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MXPA03010142A - Novel arylheteroalkylamine derivatives. - Google Patents

Novel arylheteroalkylamine derivatives.

Info

Publication number
MXPA03010142A
MXPA03010142A MXPA03010142A MXPA03010142A MXPA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A MX PA03010142 A MXPA03010142 A MX PA03010142A
Authority
MX
Mexico
Prior art keywords
arylheteroalkylamine
derivatives
novel
compounds
racemates
Prior art date
Application number
MXPA03010142A
Other languages
Spanish (es)
Inventor
Tim Brikinshaw
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE0101617A external-priority patent/SE0101617D0/en
Priority claimed from SE0103271A external-priority patent/SE0103271D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of MXPA03010142A publication Critical patent/MXPA03010142A/en

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    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
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Abstract

There are provided novel compounds of formula (I) wherein R1, R2, R3, R4, R5, R6, T, U, X, Y, V and W are as defined in the specification, and pharmaceutically acceptable salts thereof, and enantiomers and racemates thereof; together with processes for their preparation, compositions containing them and their use in therapy. The compounds are inhibitors of nitric oxide synthase and are thereby particularly useful in the treatment or prophylaxis of inflammatory disease and pain.
MXPA03010142A 2001-05-08 2002-05-06 Novel arylheteroalkylamine derivatives. MXPA03010142A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SE0101617A SE0101617D0 (en) 2001-05-08 2001-05-08 Novel compounds
SE0103271A SE0103271D0 (en) 2001-09-28 2001-09-28 Novel compounds
PCT/SE2002/000876 WO2002090332A2 (en) 2001-05-08 2002-05-06 Novel aeylheteroalkylaminε derivatives

Publications (1)

Publication Number Publication Date
MXPA03010142A true MXPA03010142A (en) 2004-03-10

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ID=26655458

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Application Number Title Priority Date Filing Date
MXPA03010142A MXPA03010142A (en) 2001-05-08 2002-05-06 Novel arylheteroalkylamine derivatives.

Country Status (15)

Country Link
US (1) US20040242871A1 (en)
EP (1) EP1572655A2 (en)
JP (1) JP2005506308A (en)
KR (1) KR20030096361A (en)
CN (1) CN100340548C (en)
AR (1) AR035700A1 (en)
AU (1) AU2002306039B2 (en)
BR (1) BR0209518A (en)
CA (1) CA2446120A1 (en)
IL (1) IL158388A0 (en)
MX (1) MXPA03010142A (en)
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US20040242871A1 (en) 2004-12-02
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WO2002090332A2 (en) 2002-11-14
AU2002306039B2 (en) 2008-05-29
BR0209518A (en) 2004-07-13
KR20030096361A (en) 2003-12-24
CA2446120A1 (en) 2002-11-14
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WO2002090332A3 (en) 2007-11-01
IL158388A0 (en) 2004-05-12

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