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MX2022009871A - Compuestos tetraciclicos para tratar la infeccion por el virus de la inmunodeficiencia humana (vih). - Google Patents

Compuestos tetraciclicos para tratar la infeccion por el virus de la inmunodeficiencia humana (vih).

Info

Publication number
MX2022009871A
MX2022009871A MX2022009871A MX2022009871A MX2022009871A MX 2022009871 A MX2022009871 A MX 2022009871A MX 2022009871 A MX2022009871 A MX 2022009871A MX 2022009871 A MX2022009871 A MX 2022009871A MX 2022009871 A MX2022009871 A MX 2022009871A
Authority
MX
Mexico
Prior art keywords
compounds
hiv infection
treating hiv
tetracyclic compounds
pharmaceutical compositions
Prior art date
Application number
MX2022009871A
Other languages
English (en)
Inventor
Michael L Mitchell
Lan Jiang
David W Lin
Gregg M Schwarzwalder
Ezra Roberts
Original Assignee
Gilead Sciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Gilead Sciences Inc filed Critical Gilead Sciences Inc
Publication of MX2022009871A publication Critical patent/MX2022009871A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/22—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed systems contains four or more hetero rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Molecular Biology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

La presente descripción se refiere en general a ciertos compuestos tetracíclicos, composiciones farmacéuticas que comprenden los compuestos y métodos para preparar los compuestos y composiciones farmacéuticas. Los compuestos de la descripción son útiles para tratar o prevenir la infección por el virus de la inmunodeficiencia humana (VIH). (ver Fórmula).
MX2022009871A 2020-02-24 2021-02-23 Compuestos tetraciclicos para tratar la infeccion por el virus de la inmunodeficiencia humana (vih). MX2022009871A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US202062980857P 2020-02-24 2020-02-24
US202063036268P 2020-06-08 2020-06-08
US202063128670P 2020-12-21 2020-12-21
PCT/US2021/019179 WO2021173522A1 (en) 2020-02-24 2021-02-23 Tetracyclic compounds for treating hiv infection

Publications (1)

Publication Number Publication Date
MX2022009871A true MX2022009871A (es) 2022-08-19

Family

ID=74885056

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2022009871A MX2022009871A (es) 2020-02-24 2021-02-23 Compuestos tetraciclicos para tratar la infeccion por el virus de la inmunodeficiencia humana (vih).

Country Status (15)

Country Link
US (2) US11697652B2 (es)
EP (1) EP4110783A1 (es)
JP (2) JP7453399B2 (es)
CN (1) CN115151545A (es)
AU (2) AU2021225809B2 (es)
BR (1) BR112022015771A2 (es)
CA (1) CA3166480A1 (es)
CO (1) CO2022011947A2 (es)
CR (1) CR20220418A (es)
DO (1) DOP2022000171A (es)
IL (1) IL295677A (es)
MX (1) MX2022009871A (es)
PE (1) PE20221569A1 (es)
TW (2) TW202248199A (es)
WO (1) WO2021173522A1 (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
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CN115151545A (zh) 2022-10-04
BR112022015771A2 (pt) 2022-10-11
CO2022011947A2 (es) 2022-08-30
CR20220418A (es) 2022-10-10
US20240010650A1 (en) 2024-01-11
TW202248199A (zh) 2022-12-16
TWI777425B (zh) 2022-09-11
JP2023184696A (ja) 2023-12-28
TW202140481A (zh) 2021-11-01
AU2021225809B2 (en) 2023-08-24
PE20221569A1 (es) 2022-10-06
IL295677A (en) 2022-10-01
EP4110783A1 (en) 2023-01-04
JP7453399B2 (ja) 2024-03-19
AU2023266279A1 (en) 2023-12-07
WO2021173522A1 (en) 2021-09-02
CA3166480A1 (en) 2021-09-02
JP2023514635A (ja) 2023-04-06
AU2021225809A1 (en) 2022-10-13
DOP2022000171A (es) 2022-10-16
US11697652B2 (en) 2023-07-11
US12122776B2 (en) 2024-10-22
US20210284642A1 (en) 2021-09-16

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