AR240924A2 - "procedimiento para preparar derivados de 1,3-oxazolidin-2-ona y sus sales". - Google Patents
"procedimiento para preparar derivados de 1,3-oxazolidin-2-ona y sus sales".Info
- Publication number
- AR240924A2 AR240924A2 AR30060485A AR30060485A AR240924A2 AR 240924 A2 AR240924 A2 AR 240924A2 AR 30060485 A AR30060485 A AR 30060485A AR 30060485 A AR30060485 A AR 30060485A AR 240924 A2 AR240924 A2 AR 240924A2
- Authority
- AR
- Argentina
- Prior art keywords
- formula
- alkyl
- oxazolidine
- derivatives
- occ13
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/02—Muscle relaxants, e.g. for tetanus or cramps
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/18—Oxygen atoms
- C07D263/20—Oxygen atoms attached in position 2
- C07D263/22—Oxygen atoms attached in position 2 with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to other ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Neurology (AREA)
- Public Health (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
UN PROCEDIMIENTO PARA PREPARAR UN DERIVADO DE 1,3-OXAZOLIDIN-2-ONA REPRESENTADO POR LA FORMULA (I), EN LA CUAL R ES ALQUILO RECTO O RAMIFICADO; N ES UN ENTERO DE 4 A 6 Y X REPRESENTA HIDROGENO, 2-3- O 4-ALQUILO 4-HALO O 4-ALCOXI, PORQUE COMPRENDE HACER REACCIONAR UN COMPUESTO DE FORMULA (II), CON UN REACTIVO ELEGIDO ENTRE EL DIALQUILCARBONATO, C1-CO-C1, C1-CO-OCC13 O C1-COO-ALQUILO, SEGUIDO EN ESTE ULTIMO CASO DE LA CICLIZACION EN PRESENCIA DE BASES DEL INTERMEDIARIO FERRADO DE FORMULA III, Y OPCIONALMENTE OBTENER LAS SALES FARMACEUTICAMENTE ACEPTABLES DE LOS COMPUESTOS OBTENIDOS DE FORMULA (I).
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP59203624A JPS6183170A (ja) | 1984-09-28 | 1984-09-28 | 新規な１，３−オキサゾリジン−２−オン誘導体およびその製造法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| AR240924A2 true AR240924A2 (es) | 1991-03-27 |
| AR240924A1 AR240924A1 (es) | 1991-03-27 |
Family
ID=16477122
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR300604A AR240924A1 (es) | 1984-09-28 | 1985-05-31 | "procedimiento para preparar derivados de 1,3-oxazolidin-2-ona y sus sales". |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US4644063A (es) |
| JP (1) | JPS6183170A (es) |
| KR (1) | KR900004323B1 (es) |
| AR (1) | AR240924A1 (es) |
| AT (1) | AT392069B (es) |
| AU (1) | AU566419B2 (es) |
| BR (1) | BR8502707A (es) |
| CA (1) | CA1252092A (es) |
| CH (1) | CH663207A5 (es) |
| CS (1) | CS273606B2 (es) |
| DE (1) | DE3519261C2 (es) |
| DK (1) | DK165952C (es) |
| ES (2) | ES8800571A1 (es) |
| FR (1) | FR2571052B1 (es) |
| GB (2) | GB8512975D0 (es) |
| HU (1) | HU199132B (es) |
| IN (1) | IN162060B (es) |
| IT (1) | IT1208807B (es) |
| MX (2) | MX161397A (es) |
| MY (1) | MY102081A (es) |
| NL (1) | NL193191C (es) |
| NZ (1) | NZ212143A (es) |
| PH (1) | PH20852A (es) |
| RO (1) | RO91422B (es) |
| SE (1) | SE463100B (es) |
| SU (2) | SU1402263A3 (es) |
| ZA (1) | ZA854001B (es) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6183147A (ja) * | 1984-09-28 | 1986-04-26 | Nippon Chemiphar Co Ltd | 新規なアミノアルコール誘導体およびその製造法並びにそれを有効成分とするグルタミン酸遮断剤 |
| JPH0759570B2 (ja) * | 1986-05-06 | 1995-06-28 | 三井東圧化学株式会社 | ２−オキサゾリジノン類の製造方法 |
| JPH0713017B2 (ja) * | 1986-06-18 | 1995-02-15 | 日本ケミファ株式会社 | 脳細胞保護作用を有する医薬組成物 |
| ES2053748T3 (es) * | 1987-09-10 | 1994-08-01 | Merck Sharp & Dohme | Oxazoles y tiazoles para el tratamiento de la demencia senil. |
