Stable formulations of testosterone undecanoate
CA2948225C (en) * 2014-06-19 2022-05-31 Solural Pharma ApS Solid oral dosage form of lipophilic compounds
WO2016033556A1 (en) 2014-08-28 2016-03-03 Lipocine Inc. BIOAVAILABLE SOLID STATE (17-β)-HYDROXY-4-ANDROSTEN-3-ONE ESTERS
US20170246187A1 (en) 2014-08-28 2017-08-31 Lipocine Inc. (17-ß)-3-OXOANDROST-4-EN-17-YL TRIDECANOATE COMPOSITIONS AND METHODS OF THEIR PREPARATION AND USE
CN106999558A (zh) * 2014-08-29 2017-08-01 来普卡公司 (17‑β)‑3‑氧雄甾‑4‑烯‑17‑基十一酸酯组合物及其制备方法和用途
CA3078723A1 (en) 2016-11-28 2018-05-31 Nachiappan Chidambaram Oral testosterone undecanoate therapy
US20200155570A1 (en) * 2018-07-20 2020-05-21 Lipocine Inc. Liver disease

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1102095A (zh) * 1993-10-30 1995-05-03 浙江医科大学 长效雄激素类制剂——十一酸睾丸注射液
GB9608719D0 (en) * 1996-04-26 1996-07-03 Scherer Ltd R P Pharmaceutical compositions
SE9700642D0 (sv) * 1997-02-24 1997-02-24 Kronvall Stefan Med Ab Medel och sätt för förebyggande och behandling av det metabola syndromet

Also Published As

Publication number Publication date
NZ514290A (en) 2003-08-29
ES2222199T3 (es) 2005-02-01
ATE269708T1 (de) 2004-07-15
PL351259A1 (en) 2003-04-07
CA2366856A1 (en) 2000-10-12
IL145524A0 (en) 2002-06-30
PT1189620E (pt) 2004-10-29
HUP0200453A2 (hu) 2002-07-29
JP2002541111A (ja) 2002-12-03
HU229455B1 (en) 2013-12-30
SK286071B6 (sk) 2008-02-05
DE60011771T2 (de) 2004-11-04
WO2000059512A1 (en) 2000-10-12
HUP0200453A3 (en) 2003-06-30
SK13722001A3 (sk) 2002-02-05
CN1346274A (zh) 2002-04-24
MXPA01009919A (es) 2002-04-24
CZ20013507A3 (cs) 2002-03-13
EP1189620B1 (en) 2004-06-23
RU2246296C2 (ru) 2005-02-20
NO20014718D0 (no) 2001-09-28
DE60011771D1 (de) 2004-07-29
EP1189620A1 (en) 2002-03-27
ID30481A (id) 2001-12-13
CA2366856C (en) 2006-05-16
NO20014718L (no) 2001-09-28
CZ298573B6 (cs) 2007-11-14
KR20010108435A (ko) 2001-12-07
PL195163B1 (pl) 2007-08-31
HK1043544A1 (en) 2002-09-20
IL145524A (en) 2006-12-31
TWI280124B (en) 2007-05-01
DK1189620T3 (da) 2004-08-16
TR200102769T2 (tr) 2002-05-21
ZA200107781B (en) 2002-12-20
NO329420B1 (no) 2010-10-18
AU4111100A (en) 2000-10-23
CN1155385C (zh) 2004-06-30
KR100666016B1 (ko) 2007-01-10
AU768537B2 (en) 2003-12-18

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: INDEFIRO O PEDIDO DE ACORDO COM O(S) ARTIGO(S) DA LPI

B09B Patent application refused [chapter 9.2 patent gazette]

Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL.