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MX2019002629A - Formas cristalinas de compuestos terapéuticos y usos de los mismos. - Google Patents

Formas cristalinas de compuestos terapéuticos y usos de los mismos.

Info

Publication number
MX2019002629A
MX2019002629A MX2019002629A MX2019002629A MX2019002629A MX 2019002629 A MX2019002629 A MX 2019002629A MX 2019002629 A MX2019002629 A MX 2019002629A MX 2019002629 A MX2019002629 A MX 2019002629A MX 2019002629 A MX2019002629 A MX 2019002629A
Authority
MX
Mexico
Prior art keywords
crystalline forms
therapeutic compounds
kits
disease
prevention
Prior art date
Application number
MX2019002629A
Other languages
English (en)
Inventor
Ngoc NGUYEN Minh
Zapanta Ong Winston
Original Assignee
Kala Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kala Pharmaceuticals Inc filed Critical Kala Pharmaceuticals Inc
Publication of MX2019002629A publication Critical patent/MX2019002629A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Se describen en la presente formas cristalinas del Compuesto 1 útiles para la prevención y el tratamiento de afecciones oculares angiogénicas; métodos para tratar una enfermedad que comprende; procesos de preparación; y equipos que comprenden, el mismo.
MX2019002629A 2016-09-08 2017-09-01 Formas cristalinas de compuestos terapéuticos y usos de los mismos. MX2019002629A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662385148P 2016-09-08 2016-09-08
PCT/US2017/049914 WO2018048746A1 (en) 2016-09-08 2017-09-01 Crystalline forms of therapeutic compounds and uses thereof

Publications (1)

Publication Number Publication Date
MX2019002629A true MX2019002629A (es) 2019-10-07

Family

ID=61281989

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2019002629A MX2019002629A (es) 2016-09-08 2017-09-01 Formas cristalinas de compuestos terapéuticos y usos de los mismos.

Country Status (10)

Country Link
US (5) US10336767B2 (es)
EP (1) EP3509421A4 (es)
JP (1) JP2019533641A (es)
KR (1) KR20190051010A (es)
CN (1) CN109688818A (es)
AU (2) AU2017324251A1 (es)
BR (1) BR112019004463A2 (es)
CA (1) CA3036065A1 (es)
MX (1) MX2019002629A (es)
WO (1) WO2018048746A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX2019002629A (es) * 2016-09-08 2019-10-07 Kala Pharmaceuticals Inc Formas cristalinas de compuestos terapéuticos y usos de los mismos.

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AU2020217446B2 (en) 2022-05-26
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US20180065977A1 (en) 2018-03-08
US20200216460A1 (en) 2020-07-09
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