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BG36348A3 - Метод за получаване на производни на тиенопиридинона - Google Patents

Метод за получаване на производни на тиенопиридинона

Info

Publication number
BG36348A3
BG36348A3 BG054209A BG5420981A BG36348A3 BG 36348 A3 BG36348 A3 BG 36348A3 BG 054209 A BG054209 A BG 054209A BG 5420981 A BG5420981 A BG 5420981A BG 36348 A3 BG36348 A3 BG 36348A3
Authority
BG
Bulgaria
Prior art keywords
preparing
derivatives
thienopyridinon
proven
formulated
Prior art date
Application number
BG054209A
Other languages
English (en)
Inventor
Robert Boigegrain
Jean-Pierre Maffrand
Norio Suzuki
Kiuichi Matsubayashi
Shinichiro Ashira
Original Assignee
Sanofi Sante Animale Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Sante Animale Sa filed Critical Sanofi Sante Animale Sa
Publication of BG36348A3 publication Critical patent/BG36348A3/bg

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02Boron compounds
    • C07F5/025Boronic and borinic acid compounds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02Silicon compounds
    • C07F7/08Compounds having one or more C—Si linkages
    • C07F7/10Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Метод за получаване на охарактеризирани и доказани в описанието производни на тиенопиридинона с обща формула..... Патентните претенции са формулирани в 3 точки.
BG054209A 1980-11-28 1981-11-19 Метод за получаване на производни на тиенопиридинона BG36348A3 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR8025274A FR2495156A1 (fr) 1980-11-28 1980-11-28 Derives de la thieno-pyridinone, leur procede de preparation et leur application therapeutique

Publications (1)

Publication Number Publication Date
BG36348A3 true BG36348A3 (bg) 1984-10-15

Family

ID=9248448

Family Applications (1)

Application Number Title Priority Date Filing Date
BG054209A BG36348A3 (bg) 1980-11-28 1981-11-19 Метод за получаване на производни на тиенопиридинона

Country Status (36)

Country Link
US (1) US4515951A (bg)
EP (1) EP0054442B1 (bg)
JP (1) JPS57120590A (bg)
KR (1) KR870000824B1 (bg)
AR (1) AR230285A1 (bg)
AT (1) ATE9160T1 (bg)
AU (1) AU559923B2 (bg)
BG (1) BG36348A3 (bg)
CA (1) CA1182458A (bg)
CS (1) CS224634B2 (bg)
CY (1) CY1281A (bg)
DD (1) DD201903A5 (bg)
DE (1) DE3165788D1 (bg)
DK (1) DK152132C (bg)
ES (1) ES8207180A1 (bg)
FI (1) FI72520C (bg)
FR (1) FR2495156A1 (bg)
GR (1) GR78021B (bg)
HK (1) HK61685A (bg)
HU (1) HU183711B (bg)
IE (1) IE51709B1 (bg)
IL (1) IL64146A (bg)
IN (1) IN155340B (bg)
MA (1) MA19331A1 (bg)
MY (1) MY8600008A (bg)
NO (1) NO155665C (bg)
NZ (1) NZ199021A (bg)
OA (1) OA06951A (bg)
PH (1) PH23776A (bg)
PL (1) PL129598B1 (bg)
PT (1) PT73988B (bg)
RO (1) RO83129B (bg)
SU (1) SU1110385A3 (bg)
YU (1) YU42448B (bg)
ZA (1) ZA817874B (bg)
ZW (1) ZW27481A1 (bg)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2528848A1 (fr) * 1982-06-16 1983-12-23 Sanofi Sa Nouveau derive de thieno-pyridone, son procede de preparation et son application therapeutique
FR2576901B1 (fr) * 1985-01-31 1987-03-20 Sanofi Sa Nouveaux derives de l'acide a-(oxo-2 hexahydro-2,4,5,6,7,7a thieno (3,2-c) pyridyl-5) phenyl acetique, leur procede de preparation et leur application therapeutique
FR2596392B1 (fr) * 1986-03-27 1988-08-05 Sanofi Sa Derives de l'acide a-(hydroxy-3 oxo-2 hexahydro-2,4,5,6,7,7a thieno (3,2-c) pyridyl-5) phenylacetique, leur procede de preparation, leur application comme medicaments et les compositions les renfermant
ATE57925T1 (de) * 1987-04-03 1990-11-15 Cl Pharma Neue 2-thienyloxyessigsaeurederivate, ein verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate.
FR2652579B1 (fr) * 1989-10-02 1992-01-24 Sanofi Sa Derives d'hydroxy-2 thiophene et furanne condenses avec un cycle azote, sur procede de preparation et leur application en therapeutique.
JP2730319B2 (ja) * 1991-04-26 1998-03-25 日本ビクター株式会社 磁気ディスク装置
JP3840662B2 (ja) * 1994-10-07 2006-11-01 宇部興産株式会社 2−シリルオキシ−テトラヒドロチエノピリジン類、その塩およびその製造方法
NZ334389A (en) * 1996-08-28 2001-05-25 Ube Industries Cyclic amine derivatives
ID25589A (id) * 1998-02-27 2000-10-19 Sankyo Company Ltd Cs Senyawa-senyawa amino siklik
DE60135780D1 (de) * 2000-12-25 2008-10-23 Daiichi Sankyo Co Ltd Aspirin enthaltende medizinische zusammensetzungen
US7557101B2 (en) * 2006-12-08 2009-07-07 Hoffman-La Roche Inc. 4,5,6,7-tetrahydro-thieno[3,2-c] pyridine derivatives
WO2009066326A2 (en) * 2007-11-19 2009-05-28 Msn Laboratories Limited Improved process for the preparation of prasugrel and its pharmaceutically acceptable salts
CN102241690B (zh) * 2010-05-13 2015-08-12 天津药物研究院 一类含腈基的噻吩并吡啶酯类衍生物、其制备方法和用途
CN101948479B (zh) * 2010-09-29 2013-01-30 横店集团家园化工有限公司 普拉格雷中间体及其制备方法
EP3241833A1 (en) 2010-10-18 2017-11-08 Cerenis Therapeutics Holding SA Compounds, compositions and methods useful for cholesterol mobilisation
CN108069981A (zh) * 2016-11-14 2018-05-25 天津药物研究院有限公司 5-取代-4,5,6,7-四氢噻吩并[3,2-c]吡啶-2(4H)-酮的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2215948B1 (bg) * 1973-02-01 1976-05-14 Centre Etd Ind Pharma
FR2345150A2 (fr) * 1975-08-06 1977-10-21 Centre Etd Ind Pharma Nouveaux derives de la thienopyridine, et leur application
FR2495157A1 (fr) * 1980-11-28 1982-06-04 Sanofi Sa Procede nouveau de preparation des tetrahydro-5, 6, 7, 7a 4h-thieno (3, 2-c) pyridinones-2
FR2508459A1 (fr) * 1981-06-30 1982-12-31 Sanofi Sa Procede de preparation de derives de la tetrahydro-5,6,7,7a 4h thieno (3,2-c) pyridinone-2

