AR114251A1 - Formas cristalinas de n-[2-(2,4-diclorofenil)ciclobutil]-2-(trifluorometl)piridin-3-carboxamida - Google Patents
Formas cristalinas de n-[2-(2,4-diclorofenil)ciclobutil]-2-(trifluorometl)piridin-3-carboxamidaInfo
- Publication number
- AR114251A1 AR114251A1 ARP190100300A ARP190100300A AR114251A1 AR 114251 A1 AR114251 A1 AR 114251A1 AR P190100300 A ARP190100300 A AR P190100300A AR P190100300 A ARP190100300 A AR P190100300A AR 114251 A1 AR114251 A1 AR 114251A1
- Authority
- AR
- Argentina
- Prior art keywords
- dichlorophenyl
- carboxamide
- crystalline forms
- cyclobutyl
- trifluoromethyl
- Prior art date
Links
- -1 2,4-DICHLOROPHENYL Chemical class 0.000 title 1
- DFPAKSUCGFBDDF-UHFFFAOYSA-N Nicotinamide Chemical compound NC(=O)C1=CC=CN=C1 DFPAKSUCGFBDDF-UHFFFAOYSA-N 0.000 title 1
- 125000004201 2,4-dichlorophenyl group Chemical group [H]C1=C([H])C(*)=C(Cl)C([H])=C1Cl 0.000 abstract 2
- 238000000634 powder X-ray diffraction Methods 0.000 abstract 2
- GBFKIHJZPMECCF-UHFFFAOYSA-N N-[2-(2,4-dichlorophenyl)cyclobutyl]-2-(trifluoromethyl)pyridine-3-carboxamide Chemical compound ClC1=C(C=CC(=C1)Cl)C1C(CC1)NC(=O)C=1C(=NC=CC=1)C(F)(F)F GBFKIHJZPMECCF-UHFFFAOYSA-N 0.000 abstract 1
- 241000244206 Nematoda Species 0.000 abstract 1
- 239000000463 material Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 244000045561 useful plants Species 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/81—Amides; Imides
- C07D213/82—Amides; Imides in position 3
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
- A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Environmental Sciences (AREA)
- Dentistry (AREA)
- Engineering & Computer Science (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Plant Pathology (AREA)
- Zoology (AREA)
- Wood Science & Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Pyridine Compounds (AREA)
- Liquid Crystal Substances (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Formas cristalinas de N-[2-(2,4-diclorofenil)ciclobutil]-2-(trifluorometil)piridin-3-carboxamida, composición agrícola o farmacéutica que las comprende y su empleo en métodos de protección de cultivos de plantas útiles y de protección del material de propagación de la planta contra los daños causados por nematodos. Reivindicación 1: Una forma cristalina de N-[2-(2,4-diclorofenil)ciclobutil-2-(trifluorometil)piridin-3-carboxamida de fórmula (1), caracterizada por un patrón de difracción de rayos X de polvos que comprende cuatro o más valores del ángulo 2-q seleccionados del grupo de 6.1 ± 0.2, 11.2 ± 0.2, 14.0 ± 0.2, 16.7 ± 0.2, 17.2 ± 0.2, 18.5 ± 0.2, 20.8 ± 0.2, 21.3 ± 0.2, 22.3 ± 0.2, 23.6 ± 0.2, 23.9 ± 0.2 y 24.5 ± 0.2 a una temperatura de 21 - 26ºC. Reivindicación 6: Una forma cristalina de N-[2-(2,4-diclorofenil)ciclobutil-2-(trifluorometil)piridin-3-carboxamida de fórmula (1), caracterizada por un patrón de difracción de rayos X de polvos que comprende cuatro o más valores del ángulo 2-q seleccionados del grupo de 10.8 ± 0.2, 14.5 ± 0.2, 17.5 ± 0.2, 19.0 ± 0.2, 23.5 ± 0.2, 24.5 ± 0.2, 26.0 ± 0.2, 30.2 ± 0.2, 32.6 ± 0.2, 33.3 ± 0.2, 34.1 ± 0.2 y 35.5 ± 0.2 a una temperatura de 21 - 26ºC.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP18156463 | 2018-02-13 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR114251A1 true AR114251A1 (es) | 2020-08-12 |
