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WO2009051956A3 - Pyrazole-substituted isoxazoline insecticides - Google Patents

Pyrazole-substituted isoxazoline insecticides Download PDF

Info

Publication number
WO2009051956A3
WO2009051956A3 PCT/US2008/078374 US2008078374W WO2009051956A3 WO 2009051956 A3 WO2009051956 A3 WO 2009051956A3 US 2008078374 W US2008078374 W US 2008078374W WO 2009051956 A3 WO2009051956 A3 WO 2009051956A3
Authority
WO
WIPO (PCT)
Prior art keywords
cyano
pyrazole
och2cf3
ocf3
cyclopropyl
Prior art date
Application number
PCT/US2008/078374
Other languages
French (fr)
Other versions
WO2009051956A2 (en
Inventor
Caleb William Holyoke Jr
George Philip Lahm
Andrew Edmund Taggi
Original Assignee
Du Pont
Caleb William Holyoke Jr
George Philip Lahm
Andrew Edmund Taggi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Du Pont, Caleb William Holyoke Jr, George Philip Lahm, Andrew Edmund Taggi filed Critical Du Pont
Publication of WO2009051956A2 publication Critical patent/WO2009051956A2/en
Publication of WO2009051956A3 publication Critical patent/WO2009051956A3/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Disclosed are compounds of Formula (1), including all stereoisomers, N-oxides, and salts thereof, wherein R1 is F, Cl, Br, CF3, OCHF2, OCF3 or OCH2CF3; R2 is H, F, Cl, Br, CH3, cyano, CF3, CHF2, OHCF2, OCF3 or OCH2CF3; R3 is H, F, Cl, Br or CF3; R4 is cyano or C(S)NH2; R5 is F, Cl, Br, I, cyano, C(S)NH2 or C(O)NHR6; and R6 is H; or R6 is C1-C3 alkyl, cyclopropyl or cyclopropylmethyl, each optionally substituted with halogen and further optionally substituted with 1 or 2 CH3; or R6 is l-(trifluoromethyl)cyclopropyl. Also disclosed are compositions containing the compounds of Formula (1) and methods for controlling an invertebrate pest comprising contacting the invertebrate pest or its environment with a biologically effective amount of a compound or a composition of the invention.
PCT/US2008/078374 2007-10-16 2008-10-01 Pyrazole-substituted isoxazoline insecticides WO2009051956A2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US99909207P 2007-10-16 2007-10-16
US60/999,092 2007-10-16

Publications (2)

Publication Number Publication Date
WO2009051956A2 WO2009051956A2 (en) 2009-04-23
WO2009051956A3 true WO2009051956A3 (en) 2009-07-30

Family

ID=40029311

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2008/078374 WO2009051956A2 (en) 2007-10-16 2008-10-01 Pyrazole-substituted isoxazoline insecticides

Country Status (1)

Country Link
WO (1) WO2009051956A2 (en)

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CN104023535A (en) 2011-09-02 2014-09-03 巴斯夫欧洲公司 Use of pesticidal active 3-arylquinazolin-4-one derivatives in soil application methods
KR20140063757A (en) 2011-09-02 2014-05-27 바스프 에스이 Insecticidal active mixtures comprising arylquinazolinone compounds
MX2014006973A (en) 2011-12-23 2014-08-01 Basf Se Isothiazoline compounds for combating invertebrate pests.
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AR111260A1 (en) 2017-03-31 2019-06-19 Intervet Int Bv PHARMACEUTICAL FORMULATION OF THE CROTONIL AMINO PIRIDINA SALT
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Citations (2)

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Patent Citations (2)

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WO2007075459A2 (en) * 2005-12-16 2007-07-05 E. I. Du Pont De Nemours And Company 5-aryl isoxazolines for controlling invertebrate pests
WO2008019760A1 (en) * 2006-08-15 2008-02-21 Bayer Cropscience Ag Insecticidal isoxazolines

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