ATA218378A - Verfahren zur herstellung von neuen ver- bindungen - Google Patents

Verfahren zur herstellung von neuen ver- bindungen

Info

Publication number: ATA218378A
Authority: AT; Austria
Prior art keywords: producing new; new connections; connections; producing; new
Prior art date: 1977-03-25

Application number

AT218378A

Other languages

English (en)

Other versions

AT360153B (de

Original Assignee

Roussel Uclaf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-03-25

Filing date

1978-03-28

Publication date

1980-05-15

1977-03-25 Priority claimed from FR7708988A external-priority patent/FR2384782A1/fr

1977-12-05 Priority claimed from FR7736512A external-priority patent/FR2421906A2/fr

1978-03-28 Application filed by Roussel Uclaf filed Critical Roussel Uclaf

1979-09-14 Priority to AT607579A priority Critical patent/AT361122B/de

1980-05-15 Publication of ATA218378A publication Critical patent/ATA218378A/de

1980-12-29 Application granted granted Critical

1980-12-29 Publication of AT360153B publication Critical patent/AT360153B/de

Status Expired legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)

AT218378A 1977-03-25 1978-03-28 Verfahren zur herstellung von neuen ver- bindungen Expired AT360153B (de)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
AT607579A AT361122B (de)	1977-12-05	1979-09-14	Verfahren zur herstellung neuer verbindungen

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
FR7708988A FR2384782A1 (fr)	1977-03-25	1977-03-25	Nouvelles oximes derivees de l'acide 3-acetoxymethyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR7736512A FR2421906A2 (fr)	1977-12-05	1977-12-05	Nouvelles oximes derivees de l'acide 3-acetoxy methyl 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments

Publications (2)

Publication Number	Publication Date
ATA218378A true ATA218378A (de)	1980-05-15
AT360153B AT360153B (de)	1980-12-29

Family

ID=26219930

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT218378A Expired AT360153B (de)	1977-03-25	1978-03-28	Verfahren zur herstellung von neuen ver- bindungen

Country Status (18)

Country	Link
US (4)	US4288434A (de)
JP (2)	JPS53119887A (de)
AT (1)	AT360153B (de)
AU (1)	AU520657B2 (de)
CA (1)	CA1125280A (de)
CH (4)	CH648555A5 (de)
DE (2)	DE2858771C2 (de)
DK (1)	DK159156C (de)
ES (2)	ES468169A1 (de)
GB (2)	GB1605175A (de)
HU (1)	HU182567B (de)
IE (1)	IE47361B1 (de)
IT (1)	IT1103478B (de)
LU (1)	LU79312A1 (de)
NL (1)	NL192041C (de)
PH (1)	PH15764A (de)
PT (1)	PT67815A (de)
SE (2)	SE439312B (de)

