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WO2010015680A1 - Dérivés fongicides de l'oxyalkylamide - Google Patents

Dérivés fongicides de l'oxyalkylamide Download PDF

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Publication number
WO2010015680A1
WO2010015680A1 PCT/EP2009/060219 EP2009060219W WO2010015680A1 WO 2010015680 A1 WO2010015680 A1 WO 2010015680A1 EP 2009060219 W EP2009060219 W EP 2009060219W WO 2010015680 A1 WO2010015680 A1 WO 2010015680A1
Authority
WO
WIPO (PCT)
Prior art keywords
substituted
alkyl
halogen atoms
group
tri
Prior art date
Application number
PCT/EP2009/060219
Other languages
English (en)
Inventor
Pierre-Yves Coqueron
Mazen Es-Sayed
Marie-Claire Grosjean-Cournoyer
Philippe Meresse
Oswald Ort
Nicola Rahn
Valérie TOQUIN
Arounarith Tuch
Jacky Vidal
Ulrike Wachendorff-Neumann
Original Assignee
Bayer Cropscience Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Sa filed Critical Bayer Cropscience Sa
Publication of WO2010015680A1 publication Critical patent/WO2010015680A1/fr

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20—Oxygen atoms

Definitions

  • any of the compounds according to the invention can exist as one or more stereoisomers depending on the number of stereogenic units (as defined by the IUPAC rules) in the compound.
  • the invention thus relates equally to all the stereoisomers, and to the mixtures of all the possible stereoisomers, in all proportions.
  • the stereoisomers can be separated according to the methods which are known per se by the man ordinary skilled in the art.
  • R 3 represents -(CR a R b )p-R 4 and:
  • the palladium complex is directly generated in the reaction mixture by separately adding to the reaction mixture a palladium salt and a complex ligand such as a phosphine, for example triethylphosphine, tri-tert-butylphosphine, tricyclohexylphosphine, 2- (dicyclohexylphosphine)biphenyl, 2-(di-tert-butylphosphin)biphenyl, 2-
  • a complex ligand such as a phosphine, for example triethylphosphine, tri-tert-butylphosphine, tricyclohexylphosphine, 2- (dicyclohexylphosphine)biphenyl, 2-(di-tert-butylphosphin)biphenyl, 2-
  • additional components can also be included, e.g. protective colloids, adhesives, thickeners, thixotropic agents, penetration agents, stabilisers, sequestering agents.
  • the active compounds can be combined with any solid or liquid additive, that complies with the usual formulation techniques.
  • compositions according to the invention can be used in various forms such as aerosol dispenser, capsule suspension, cold fogging concentrate, dustable powder, emulsifiable concentrate, emulsion oil in water, emulsion water in oil, encapsulated granule, fine granule, flowable concentrate for seed treatment, gas (under pressure), gas generating product, granule, hot fogging concentrate, macrogranule, microgranule, oil dispersible powder, oil miscible flowable concentrate, oil miscible liquid, paste, plant rodlet, powder for dry seed treatment, seed coated with a pesticide, soluble concentrate, soluble powder, solution for seed treatment, suspension concentrate (flowable concentrate), ultra low volume (ULV) liquid, ultra low volume (ULV) suspension, water dispersible granules or tablets, water dispersible powder for slurry treatment, water soluble granules or tablets, water soluble powder for seed treatment and wettable powder.
  • These compositions include not only compositions that are ready to be applied to the plant or seed to
  • Inhibitors of the nucleic acid synthesis for example benalaxyl, benalaxyl-M, bupirimate, clozylacon, dimethirimol, ethirimol, furalaxyl, hymexazol, metalaxyl, metalaxyl-M, ofurace, oxadixyl and oxolinic acid.
  • plants which contain a stress tolerance enhancing transgene coding for a plant-functional enzyme of the nicotinamide adenine dinucleotide salvage synthesis pathway including nicotinamidase, nicotinate phosphoribosyltransferase, nicotinic acid mononucleotide adenyl transferase, nicotinamide adenine dinucleotide synthetase or nicotine amide phosphoribosyltransferase as described e.g. in WO2006/032469 or WO 2006/133827 or PCT/EP07/002433.
  • Blumeria diseases caused for example by Blumeha graminis ;
  • Podosphaera diseases caused for example by Podosphaera leucothcha ;
  • Sphaerotheca diseases caused for example by Sphaerotheca fuliginea ;
  • Uncinula diseases caused for example by Uncinula necator ;
  • Puccinia diseases caused for example by Puccinia recondita ;
  • Penicillium diseases caused for example by Penicillium expansum ; Rhizopus diseases caused by example by Rhizopus stolonifer Sclerotinia diseases, caused for example by Sclerotinia sclerotiorum ; Verticilium diseases, caused for example by Verticilium alboatrum ; • Seed and soil borne decay, mould, wilt, rot and damping-off diseases such as :
  • Alternaria diseases caused for example by Alternaria brassicicola Aphanomyces diseases, caused for example by Aphanomyces euteiches Ascochyta diseases, caused for example by Ascochyta lentis Aspergillus diseases, caused for example by Aspergillus flavus Cladosporium diseases, caused for example by Cladosporium herbarum
  • the fungicide composition according to the invention can also be used in the treatment of genetically modified organisms with the compounds according to the invention or the agrochemical compositions according to the invention.
  • Genetically modified plants are plants into genome of that a heterologous gene encoding a protein of interest has been stably integrated.
  • the expression "heterologous gene encoding a protein of interest” essentially means genes that give the transformed plant new agronomic properties, or genes for improving the agronomic quality of the modified plant.
  • the compounds tested are solubilized in DMSO and added to sterile liquid glucose/mycopeptone medium (14.6 g/l of D-glucose, 7.1 g/l of mycological peptone (Oxoid) and 1.4 g/l of yeast extract (Merck)) at a concentration of 2 ppm.
  • the medium is inoculated with cryopreserved Botrytis cinerea spore suspension at a concentration of 500 spores per ml.
  • the efficacy of the active ingredient is assessed by OD measurement at 620 nm after 5 days at 2O 0 C in comparison with a control.