Family
ID=61198760
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ARP190100300A AR114251A1 (es) | 2018-02-13 | 2019-02-07 | Formas cristalinas de n-[2-(2,4-diclorofenil)ciclobutil]-2-(trifluorometl)piridin-3-carboxamida |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US11053201B2 (es) |
| EP (1) | EP3752489A1 (es) |
| JP (1) | JP7348904B2 (es) |
| KR (1) | KR20200120933A (es) |
| CN (1) | CN111741945B (es) |
| AR (1) | AR114251A1 (es) |
| AU (1) | AU2019220997B2 (es) |
| BR (1) | BR112020016431A2 (es) |
| CA (1) | CA3090960A1 (es) |
| CL (2) | CL2020002056A1 (es) |
| CO (1) | CO2020009901A2 (es) |
| EA (1) | EA202091893A1 (es) |
| EC (1) | ECSP20048382A (es) |
| IL (1) | IL276644B2 (es) |
| JO (1) | JOP20200194A1 (es) |
| MA (1) | MA51819A (es) |
| MX (1) | MX2020008367A (es) |
| PE (1) | PE20211478A1 (es) |
| PH (1) | PH12020551304A1 (es) |
| TW (1) | TWI815859B (es) |
| UY (1) | UY38085A (es) |
| WO (1) | WO2019158476A1 (es) |
| ZA (1) | ZA202004700B (es) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3853222A1 (en) * | 2018-09-19 | 2021-07-28 | Syngenta Participations Ag | Methods of controlling or preventing infestation of cereal plants by the phytopathogenic microorganism fusarium pseudograminearum |
| BR112022014935A2 (pt) * | 2020-01-30 | 2022-09-20 | Syngenta Crop Protection Ag | Métodos de controle ou prevenção do mal-do-panamá em plantas de banana |
| WO2022073797A1 (en) | 2020-10-08 | 2022-04-14 | Basf Se | Mixtures containing cyclobutrifluram |
| US20240016150A1 (en) | 2020-12-01 | 2024-01-18 | Basf Se | Mixtures containing metarylpicoxamid |
| CN112602718A (zh) * | 2020-12-15 | 2021-04-06 | 美丰农业科技(上海)有限公司 | 一种含氟唑菌酰羟胺和Cyclobutrifluram的杀线虫农用组合物 |
| CN112602721A (zh) * | 2020-12-15 | 2021-04-06 | 美丰农业科技(上海)有限公司 | 一种杀线虫农用组合物 |
| CN116634867A (zh) * | 2020-12-17 | 2023-08-22 | 先正达农作物保护股份公司 | 控制或预防植物被曲霉属的植物病原性微生物侵染的方法 |
| CN115067341B (zh) * | 2021-03-15 | 2024-03-01 | 江苏龙灯化学有限公司 | 一种杀线虫组合物 |
| CN115067343B (zh) * | 2021-03-15 | 2023-09-29 | 江苏龙灯化学有限公司 | 一种杀线虫组合物 |
| CN113615698B (zh) * | 2021-08-26 | 2023-09-15 | 青岛海利尔生物科技有限公司 | 一种杀线虫组合物及其用途 |
| CN114208839A (zh) * | 2021-12-23 | 2022-03-22 | 青岛海利尔生物科技有限公司 | 一种杀线虫组合物及其用途 |
| CN114271281B (zh) * | 2022-01-13 | 2023-05-30 | 青岛海利尔生物科技有限公司 | 一种杀线虫组合物及其应用 |
| CN114375958B (zh) * | 2022-01-24 | 2023-09-15 | 青岛海利尔生物科技有限公司 | 一种含Cyclobutrifluram的杀线虫组合物及其应用 |
| WO2024141326A1 (en) | 2022-12-30 | 2024-07-04 | Syngenta Crop Protection Ag | Compositions comprising 4-membered ring carboxamide compounds |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101125932B1 (ko) | 2006-12-06 | 2012-03-22 | 아이디유엔 파마슈티칼즈, 인코포레이티드 | (3ｓ)-3-［ｎ-(ｎ'-(2-ｔｅｒｔ-부틸페닐)옥사밀)알라니닐］아미노-5-(2',3',5',6'-테트라플루오로페녹시)-4-옥소펜탄산의 결정 형태 |