Families Citing this family (32)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE878514A (fr) *	1978-09-04	1980-02-29	Fujisawa Pharmaceutical Co	Procede de preparation de composes d'acide 3-cephem-4-carboxylique a disubstitution en positions 3 et 7, nouveaux produits ainsi obtenus et leur utilisation pour leur activite antibacterienne
PH17188A (en)	1977-03-14	1984-06-14	Fujisawa Pharmaceutical Co	New cephem and cepham compounds and their pharmaceutical compositions and method of use
US4409217A (en)	1977-03-14	1983-10-11	Fujisawa Pharmaceutical Co., Ltd.	Cephem compounds
SE439312B (sv) *	1977-03-25	1985-06-10	Roussel Uclaf	Sett att framstella nya oximderivat av 3-acetoximetyl-7-aminotiazolylacetamido cefalosporansyra
FR2410655A1 (fr) *	1977-12-05	1979-06-29	Roussel Uclaf	Nouvelles oximes derivees de l'acide 3-substitue 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR2432521A1 (fr) *	1978-03-31	1980-02-29	Roussel Uclaf	Nouvelles oximes o-substituees derivees de l'acide 7-amino thiazolyl acetamido cephalosporanique, leur procede de preparation et leur application comme medicaments
FR2421907A1 (fr) *	1978-04-07	1979-11-02	Roussel Uclaf	Nouvelles cephalosporines derivees de l'acide 7-/2-(2-amino 4-thiazolyl)2-(carboxymethoxyimino/acetamido 3-substitue cephalosporanique, leur procede de preparation et leur application comme medicaments
US4288435A (en)	1978-07-17	1981-09-08	Fujisawa Pharmaceutical Co., Ltd.	3,7-Disubstituted-3-cephem-4-carboxylic acid compounds and pharmaceutical antibacterial compositions containing them
US4284631A (en) *	1978-07-31	1981-08-18	Fujisawa Pharmaceutical Co., Ltd.	7-Substituted cephem compounds and pharmaceutical antibacterial compositions containing them
US4372952A (en)	1978-07-31	1983-02-08	Fujisawa Pharmaceutical Co., Ltd.	Cephem compounds
US4341775A (en) *	1978-09-11	1982-07-27	Fujisawa Pharmaceutical Co., Ltd.	Cephem compounds
DE2945248A1 (de) *	1978-11-13	1980-05-22	Fujisawa Pharmaceutical Co	Cephem-verbindungen, verfahren zu ihrer herstellung und sie enthaltende antibakterielle pharmazeutische mittel
US4237128A (en)	1979-04-12	1980-12-02	E. R. Squibb & Sons, Inc.	7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides
AU538653B2 (en) *	1979-10-02	1984-08-23	Glaxo Group Limited	7-(2-(2-amino thiazol-4-yl)-2-(carboxymethoxyimino) acetamioo)-3-(1-pyridiniammethyl)-ceph-3-em-4-carboxylate
US4409214A (en) *	1979-11-19	1983-10-11	Fujisawa Pharmaceutical, Co., Ltd.	7-Acylamino-3-vinylcephalosporanic acid derivatives and processes for the preparation thereof
US4252802A (en) *	1980-03-13	1981-02-24	E. R. Squibb & Sons, Inc.	Hydroxamic acid derivatives of 7-[(2-amino-4-thiazolyl)-oximino] cephalosporins
GR76342B (de) *	1981-02-02	1984-08-06	Fujisawa Pharmaceutical Co
EP0058250A3 (de) *	1981-02-17	1983-08-17	F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft	Cephalosporinderivate, deren Herstellung und entsprechende pharmazeutische Präparate
IE53429B1 (en) *	1981-08-03	1988-11-09	Fujisawa Pharmaceutical Co	New cephem compounds and processes for preparation thereof
DE3265277D1 (en) *	1981-11-13	1985-09-12	Glaxo Group Ltd	Thiazole derivatives and their use in the manufacture of beta lactam antibiotics
JPS58135872A (ja) *	1981-11-13	1983-08-12	グラクソ・グル−プ・リミテツド	新規な化合物およびその製法
ATE30724T1 (de)	1982-06-28	1987-11-15	Bristol Myers Co	Cephalosporinderivate, verfahren zu ihrer herstellung und pharmazeutische zusammensetzungen die sie enthalten.
EP0115770B2 (de) *	1983-01-07	1996-06-19	Takeda Chemical Industries, Ltd.	Thiazolderivate
US4652651A (en) *	1983-05-31	1987-03-24	Hoffmann-La Roche Inc.	Process for the manufacture of 1-sulpho-2-oxoazetidine carboxylic acid intermediates via catalytic ester cleavage
EP0150507B1 (de) *	1983-12-29	1992-08-05	Mochida Pharmaceutical Co., Ltd.	Cephalosporinverbindungen, Verfahren zu ihrer Herstellung und pharmazeutishe Präparate
AT381496B (de) *	1984-04-10	1986-10-27	Biochemie Gmbh	Verfahren zur herstellung von cephalosporinantibiotika
US4680409A (en) *	1984-10-09	1987-07-14	E. R. Squibb & Sons, Inc.	Hydrazide containing derivatives of 2-amino-4-thiazole-acetic acid
US4610824A (en) *	1984-10-09	1986-09-09	E. R. Squibb & Sons, Inc.	Hydrazide derivatives of monocyclic beta-lactam antibiotics
US4840945A (en) *	1985-04-01	1989-06-20	Mochida Pharmaceutical Co., Ltd.	Cephalosporin derivatives
US4647660A (en) *	1985-05-02	1987-03-03	E. R. Squibb & Sons, Inc.	3-acylamino-2-oxo-1-azetidinesulfonic acids
IL84128A (en) *	1986-10-13	1992-12-01	Eisai Co Ltd	3-propenylcephem derivatives, their preparation and pharmaceutical compositions containing them
CN1313452C (zh) *	2005-06-08	2007-05-02	浙江普洛化学有限公司	制备(z)－2－(2－氨基－4－噻唑)－2－羟基亚胺乙酸酯及其衍生物的方法