Also Published As

Publication number Publication date
DK152132B (da) 1988-02-01
AR230285A1 (es) 1984-03-01
CA1182458A (en) 1985-02-12
NO155665B (no) 1987-01-26
FI813730L (fi) 1982-05-29
NO814055L (no) 1982-06-01
NZ199021A (en) 1984-03-30
OA06951A (fr) 1983-07-31
FR2495156B1 (bg) 1983-08-05
IE812683L (en) 1982-05-28
RO83129A (ro) 1984-02-21
ES507705A0 (es) 1982-09-01
YU279081A (en) 1983-06-30
PH23776A (en) 1989-11-03
DD201903A5 (de) 1983-08-17
SU1110385A3 (ru) 1984-08-23
IE51709B1 (en) 1987-02-18
HU183711B (en) 1984-05-28
KR870000824B1 (ko) 1987-04-23
ATE9160T1 (de) 1984-09-15
FI72520C (fi) 1987-06-08
FI72520B (fi) 1987-02-27
IL64146A (en) 1984-12-31
PT73988A (fr) 1981-12-01
DE3165788D1 (en) 1984-10-04
AU7742981A (en) 1982-06-03
CS224634B2 (en) 1984-01-16
KR830007662A (ko) 1983-11-04
GR78021B (bg) 1984-09-26
PL233979A1 (bg) 1982-08-02
MY8600008A (en) 1986-12-31
DK520781A (da) 1982-05-29
AU559923B2 (en) 1987-03-26
JPS57120590A (en) 1982-07-27
IN155340B (bg) 1985-01-19
US4515951A (en) 1985-05-07
EP0054442B1 (fr) 1984-08-29
PL129598B1 (en) 1984-05-31
ZA817874B (en) 1982-10-27
FR2495156A1 (fr) 1982-06-04
EP0054442A1 (fr) 1982-06-23
HK61685A (en) 1985-08-23
ES8207180A1 (es) 1982-09-01
ZW27481A1 (en) 1982-02-17
PT73988B (fr) 1983-04-14
IL64146A0 (en) 1982-01-31
JPH0239517B2 (bg) 1990-09-05
CY1281A (en) 1985-07-05
DK152132C (da) 1988-06-20
RO83129B (ro) 1984-02-28
YU42448B (en) 1988-08-31
NO155665C (no) 1987-05-06
MA19331A1 (fr) 1982-07-01

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