| CA1329128C (en) * | 1988-03-24 | 1994-05-03 | Nobuyoshi Iwata | Isoxazolinones as cerebro-active drugs |
| JPH0314562A (ja) * | 1988-04-11 | 1991-01-23 | Nippon Chemiphar Co Ltd | 新規なアルキレンジアミン誘導体およびグルタミン酸遮断剤 |
| US5187171A (en) * | 1989-01-09 | 1993-02-16 | G. D. Searle & Co. | Use of a glycine b partial agonist as an antipsychotic |
| ES2121036T3 (es) * | 1992-07-14 | 1998-11-16 | Nippon Chemiphar Co | Derivados de alquilenodiamina. |
| US5698573A (en) * | 1993-09-15 | 1997-12-16 | Merck, Sharp & Dohme, Ltd. | Imidazolone and oxazolone derivatives as dopamine antagonists |
| DE4425613A1 (de) * | 1994-07-20 | 1996-01-25 | Bayer Ag | 5-gliedrige Heteroaryl-oxazolidinone |
| US6037354A (en) | 1997-06-18 | 2000-03-14 | Merck & Co., Inc. | Alpha 1a adrenergic receptor antagonists |
| AU2014230940B2 (en) | 2013-03-14 | 2016-12-08 | Akzo Nobel Chemicals International B.V. | Cellulose ether as a drift control agent and rainfastness agent |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2437389A (en) * | 1948-03-09 | Oxazoeidones and erocesstok | ||
| DE1135461B (de) * | 1959-05-08 | 1962-08-30 | Knoll Ag | Verfahren zur Herstellung von basisch substituierten Phthalimidinen |
| FR1301267A (fr) * | 1961-04-04 | 1962-08-17 | Science Union Et Compagnie Soc | Nouveaux dérivés de l'oxazolidinone-2 et leurs procédés de préparation |
| US3131197A (en) * | 1963-03-13 | 1964-04-28 | Smith Kline French Lab | 5-(3, 4-carbonyldioxyphenyl)-3-isopropyl-2-oxazolidone |
| US3576808A (en) * | 1967-09-15 | 1971-04-27 | Miles Lab | N-4-phenyl-1-piperazinylalkyl-5-phenyl-oxazolidinones |
| GB1222708A (en) * | 1968-10-22 | 1971-02-17 | Delalande Sa | Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation |
| FR2179582B1 (es) * | 1972-04-13 | 1975-10-10 | Synthelabo |
-
1984
- 1984-09-28 JP JP59203624A patent/JPS6183170A/ja active Granted
-
1985
- 1985-05-21 NZ NZ212143A patent/NZ212143A/en unknown
- 1985-05-22 GB GB858512975A patent/GB8512975D0/en active Pending
- 1985-05-22 SE SE8502525A patent/SE463100B/sv not_active IP Right Cessation
- 1985-05-23 DK DK230185A patent/DK165952C/da not_active IP Right Cessation
- 1985-05-23 IN IN382/MAS/85A patent/IN162060B/en unknown
- 1985-05-24 DE DE3519261A patent/DE3519261C2/de not_active Expired - Fee Related
- 1985-05-24 PH PH32310A patent/PH20852A/en unknown
- 1985-05-27 ES ES543517A patent/ES8800571A1/es not_active Expired
- 1985-05-27 ZA ZA854001A patent/ZA854001B/xx unknown
- 1985-05-28 CA CA000482506A patent/CA1252092A/en not_active Expired
- 1985-05-29 KR KR1019850003726A patent/KR900004323B1/ko not_active IP Right Cessation
- 1985-05-29 US US06/739,059 patent/US4644063A/en not_active Expired - Lifetime
- 1985-05-30 SU SU853902250A patent/SU1402263A3/ru active
- 1985-05-30 FR FR8508128A patent/FR2571052B1/fr not_active Expired
- 1985-05-30 GB GB08513685A patent/GB2165237B/en not_active Expired
- 1985-05-30 HU HU852082A patent/HU199132B/hu not_active IP Right Cessation
- 1985-05-30 IT IT8567500A patent/IT1208807B/it active
- 1985-05-30 RO RO118984A patent/RO91422B/ro unknown
- 1985-05-31 BR BR8502707A patent/BR8502707A/pt not_active IP Right Cessation
- 1985-05-31 MX MX205493A patent/MX161397A/es unknown
- 1985-05-31 CH CH2317/85A patent/CH663207A5/fr not_active IP Right Cessation