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

La présente invention concerne des dérivés fongicides de l'oxyalkylamide de la formule (I), leur procédé de préparation, leur utilisation en tant que fongicides, en particulier sous la forme de compositions fongicides, et des procédés pour la lutte contre les champignons phytopathogènes de plantes à l'aide de ces composés ou de leurs compositions. Dans la formule (I), Q1 à Q3, R1 à R3 et L représentent différents substituants.
PCT/EP2009/060219 2008-08-07 2009-08-06 Dérivés fongicides de l'oxyalkylamide WO2010015680A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08356118 2008-08-07
EP08356118.3 2008-08-07

Publications (1)

Publication Number Publication Date
WO2010015680A1 true WO2010015680A1 (fr) 2010-02-11

Family

ID=40210567

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/EP2009/060219 WO2010015680A1 (fr) 2008-08-07 2009-08-06 Dérivés fongicides de l'oxyalkylamide

Country Status (2)

Country Link
AR (1) AR073049A1 (fr)
WO (1) WO2010015680A1 (fr)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20140045890A1 (en) * 2011-03-31 2014-02-13 Syngenta Participations Ag Novel compounds
WO2020245044A1 (fr) * 2019-06-03 2020-12-10 Bayer Aktiengesellschaft Acides 1-phényl-5-azinylpyrazolyl-3-oxyalkyliques et leur utilisation pour lutter contre la croissance de plantes adventices

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004039764A1 (fr) * 2002-10-31 2004-05-13 Boehringer Ingelheim Pharma Gmbh & Co. Kg Nouveaux composes de type amide exerçant une action antagoniste sur l'hormone mch, et medicaments contenant ces composes
WO2004047538A1 (fr) * 2002-11-26 2004-06-10 Syngenta Limited Oxyalkylamides de quinoline, d'isoquinoline et de quinazoline et leur utilisation comme fongicides
WO2004108663A1 (fr) * 2003-06-04 2004-12-16 Syngenta Limited Derives de n-alkynyle-2- (substitue aryloxy) alkylthioamide comme fongicides
WO2008028624A1 (fr) * 2006-09-06 2008-03-13 Syngenta Participations Ag Fongicides
WO2008110355A1 (fr) * 2007-03-14 2008-09-18 Syngenta Participations Ag Dérivés de quinoléine en tant que fongicides

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004039764A1 (fr) * 2002-10-31 2004-05-13 Boehringer Ingelheim Pharma Gmbh & Co. Kg Nouveaux composes de type amide exerçant une action antagoniste sur l'hormone mch, et medicaments contenant ces composes
WO2004047538A1 (fr) * 2002-11-26 2004-06-10 Syngenta Limited Oxyalkylamides de quinoline, d'isoquinoline et de quinazoline et leur utilisation comme fongicides
WO2004108663A1 (fr) * 2003-06-04 2004-12-16 Syngenta Limited Derives de n-alkynyle-2- (substitue aryloxy) alkylthioamide comme fongicides
WO2008028624A1 (fr) * 2006-09-06 2008-03-13 Syngenta Participations Ag Fongicides
WO2008110355A1 (fr) * 2007-03-14 2008-09-18 Syngenta Participations Ag Dérivés de quinoléine en tant que fongicides

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20140045890A1 (en) * 2011-03-31 2014-02-13 Syngenta Participations Ag Novel compounds
WO2020245044A1 (fr) * 2019-06-03 2020-12-10 Bayer Aktiengesellschaft Acides 1-phényl-5-azinylpyrazolyl-3-oxyalkyliques et leur utilisation pour lutter contre la croissance de plantes adventices
CN114071999A (zh) * 2019-06-03 2022-02-18 拜耳公司 1-苯基-5-吖嗪基吡唑基-3-氧基烷基酸及其用于控制不需要的植物生长的用途
CN114071999B (zh) * 2019-06-03 2024-08-27 拜耳公司 1-苯基-5-吖嗪基吡唑基-3-氧基烷基酸及其用于控制不需要的植物生长的用途
US12180187B2 (en) 2019-06-03 2024-12-31 Bayer Aktiengesellschaft 1-phenyl-5-azinylpyrazolyl-3-oxyalkyl acids and their use for controlling unwanted plant growth

Also Published As

Publication number Publication date
AR073049A1 (es) 2010-10-13

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