| EP2644595A1 (en) * | 2012-03-26 | 2013-10-02 | Syngenta Participations AG. | N-Cyclylamides as nematicides |
| KR102287817B1 (ko) * | 2013-07-08 | 2021-08-09 | 신젠타 파티서페이션즈 아게 | 살선충제로서 사용되는 4 원 고리 카복스아미드 |
-
2019
- 2019-02-07 AR ARP190100300A patent/AR114251A1/es unknown
- 2019-02-11 WO PCT/EP2019/053292 patent/WO2019158476A1/en active Application Filing
- 2019-02-11 KR KR1020207026056A patent/KR20200120933A/ko not_active Application Discontinuation
- 2019-02-11 US US16/969,798 patent/US11053201B2/en active Active
- 2019-02-11 JP JP2020543281A patent/JP7348904B2/ja active Active
- 2019-02-11 EP EP19704613.9A patent/EP3752489A1/en active Pending
- 2019-02-11 JO JOP/2020/0194A patent/JOP20200194A1/ar unknown
- 2019-02-11 AU AU2019220997A patent/AU2019220997B2/en active Active
- 2019-02-11 CA CA3090960A patent/CA3090960A1/en active Pending
- 2019-02-11 MX MX2020008367A patent/MX2020008367A/es unknown
- 2019-02-11 TW TW108104399A patent/TWI815859B/zh active
- 2019-02-11 EA EA202091893A patent/EA202091893A1/ru unknown
- 2019-02-11 PE PE2020001214A patent/PE20211478A1/es unknown
- 2019-02-11 MA MA051819A patent/MA51819A/fr unknown
- 2019-02-11 BR BR112020016431-3A patent/BR112020016431A2/pt unknown
- 2019-02-11 IL IL276644A patent/IL276644B2/en unknown
- 2019-02-11 CN CN201980013098.5A patent/CN111741945B/zh active Active
- 2019-02-12 UY UY38085A patent/UY38085A/es unknown
-
2020
- 2020-07-29 ZA ZA2020/04700A patent/ZA202004700B/en unknown
- 2020-08-07 CL CL2020002056A patent/CL2020002056A1/es unknown
- 2020-08-12 CO CONC2020/0009901A patent/CO2020009901A2/es unknown
- 2020-08-13 PH PH12020551304A patent/PH12020551304A1/en unknown
- 2020-08-13 EC ECSENADI202048382A patent/ECSP20048382A/es unknown
-
2022
- 2022-12-12 CL CL2022003528A patent/CL2022003528A1/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EA202091893A1 (ru) | 2020-12-22 |
| JP7348904B2 (ja) | 2023-09-21 |
| JP2021514356A (ja) | 2021-06-10 |
| KR20200120933A (ko) | 2020-10-22 |
| CL2022003528A1 (es) | 2023-06-02 |
| CA3090960A1 (en) | 2019-08-22 |
| MA51819A (fr) | 2021-05-19 |
| IL276644A (en) | 2020-09-30 |
| TWI815859B (zh) | 2023-09-21 |
| UY38085A (es) | 2019-10-01 |
| MX2020008367A (es) | 2020-09-25 |
| ZA202004700B (en) | 2021-09-29 |
| PE20211478A1 (es) | 2021-08-05 |
| AU2019220997B2 (en) | 2024-03-28 |
| BR112020016431A2 (pt) | 2020-12-15 |
| IL276644B2 (en) | 2023-11-01 |
| CO2020009901A2 (es) | 2020-08-21 |
| CL2020002056A1 (es) | 2020-10-23 |
| WO2019158476A1 (en) | 2019-08-22 |
| IL276644B1 (en) | 2023-07-01 |
| JOP20200194A1 (ar) | 2020-08-11 |
| TW202003468A (zh) | 2020-01-16 |
| CN111741945A (zh) | 2020-10-02 |
| ECSP20048382A (es) | 2020-09-30 |
| US11053201B2 (en) | 2021-07-06 |
| US20200369614A1 (en) | 2020-11-26 |
| AU2019220997A1 (en) | 2020-09-03 |
| CN111741945B (zh) | 2024-01-09 |
| PH12020551304A1 (en) | 2021-08-16 |
| EP3752489A1 (en) | 2020-12-23 |
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