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WO2007072201A3 - 3-aminocyclopentanecarboxamides as modulators of chemokine receptors - Google Patents

3-aminocyclopentanecarboxamides as modulators of chemokine receptors Download PDF

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Publication number
WO2007072201A3
WO2007072201A3 PCT/IB2006/003739 IB2006003739W WO2007072201A3 WO 2007072201 A3 WO2007072201 A3 WO 2007072201A3 IB 2006003739 W IB2006003739 W IB 2006003739W WO 2007072201 A3 WO2007072201 A3 WO 2007072201A3
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WO
WIPO (PCT)
Prior art keywords
modulators
aminocyclopentanecarboxamides
chemokine receptors
chemokine
compounds
Prior art date
Application number
PCT/IB2006/003739
Other languages
French (fr)
Other versions
WO2007072201A2 (en
Inventor
Chu-Biao Xue
Original Assignee
Incyte Corp
Chu-Biao Xue
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38126410&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=WO2007072201(A3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority to MEP-10/08A priority Critical patent/MEP1008A/en
Priority to AP2008004487A priority patent/AP2008004487A0/en
Priority to BRPI0620073-7A priority patent/BRPI0620073A2/en
Priority to EA200801220A priority patent/EA200801220A1/en
Priority to AU2006327823A priority patent/AU2006327823A1/en
Priority to CA002634636A priority patent/CA2634636A1/en
Priority to EP06831787A priority patent/EP1971576A2/en
Application filed by Incyte Corp, Chu-Biao Xue filed Critical Incyte Corp
Priority to RSP-2008/0246A priority patent/RS20080246A/en
Priority to JP2008546684A priority patent/JP2009520809A/en
Publication of WO2007072201A2 publication Critical patent/WO2007072201A2/en
Publication of WO2007072201A3 publication Critical patent/WO2007072201A3/en
Priority to NO20082285A priority patent/NO20082285L/en
Priority to IL191602A priority patent/IL191602A0/en
Priority to TNP2008000275A priority patent/TNSN08275A1/en

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    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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Abstract

The present invention is directed to compounds of Formula (I) which are modulators of chemokine, receptors. The compounds of the invention, and compositions thereof, are useful in the treatment of diseases related to chemokine receptor expression and/or activity.
PCT/IB2006/003739 2005-12-21 2006-12-18 3-aminocyclopentanecarboxamides as modulators of chemokine receptors WO2007072201A2 (en)

Priority Applications (12)

Application Number Priority Date Filing Date Title
MEP-10/08A MEP1008A (en) 2005-12-21 2006-12-11 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
JP2008546684A JP2009520809A (en) 2005-12-21 2006-12-18 3-Aminocyclopentanecarboxamide as modulator of chemokine receptor
RSP-2008/0246A RS20080246A (en) 2005-12-21 2006-12-18 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
EA200801220A EA200801220A1 (en) 2005-12-21 2006-12-18 3-AMINOCYCLOPENTANECARBOXAMIDES AS CHEMOKINE RECEPTOR MODULATORS
AU2006327823A AU2006327823A1 (en) 2005-12-21 2006-12-18 3-Aminocyclopentanecarboxamides as modulators of chemokine receptors
CA002634636A CA2634636A1 (en) 2005-12-21 2006-12-18 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
EP06831787A EP1971576A2 (en) 2005-12-21 2006-12-18 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
AP2008004487A AP2008004487A0 (en) 2005-12-21 2006-12-18 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
BRPI0620073-7A BRPI0620073A2 (en) 2005-12-21 2006-12-18 3-aminocyclopentanecarboxamides as chemokine receptor modulators
NO20082285A NO20082285L (en) 2005-12-21 2008-05-19 3-Aminocyclopentanecarboxamides as modulators of chemokine receptors
IL191602A IL191602A0 (en) 2005-12-21 2008-05-21 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
TNP2008000275A TNSN08275A1 (en) 2005-12-21 2008-06-20 3-AMINOCYCLOPENTANECARBOXAMIDES AS MODULATORS OF CHEMOKINE RECEPTORS

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US75247705P 2005-12-21 2005-12-21
US75232005P 2005-12-21 2005-12-21
US60/752,320 2005-12-21
US60/752,477 2005-12-21

Publications (2)

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WO2007072201A2 WO2007072201A2 (en) 2007-06-28
WO2007072201A3 true WO2007072201A3 (en) 2007-10-04

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PCT/IB2006/003739 WO2007072201A2 (en) 2005-12-21 2006-12-18 3-aminocyclopentanecarboxamides as modulators of chemokine receptors

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US (2) US7700624B2 (en)
EP (1) EP1971576A2 (en)
JP (1) JP2009520809A (en)
KR (1) KR20080070868A (en)
AP (1) AP2008004487A0 (en)
AR (1) AR058402A1 (en)
AU (1) AU2006327823A1 (en)
BR (1) BRPI0620073A2 (en)
CA (1) CA2634636A1 (en)
CR (1) CR10060A (en)
EA (1) EA200801220A1 (en)
EC (1) ECSP088527A (en)
IL (1) IL191602A0 (en)
MA (1) MA30077B1 (en)
ME (1) MEP1008A (en)
NL (1) NL2000380C2 (en)
NO (1) NO20082285L (en)
RS (1) RS20080246A (en)
TW (1) TW200734323A (en)
UY (1) UY30052A1 (en)
WO (1) WO2007072201A2 (en)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
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BRPI0316732B8 (en) * 2002-11-27 2021-05-25 Incyte Corp 3-aminopyrrolidine derivative compound and its pharmaceutical composition
EA015517B1 (en) 2004-04-13 2011-08-30 Инсайт Корпорейшн Piperazinylpiperidine derivatives as chemokine receptor antagonists
AU2005260013A1 (en) * 2004-06-28 2006-01-12 Incyte Corporation 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
US8067415B2 (en) 2005-11-01 2011-11-29 Millennium Pharmaceuticals, Inc. Compounds useful as antagonists of CCR2
WO2007053498A1 (en) 2005-11-01 2007-05-10 Millennium Pharmaceuticals, Inc. Compounds useful as antagonists of ccr2
MEP1008A (en) * 2005-12-21 2010-02-10 Incyte Corp 3-aminocyclopentanecarboxamides as modulators of chemokine receptors
WO2007143600A2 (en) 2006-06-05 2007-12-13 Incyte Corporation Sheddase inhibitors combined with cd30-binding immunotherapeutics for the treatment of cd30 positive diseases
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