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Schisandrin B shows neuroprotective effect in 6-OHDA-induced Parkinson's disease via inhibiting the negative modulation of miR-34a on Nrf2 pathway

Biomed Pharmacother. 2015 Oct:75:165-72. doi: 10.1016/j.biopha.2015.07.034. Epub 2015 Aug 15.

Abstract

Background: MiR-34 family members have been previously shown to play potential functional role in Parkinson's disease (PD) pathogenesis. However, the regulatory role of miR-34a has not been demonstrated in PD yet. This study aims to clarify the potential neuroprotective effect of Schisandrin B (Sch B) involving miR-34a function in 6-OHDA-induced PD model.

Methods: The expression changes of miR-34a and Nrf2 pathway related genes were detected in 6-OHDA-treated SH-SY5Y cells under Sch B pretreatment. Cell viability and PD feathers of 6-OHDA-induced PD mice were measured for neuroprotection assessment. The regulation of miR-34a on Nrf2 activity and expression was demonstrated through gain-of-function and loss-of-function studies, while the regulatory role of miR-34a in the neuroprotection of Sch B was investigated both in vitro and in vivo.

Results: Sch B pretreatment ameliorated 6-OHDA-induced changes in vitro, like upregulated miR-34a expression, inhibited Nrf2 pathways and decreased cell survival, and PD feathers in vivo. Moreover, Nrf2 was negatively regulated by miR-34a, while miR-34a overexpression inhibited the neuroprotection of Sch B in both dopaminergic SH-SY5Y cells and PD mice.

Conclusion: Sch B showed neuroprotective effect in 6-OHDA-induced PD pathogenesis, which could be inhibited by miR-34a, involving the negative regulatory mechanism of miR-34a on Nrf2 pathways.

Keywords: 6-OHDA; MiR-34a; Nrf2; Parkinson’s disease; Schisandrin B.

MeSH terms

  • 3' Untranslated Regions
  • Animals
  • Behavior, Animal
  • Binding Sites
  • Brain / drug effects*
  • Brain / metabolism
  • Brain / pathology
  • Cell Line, Tumor
  • Cell Survival / drug effects
  • Cyclooctanes / pharmacology
  • Disease Models, Animal
  • Humans
  • Lignans / pharmacology*
  • Male
  • Mice, Inbred C57BL
  • MicroRNAs / genetics*
  • MicroRNAs / metabolism
  • Motor Activity / drug effects
  • NF-E2-Related Factor 2 / genetics*
  • NF-E2-Related Factor 2 / metabolism
  • Neurons / drug effects*
  • Neurons / metabolism
  • Neurons / pathology
  • Neuroprotective Agents / pharmacology*
  • Oxidopamine*
  • Parkinsonian Disorders / genetics
  • Parkinsonian Disorders / metabolism
  • Parkinsonian Disorders / pathology
  • Parkinsonian Disorders / prevention & control*
  • Polycyclic Compounds / pharmacology*
  • Signal Transduction / drug effects
  • Transfection

Substances

  • 3' Untranslated Regions
  • Cyclooctanes
  • Lignans
  • MIRN34 microRNA, human
  • MIRN34a microRNA, mouse
  • MicroRNAs
  • NF-E2-Related Factor 2
  • NFE2L2 protein, human
  • Neuroprotective Agents
  • Nfe2l2 protein, mouse
  • Polycyclic Compounds
  • schizandrin B
  • Oxidopamine