WO2006017295A3 - Tetrapeptide analogs - Google Patents
Tetrapeptide analogs Download PDFInfo
- Publication number
- WO2006017295A3 WO2006017295A3 PCT/US2005/024700 US2005024700W WO2006017295A3 WO 2006017295 A3 WO2006017295 A3 WO 2006017295A3 US 2005024700 W US2005024700 W US 2005024700W WO 2006017295 A3 WO2006017295 A3 WO 2006017295A3
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- WO
- WIPO (PCT)
- Prior art keywords
- tetrapeptide analogs
- tetrapeptide
- analogs
- cancer
- compositions
- Prior art date
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- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000003463 hyperproliferative effect Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
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- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
- C07K5/1008—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
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EA200700225A EA200700225A1 (en) | 2004-07-12 | 2005-07-12 | TETRAPTIDE ANALOGUES |
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BRPI0513310-6A BRPI0513310A (en) | 2004-07-12 | 2005-07-12 | tetrapeptide analogs |
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WO (1) | WO2006017295A2 (en) |
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US7838496B2 (en) * | 2003-05-02 | 2010-11-23 | Polyphor Ag/Ltd. | Template-fixed peptidomimetics as medicaments against HIV and cancer |
CN1960728A (en) * | 2004-01-16 | 2007-05-09 | 密歇根大学董事会 | Conformationally constrained SMAC mimetics and the uses thereof |
WO2006014361A1 (en) * | 2004-07-02 | 2006-02-09 | Genentech, Inc. | Inhibitors of iap |
-
2005
- 2005-07-12 EP EP11184396A patent/EP2457895A1/en not_active Withdrawn
- 2005-07-12 KR KR1020077003279A patent/KR20070043831A/en not_active Application Discontinuation
- 2005-07-12 WO PCT/US2005/024700 patent/WO2006017295A2/en active Application Filing
- 2005-07-12 JP JP2007521572A patent/JP2008505976A/en active Pending
- 2005-07-12 AU AU2005271831A patent/AU2005271831A1/en not_active Abandoned
- 2005-07-12 BR BRPI0513310-6A patent/BRPI0513310A/en not_active Application Discontinuation
- 2005-07-12 EP EP11184402A patent/EP2457896A1/en not_active Withdrawn
- 2005-07-12 US US11/632,441 patent/US20100190688A1/en not_active Abandoned
- 2005-07-12 CA CA002573644A patent/CA2573644A1/en not_active Abandoned
- 2005-07-12 MX MX2007000490A patent/MX2007000490A/en unknown
- 2005-07-12 EA EA200700225A patent/EA200700225A1/en unknown
- 2005-07-12 EP EP05771672A patent/EP1773348A4/en not_active Withdrawn
-
2007
- 2007-01-10 MA MA29613A patent/MA28841B1/en unknown
- 2007-01-11 TN TNP2007000005A patent/TNSN07005A1/en unknown
- 2007-01-11 IL IL180677A patent/IL180677A0/en unknown
- 2007-01-12 ZA ZA2007/00357A patent/ZA200700357B/en unknown
- 2007-01-12 GB GB0700629A patent/GB2430935A/en not_active Withdrawn
- 2007-02-09 NO NO20070782A patent/NO20070782L/en not_active Application Discontinuation
- 2007-02-12 CR CR8919A patent/CR8919A/en not_active Application Discontinuation
-
2011
- 2011-01-06 JP JP2011000916A patent/JP2011102312A/en active Pending
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6911426B2 (en) * | 2001-11-21 | 2005-06-28 | The Burnham Institute | Methods and compositions for derepression of IAP-inhibited caspase |
Also Published As
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CR8919A (en) | 2007-08-31 |
GB2430935A (en) | 2007-04-11 |
GB0700629D0 (en) | 2007-02-21 |
CA2573644A1 (en) | 2006-02-16 |
NO20070782L (en) | 2007-04-02 |
KR20070043831A (en) | 2007-04-25 |
AU2005271831A1 (en) | 2006-02-16 |
ZA200700357B (en) | 2008-11-26 |
MA28841B1 (en) | 2007-09-03 |
IL180677A0 (en) | 2008-04-13 |
WO2006017295A2 (en) | 2006-02-16 |
MX2007000490A (en) | 2007-06-11 |
TNSN07005A1 (en) | 2008-06-02 |
EP1773348A2 (en) | 2007-04-18 |
JP2011102312A (en) | 2011-05-26 |
EP2457896A1 (en) | 2012-05-30 |
US20100190688A1 (en) | 2010-07-29 |
BRPI0513310A (en) | 2008-05-06 |
EP2457895A1 (en) | 2012-05-30 |
EA200700225A1 (en) | 2008-02-28 |
JP2008505976A (en) | 2008-02-28 |
EP1773348A4 (en) | 2009-05-20 |
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