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MA32224B1 - Derives de (pyrazolyl-carbonyl) imidazolidinone pour le traitement de maladies retrovirales - Google Patents

Derives de (pyrazolyl-carbonyl) imidazolidinone pour le traitement de maladies retrovirales

Info

Publication number
MA32224B1
MA32224B1 MA33241A MA33241A MA32224B1 MA 32224 B1 MA32224 B1 MA 32224B1 MA 33241 A MA33241 A MA 33241A MA 33241 A MA33241 A MA 33241A MA 32224 B1 MA32224 B1 MA 32224B1
Authority
MA
Morocco
Prior art keywords
treatment
carbonyl
pyrazolyl
diseases
retroviral diseases
Prior art date
Application number
MA33241A
Other languages
Arabic (ar)
English (en)
Inventor
Kai Thede
Susanne Greschat
Steffen Wildum
Daniela Paulsen
Original Assignee
Aicuris Gmbh & Co Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aicuris Gmbh & Co Kg filed Critical Aicuris Gmbh & Co Kg
Publication of MA32224B1 publication Critical patent/MA32224B1/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Health & Medical Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La présente invention concerne de nouvelles (pyrazolyl-carbonyl)imidazolidinones (i) substituées, leur procédé de fabrication, leur utilisation pour le traitement et/ou la prophylaxie de maladies, ainsi que leur utilisation pour la préparation de médicaments pour le traitement et/ou la prophylaxie de maladies, en particulier de maladies rétrovirales, chez l'homme et/ou l'animal.
MA33241A 2008-03-17 2010-10-11 Derives de (pyrazolyl-carbonyl) imidazolidinone pour le traitement de maladies retrovirales MA32224B1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE102008015033A DE102008015033A1 (de) 2008-03-17 2008-03-17 Substituierte (Pyrazolyl-carbonyl)imidazolidinone und ihre Verwendung
PCT/EP2009/001714 WO2009115213A1 (fr) 2008-03-17 2009-03-10 Dérivés de (pyrazolyl-carbonyl)imidazolidinone pour le traitement de maladies rétrovirales

Publications (1)

Publication Number Publication Date
MA32224B1 true MA32224B1 (fr) 2011-04-01

Family

ID=40565083

Family Applications (1)

Application Number Title Priority Date Filing Date
MA33241A MA32224B1 (fr) 2008-03-17 2010-10-11 Derives de (pyrazolyl-carbonyl) imidazolidinone pour le traitement de maladies retrovirales

Country Status (22)

Country Link
US (1) US8399682B2 (fr)
EP (1) EP2254885B1 (fr)
JP (1) JP5576853B2 (fr)
KR (1) KR20100124337A (fr)
CN (1) CN101977908B (fr)
AP (1) AP2774A (fr)
AR (1) AR070919A1 (fr)
AU (1) AU2009226656A1 (fr)
CA (1) CA2718685C (fr)
CL (1) CL2009000636A1 (fr)
DE (1) DE102008015033A1 (fr)
IL (1) IL207649A0 (fr)
MA (1) MA32224B1 (fr)
MX (1) MX2010010230A (fr)
NZ (1) NZ588141A (fr)
PE (1) PE20091718A1 (fr)
RU (1) RU2010141578A (fr)
TW (1) TW200951125A (fr)
UA (1) UA102390C2 (fr)
UY (1) UY31717A1 (fr)
WO (1) WO2009115213A1 (fr)
ZA (1) ZA201007361B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102008015033A1 (de) 2008-03-17 2009-09-24 Aicuris Gmbh & Co. Kg Substituierte (Pyrazolyl-carbonyl)imidazolidinone und ihre Verwendung
DE102008015032A1 (de) * 2008-03-17 2009-09-24 Aicuris Gmbh & Co. Kg Substituierte Pyrazolamide und ihre Verwendung
DE102008062878A1 (de) 2008-12-17 2010-06-24 Aicuris Gmbh & Co. Kg Substituierte Furancarboxamide und ihre Verwendung
DE102008062863A1 (de) 2008-12-17 2010-06-24 Aicuris Gmbh & Co. Kg Substituierte (Thiophenyl-carbonyl)imidazolidinone und ihre Verwendung
EP2295038B1 (fr) * 2009-09-11 2013-05-29 AiCuris GmbH & Co. KG Dispersion solide comprenant un agent anti-VIH
DE102011055815A1 (de) 2011-11-29 2013-05-29 Aicuris Gmbh & Co. Kg Carboxamid-substituierte Heteroaryl-Pyrazole und ihre Verwendung
DE102012016908A1 (de) 2012-08-17 2014-02-20 Aicuris Gmbh & Co. Kg Tris-(Hetero)Aryl-Pyrazole und ihre Verwendung

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US5571810A (en) * 1990-06-11 1996-11-05 Fujisawa Pharmaceutical Co., Ltd. Thiophene derivatives
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FR2692575B1 (fr) 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
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FR2728571B1 (fr) * 1994-12-22 1997-01-31 Adir Nouveaux ethers d'oximes tricycliques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
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WO2003014107A1 (fr) 2001-08-01 2003-02-20 Basell Polyolefine Gmbh Procede de preparation de derives heterocycliques de pentalene
EP1451160B1 (fr) 2001-11-01 2010-01-13 Icagen, Inc. Pyrazole-amides pour utilisation dans le traitement de la douleur
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Also Published As

Publication number Publication date
NZ588141A (en) 2012-05-25
AP2774A (en) 2013-09-30
KR20100124337A (ko) 2010-11-26
WO2009115213A1 (fr) 2009-09-24
CA2718685A1 (fr) 2009-09-24
AP2010005422A0 (en) 2010-10-31
US8399682B2 (en) 2013-03-19
ZA201007361B (en) 2011-12-28
TW200951125A (en) 2009-12-16
PE20091718A1 (es) 2009-12-11
JP2011514366A (ja) 2011-05-06
CN101977908A (zh) 2011-02-16
JP5576853B2 (ja) 2014-08-20
UA102390C2 (ru) 2013-07-10
DE102008015033A1 (de) 2009-09-24
MX2010010230A (es) 2010-11-09
RU2010141578A (ru) 2012-04-27
EP2254885B1 (fr) 2013-12-04
AU2009226656A1 (en) 2009-09-24
CL2009000636A1 (es) 2010-05-07
US20110124618A1 (en) 2011-05-26
CN101977908B (zh) 2014-04-23
CA2718685C (fr) 2016-11-29
AR070919A1 (es) 2010-05-12
IL207649A0 (en) 2010-12-30
EP2254885A1 (fr) 2010-12-01
UY31717A1 (es) 2009-08-31

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