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3971778A (en) *	1972-05-12	1976-07-27	Glaxo Laboratories Limited	Cephalosporins having (α-etherified oximino)acylamido groups at the 7-position
GB1399086A (en)	1971-05-14	1975-06-25	Glaxo Lab Ltd	Cephalosporin compounds
GB1472534A (en) *	1973-07-06	1977-05-04	Glaxo Lab Ltd	7beta-hydroxyiminoacylamido-cephalosporins
US4095021A (en) *	1973-12-21	1978-06-13	Glaxo Laboratories Limited	3-Carbamoyloxymethyl or N-methyl-carbamoyloxymethyl-7-[2-carboxymethoxyimino-2-(fur-2-yl or thien-2-yl)acetamido]ceph-3-em-4-carboxylic acids and derivatives thereof
SE7416195L (sv) *	1973-12-21	1975-09-22	Glaxo Lab Ltd	Forfarande for framstellning av cefalosporiner.
DK154939C (da)	1974-12-19	1989-06-12	Takeda Chemical Industries Ltd	Analogifremgangsmaade til fremstilling af thiazolylacetamido-cephemforbindelser eller farmaceutisk acceptable salte eller estere deraf
US4203899A (en) *	1974-12-19	1980-05-20	Takeda Chemical Industries, Ltd.	Thiazolylacetamido compounds
DE2760123C2 (de) *	1976-01-23	1986-04-30	Roussel-Uclaf, Paris	7-Aminothiazolyl-syn-oxyiminoacetamidocephalosporansäuren, ihre Herstellung und sie enthaltende pharmazeutische Zusammensetzungen
US4376203A (en) *	1976-01-23	1983-03-08	Roussell Uclaf	Novel 3-acetoxymethyl-7-(iminoacetamido)-cephalosporanic acid derivatives
US4166115A (en) *	1976-04-12	1979-08-28	Fujisawa Pharmaceutical Co., Ltd.	Syn 7-oxoimino substituted derivatives of cephalosporanic acid
GB1576625A (en) *	1976-04-12	1980-10-08	Fujisawa Pharmaceutical Co	Syn isomer 3,7 disubstituted 3 cephem 4 carboxylic acid compounds and processes for the preparation thereof
DK162391C (da) *	1976-04-12	1992-03-09	Fujisawa Pharmaceutical Co	Analogifremgangsmaade til fremstilling af syn-isomerer af 3,7-disubstituerede 3-cephem-4-carboxylsyreforbindelser
JPS6011713B2 (ja) *	1976-09-08	1985-03-27	武田薬品工業株式会社	セフアロスポリン誘導体およびその製造法
PH17188A (en) *	1977-03-14	1984-06-14	Fujisawa Pharmaceutical Co	New cephem and cepham compounds and their pharmaceutical compositions and method of use
SE439312B (sv) *	1977-03-25	1985-06-10	Roussel Uclaf	Sett att framstella nya oximderivat av 3-acetoximetyl-7-aminotiazolylacetamido cefalosporansyra