- 1985-05-31 NL NL8501579A patent/NL193191C/nl not_active IP Right Cessation
- 1985-05-31 CS CS392785A patent/CS273606B2/cs unknown
- 1985-05-31 AT AT0165685A patent/AT392069B/de not_active IP Right Cessation
- 1985-05-31 AR AR300604A patent/AR240924A1/es active
- 1985-07-09 AU AU44697/85A patent/AU566419B2/en not_active Ceased
-
1986
- 1986-05-13 SU SU864027452A patent/SU1431679A3/ru active
- 1986-09-18 ES ES557075A patent/ES8802152A1/es not_active Expired
-
1987
- 1987-09-29 MY MYPI87002215A patent/MY102081A/en unknown
-
1990
- 1990-07-16 MX MX2159290A patent/MX21592A/es unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AR240924A2 (es) | "procedimiento para preparar derivados de 1,3-oxazolidin-2-ona y sus sales". | |
| SE7604052L (sv) | Nya erytromycinderivat och forfarande for framstellning derav | |
| SE8404019L (sv) | Oftalmiska antiinflammatoriska medel | |
| ES521655A0 (es) | Procedimiento para la preparacion de aminoacidos ciclicos o esteres de los mismos. | |
| AR247891A1 (es) | Procedimiento para preparar nuevos derivados de 2'-halometilidencitidina y uridina | |
| DK0406119T3 (da) | Hidtil ukendte peptidderivater, fremgangsmåde til fremstilling heraf og farmaceutiske midler indeholdende dem | |
| SE7705143L (sv) | Nya omega-aminokarboxylsyraamider jemte sett for deras framstellning | |
| GB2080683B (en) | Stabilization of pharmaceutical compositions containing acid addition salts of thieno-pyridine derivatives | |
| FI891245A (fi) | Starka soetningsmedel. | |
| SE7707689L (sv) | 2-brom-6-fluor-n-2-imidazolidinylidenbensamin dess syraadditionssalter, lekemedel innehallande dessa och forfarande for framstellning derav | |
| JPS5227721A (en) | Process for preparation of substituted phosphonic acid derivatives | |
| ES2043070T3 (es) | Procedimiento para la preparacion de derivados de la benzotiazolamina-2. | |
| MX168931B (es) | Procedimiento para preparar compuestos de organofosforo | |
| ES2128554T3 (es) | Nuevos derivados del acido glutamico, procedimiento para su preparacion y su utilizacion como medicamentos para el aumento de la memoria y aprendizaje. | |
| SE7609495L (sv) | N-tetrahydrofurfuryl-noroximorfon, dess syraadditionssalter, lekemedel innehallande dessa samt forfarande for framstellning derav | |
| SE7902083L (sv) | Bicyklooktanderivat till anvendning som medel mot trombos | |
| SE8102489L (sv) | Sett att framstella adenosinderivat | |
| ES2060592T3 (es) | Un tioester y su uso en la preparacion de composiciones farmaceuticas para el tratamiento de los sindromes de isquemia y reperfusion. | |
| ES2040226T3 (es) | Procedimiento para preparar nuevos tetrahidro-benzotiazoles. | |
| ES2051731T3 (es) | Un procedimiento para preparar antibioticos macrolidos y su uso. | |
| ES2075365T3 (es) | Procedimiento para la preparacion de derivados de 3-alcoximetil cefalosporina. | |
| ES2117003T3 (es) | Derivados oligopeptidicos de hipoxantina dotados de actividad inmunomoduladora, y composiciones farmaceuticas que los contienen. | |
| AR240788A2 (es) | Una composicion promotora del crecimiento de vegetales. | |
| FI813290L (fi) | Fosfonoformaldehyd foerfarande foer dess framstaellning och dess anvaendning som mellanprodukt vid framstaellning av laekemedel | |
| ES2038636T3 (es) | Procedimiento para la obtencion de derivados de aminotiofeno. |