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NO20060091L - Anvendelse av kondenserte heterocykliske forbindelser som SCCE-inhibitorer for behandling av hudproblemer eller kreft - Google Patents

Anvendelse av kondenserte heterocykliske forbindelser som SCCE-inhibitorer for behandling av hudproblemer eller kreft

Info

Publication number
NO20060091L
NO20060091L NO20060091A NO20060091A NO20060091L NO 20060091 L NO20060091 L NO 20060091L NO 20060091 A NO20060091 A NO 20060091A NO 20060091 A NO20060091 A NO 20060091A NO 20060091 L NO20060091 L NO 20060091L
Authority
NO
Norway
Prior art keywords
cancer
treatment
skin problems
scce
condensed heterocycles
Prior art date
Application number
NO20060091A
Other languages
English (en)
Inventor
Marcel Linschoten
Original Assignee
Arexis Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Arexis Ab filed Critical Arexis Ab
Publication of NO20060091L publication Critical patent/NO20060091L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/536—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with carbocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/04—Antipruritics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/10—Anti-acne agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/12—Keratolytics, e.g. wart or anti-corn preparations
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Cosmetics (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Det beskrives heterosykliske inhibitorer av stratumcorneurnkymotryptisk enzym (SCCE). Mer spesielt beskrives anvendelsen av forbindelser med formel (I) eller (II) for behandling av visse sykdommer og særlig hudsykdommer som pruritt og også cancer som ovariecancer.
NO20060091A 2003-06-06 2006-01-06 Anvendelse av kondenserte heterocykliske forbindelser som SCCE-inhibitorer for behandling av hudproblemer eller kreft NO20060091L (no)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
DKPA200300844 2003-06-06
DKPA200300843 2003-06-06
DKPA200300842 2003-06-06
DKPA200300840 2003-06-06
PCT/DK2004/000388 WO2004108139A2 (en) 2003-06-06 2004-06-07 Use of fused heterocyclic compounds as scce inhibitors for the treatment of skin conditions or cancer

Publications (1)

Publication Number Publication Date
NO20060091L true NO20060091L (no) 2006-03-06

Family

ID=33514772

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20060091A NO20060091L (no) 2003-06-06 2006-01-06 Anvendelse av kondenserte heterocykliske forbindelser som SCCE-inhibitorer for behandling av hudproblemer eller kreft

Country Status (18)

Country Link
US (1) US7872052B2 (no)
EP (1) EP1631295B1 (no)
JP (1) JP5044214B2 (no)
KR (2) KR101099409B1 (no)
CN (1) CN101152185B (no)
AT (1) ATE459359T1 (no)
CA (1) CA2525383C (no)
CY (1) CY1110084T1 (no)
DE (1) DE602004025803D1 (no)
DK (1) DK1631295T3 (no)
ES (1) ES2341545T3 (no)
HK (2) HK1091731A1 (no)
NO (1) NO20060091L (no)
NZ (1) NZ543636A (no)
PL (1) PL1631295T3 (no)
PT (1) PT1631295E (no)
SI (1) SI1631295T1 (no)
WO (1) WO2004108139A2 (no)

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Also Published As

Publication number Publication date
PT1631295E (pt) 2010-05-24
CN101152185A (zh) 2008-04-02
US7872052B2 (en) 2011-01-18
EP1631295B1 (en) 2010-03-03
CA2525383A1 (en) 2004-12-16
DK1631295T3 (da) 2010-06-21
KR101205257B1 (ko) 2012-11-27
HK1091731A1 (en) 2007-01-26
KR101099409B1 (ko) 2011-12-27
CY1110084T1 (el) 2015-01-14
KR20060008331A (ko) 2006-01-26
DE602004025803D1 (de) 2010-04-15
AU2004244704A1 (en) 2004-12-16
CN101152185B (zh) 2010-12-08
WO2004108139A8 (en) 2005-04-28
NZ543636A (en) 2009-07-31
WO2004108139A3 (en) 2005-03-10
JP5044214B2 (ja) 2012-10-10
CA2525383C (en) 2012-03-06
ATE459359T1 (de) 2010-03-15
PL1631295T3 (pl) 2010-09-30
JP2006526581A (ja) 2006-11-24
SI1631295T1 (sl) 2010-06-30
ES2341545T3 (es) 2010-06-22
US20060258651A1 (en) 2006-11-16
WO2004108139A2 (en) 2004-12-16
EP1631295A2 (en) 2006-03-08
KR20110120960A (ko) 2011-11-04
HK1120209A1 (en) 2009-03-27

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