1978
- 1978-03-13 SE SE7802833A patent/SE439312B/sv not_active IP Right Cessation
- 1978-03-14 US US05/886,421 patent/US4288434A/en not_active Expired - Lifetime
- 1978-03-22 DE DE2858771A patent/DE2858771C2/de not_active Expired - Lifetime
- 1978-03-22 ES ES468169A patent/ES468169A1/es not_active Expired
- 1978-03-22 DK DK129578A patent/DK159156C/da not_active IP Right Cessation
- 1978-03-22 HU HU78RO972A patent/HU182567B/hu unknown
- 1978-03-22 DE DE19782812625 patent/DE2812625A1/de active Granted
- 1978-03-23 PT PT67815A patent/PT67815A/pt unknown
- 1978-03-23 CH CH1361/84A patent/CH648555A5/fr not_active IP Right Cessation
- 1978-03-23 AU AU34471/78A patent/AU520657B2/en not_active Expired
- 1978-03-23 CA CA299,661A patent/CA1125280A/fr not_active Expired
- 1978-03-23 GB GB11613/78A patent/GB1605175A/en not_active Expired
- 1978-03-23 GB GB16825/80A patent/GB1605176A/en not_active Expired
- 1978-03-23 NL NL7803166A patent/NL192041C/nl not_active IP Right Cessation
- 1978-03-23 CH CH322978A patent/CH633292A5/fr not_active IP Right Cessation
- 1978-03-24 IT IT48604/78A patent/IT1103478B/it active
- 1978-03-24 JP JP3319378A patent/JPS53119887A/ja active Granted
- 1978-03-24 LU LU79312A patent/LU79312A1/xx unknown
- 1978-03-27 PH PH20927A patent/PH15764A/en unknown
- 1978-03-28 AT AT218378A patent/AT360153B/de not_active Expired
- 1978-03-29 IE IE604/78A patent/IE47361B1/en not_active IP Right Cessation
1979
- 1979-02-09 ES ES477592A patent/ES477592A1/es not_active Expired
1981
- 1981-05-04 US US06/260,311 patent/US4386210A/en not_active Expired - Lifetime
1982
- 1982-06-18 CH CH386882A patent/CH639652A5/fr not_active IP Right Cessation
1983
- 1983-02-25 US US06/469,710 patent/US4487937A/en not_active Expired - Lifetime
- 1983-08-02 SE SE8304239A patent/SE453192B/sv not_active IP Right Cessation
- 1983-12-02 CH CH644383A patent/CH646159A5/fr not_active IP Right Cessation
1984
- 1984-01-30 US US06/574,876 patent/US4483981A/en not_active Expired - Lifetime
1988
- 1988-06-22 JP JP63152471A patent/JPS6425768A/ja active Granted

Also Published As

Publication number	Publication date
IT7848604A0 (it)	1978-03-24
GB1605176A (en)	1982-11-17
US4487937A (en)	1984-12-11
SE453192B (sv)	1988-01-18
DK129578A (da)	1978-09-26
NL192041C (nl)	1997-01-07
JPS53119887A (en)	1978-10-19
JPS6425768A (en)	1989-01-27
HU182567B (en)	1984-02-28
CH648555A5 (fr)	1985-03-29
LU79312A1 (fr)	1978-11-03
JPS6237037B2 (de)	1987-08-10
IT1103478B (it)	1985-10-14
ES468169A1 (es)	1979-07-16
JPH0362711B2 (de)	1991-09-26
IE780604L (en)	1978-09-25
AT360153B (de)	1980-12-29
DK159156C (da)	1991-02-11
US4386210A (en)	1983-05-31
CH639652A5 (fr)	1983-11-30
SE8304239D0 (sv)	1983-08-02
CH633292A5 (fr)	1982-11-30
PH15764A (en)	1983-03-24
AU3447178A (en)	1979-09-27
CH646159A5 (fr)	1984-11-15
US4288434A (en)	1981-09-08
GB1605175A (en)	1982-11-17
SE8304239L (sv)	1983-08-02
US4483981A (en)	1984-11-20
DE2812625C2 (de)	1990-08-23
ES477592A1 (es)	1979-08-01
SE7802833L (sv)	1978-11-02
DK159156B (da)	1990-09-10
IE47361B1 (en)	1984-03-07
AU520657B2 (en)	1982-02-18
NL192041B (nl)	1996-09-02
CA1125280A (fr)	1982-06-08
DE2858771C2 (de)	1990-09-06
PT67815A (fr)	1978-04-01
DE2812625A1 (de)	1978-09-28
SE439312B (sv)	1985-06-10
NL7803166A (nl)	1978-09-27

Publication	Publication Date	Title
AT360153B (de)	1980-12-29	Verfahren zur herstellung von neuen ver- bindungen
AT372093B (de)	1983-08-25	Verfahren zur herstellung von neuen corticoid-17- alkylcarbonaten
AT367425B (de)	1982-07-12	Verfahren zur herstellung von neuen cephemderivaten
AT367426B (de)	1982-07-12	Verfahren zur herstellung von neuen cephemderivaten
AT362065B (de)	1981-04-27	Verfahren zur herstellung von neuen pleuromutilinglycosidderivaten
LU79212A1 (de)	1979-05-25	Verfahren zur herstellung von neuen 4-acylamino-phenylaethanolaminen
AT363182B (de)	1981-07-10	Verfahren zur herstellung von neuen cephemderivaten
AT371455B (de)	1983-06-27	Verfahren zur herstellung von neuen prostanderivaten
AT368753B (de)	1982-11-10	Verfahren zur herstellung von neuen azacycloalkanen
AT361455B (de)	1981-03-10	Verfahren zur herstellung von neuen substituierten 3-phenyl-cycloalkan- oder - -cycloalken-1-olen
AT368137B (de)	1982-09-10	Verfahren zur herstellung von neuen 4-amino-5alkylthiopyrimidinen
AT366368B (de)	1982-04-13	Verfahren zur herstellung von neuen chinolylguanidinen
AT357673B (de)	1980-07-25	Verfahren zur herstellung von neuen 9-amino- desoxyclavulansaeurederivaten
AT361622B (de)	1981-03-25	Verfahren zur herstellung von neuen anthra- cyclinglycosid-anitbiotika
AT365591B (de)	1982-01-25	Verfahren zur herstellung von neuen indolderivaten
ATA472577A (de)	1980-02-15	Verfahren zur herstellung von neuen 1-acyl-4- -hydroxy-imidazol-5-carboxamid-derivaten
AT358169B (de)	1980-08-25	Verfahren zur herstellung von neuen ver- bindungen
AT362368B (de)	1981-05-11	Verfahren zur herstellung von neuen oxazolidin- 2-on-derivaten
AT372690B (de)	1983-11-10	Verfahren zur herstellung von neuen polyhydantoinen
AT360676B (de)	1981-01-26	Verfahren zur herstellung von neuen 17beta- -hydroxy-4-androsten-3-onen
AT371109B (de)	1983-06-10	Verfahren zur herstellung von neuen benzolsulfonamidderivaten
ATA750578A (de)	1981-07-15	Verfahren zur herstellung von neuen pyridothiazo- linen
AT365203B (de)	1981-12-28	Verfahren zur herstellung von neuen 9-fluorprednisolon-derivaten
AT371119B (de)	1983-06-10	Verfahren zur herstellung von neuen sulfoximid-derivaten
AT359517B (de)	1980-11-10	Verfahren zur herstellung von neuen alfa- -halogenaethylcarbamidsaeurehalogeniden

Legal Events

Date	Code	Title	Description
1999-01-15	ELA	Expired due to lapse of time
2002-12-15	RER	Ceased as to paragraph 5 lit. 3 law introducing patent treaties