UY31587A1 - Derivados de n-heterociclico-imidazo[1,2-a]piridina-2-carboxamidas, su preparacion y su aplicacion en terapéutica. - Google Patents
Derivados de n-heterociclico-imidazo[1,2-a]piridina-2-carboxamidas, su preparacion y su aplicacion en terapéutica.Info
- Publication number
- UY31587A1 UY31587A1 UY31587A UY31587A UY31587A1 UY 31587 A1 UY31587 A1 UY 31587A1 UY 31587 A UY31587 A UY 31587A UY 31587 A UY31587 A UY 31587A UY 31587 A1 UY31587 A1 UY 31587A1
- Authority
- UY
- Uruguay
- Prior art keywords
- carboxamidas
- heterociclico
- piridina
- imidazo
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Psychology (AREA)
- Addiction (AREA)
- Hospice & Palliative Care (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
DERIVADOS DE N-HETEROCICLICO-IMIDAZO[1,2-a] PIRIDINA-2-CARBOXAMIDAS de formula (I) en el estado de base o de sal de adicion a un ácido, en la que los sustituyentes y los índices son segun están especificados en la Memoria descriptiva y en las reivindicaciones. Se divulga los métodos de preparacion, la de los intermediarios y su aplicacion en el tratamiento o prevencion de enfermedades que implican los receptores nucleares Nurr-1 denominados NR4A2, NOT, TINUR, RNR-1 y HZF3.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0800003A FR2925901B1 (fr) | 2008-01-02 | 2008-01-02 | DERIVES DE N-HETEROCYCLIQUE-IMIDAZO°1,2-a!PYRIDINE-2- CARBOXAMIDES, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY31587A1 true UY31587A1 (es) | 2009-08-03 |
Family
ID=39712153
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY3816F UY3816Q (es) | 2008-01-02 | 2008-06-12 | Frasco para productos de perfumeria |
| UY31587A UY31587A1 (es) | 2008-01-02 | 2008-12-30 | Derivados de n-heterociclico-imidazo[1,2-a]piridina-2-carboxamidas, su preparacion y su aplicacion en terapéutica. |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY3816F UY3816Q (es) | 2008-01-02 | 2008-06-12 | Frasco para productos de perfumeria |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US20100317673A1 (es) |
| EP (1) | EP2225242A2 (es) |
| JP (1) | JP2011509250A (es) |
| KR (1) | KR20100099244A (es) |
| CN (1) | CN101910172A (es) |
| AR (1) | AR070072A1 (es) |
| AU (1) | AU2008351927A1 (es) |
| BR (1) | BRPI0821992A2 (es) |
| CA (1) | CA2710860A1 (es) |
| CL (1) | CL2008003933A1 (es) |
| CO (1) | CO6331306A2 (es) |
| EA (1) | EA201070813A1 (es) |
| FR (1) | FR2925901B1 (es) |
| IL (1) | IL206671A0 (es) |
| MA (1) | MA32059B1 (es) |
| MX (1) | MX2010007349A (es) |
| TW (1) | TW200934777A (es) |
| UY (2) | UY3816Q (es) |
| WO (1) | WO2009106749A2 (es) |
| ZA (1) | ZA201004643B (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2903108B1 (fr) * | 2006-07-03 | 2008-08-29 | Sanofi Aventis Sa | Utilisation de derives d'imidazo[1,2-a] pyridine-2-carboxamides en therapeutique. |
| SG191129A1 (en) | 2010-12-13 | 2013-07-31 | Array Biopharma Inc | SUBSTITUTED N-(1H-INDAZOL-4-YL)IMIDAZO[1,2-a]PYRIDINE-3-CARBOXAMIDE COMPOUNDS AS TYPE III RECEPTOR TYROSINE KINASE INHIBITORS |
| WO2012147890A1 (ja) * | 2011-04-27 | 2012-11-01 | 持田製薬株式会社 | 新規アゾール誘導体 |
| EP2939675B1 (en) * | 2012-12-28 | 2019-09-04 | Shin Nippon Biomedical Laboratories, Ltd. | Oct3 activity inhibitor containing imidazopyridine derivative as active component, and oct3 detection agent |
| CN113905787A (zh) * | 2019-04-05 | 2022-01-07 | 斯托姆治疗有限公司 | Mettl3抑制化合物 |
| WO2022074379A1 (en) * | 2020-10-06 | 2022-04-14 | Storm Therapeutics Limited | Mettl3 inhibitory compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5260303A (en) * | 1991-03-07 | 1993-11-09 | G. D. Searle & Co. | Imidazopyridines as serotonergic 5-HT3 antagonists |
| US7544803B2 (en) * | 2004-01-23 | 2009-06-09 | Amgen Inc. | Vanilloid receptor ligands and their use in treatments |
| FR2903107B1 (fr) * | 2006-07-03 | 2008-08-22 | Sanofi Aventis Sa | Derives d'imidazopyridine-2-carboxamides, leur preparation et leur application en therapeutique |
| JP5358962B2 (ja) * | 2007-02-06 | 2013-12-04 | 住友化学株式会社 | 組成物及び該組成物を用いてなる発光素子 |
| EP2219646A4 (en) * | 2007-12-21 | 2010-12-22 | Univ Rochester | METHOD FOR MODIFYING THE LIFETIME OF EUKARYOTIC ORGANISMS |
-
2008
- 2008-01-02 FR FR0800003A patent/FR2925901B1/fr not_active Expired - Fee Related
- 2008-06-12 UY UY3816F patent/UY3816Q/es not_active IP Right Cessation
- 2008-12-30 CL CL2008003933A patent/CL2008003933A1/es unknown
- 2008-12-30 UY UY31587A patent/UY31587A1/es not_active Application Discontinuation
- 2008-12-30 AR ARP080105777A patent/AR070072A1/es unknown
- 2008-12-31 CA CA2710860A patent/CA2710860A1/fr not_active Abandoned
- 2008-12-31 KR KR1020107014639A patent/KR20100099244A/ko not_active Application Discontinuation
- 2008-12-31 JP JP2010541083A patent/JP2011509250A/ja not_active Withdrawn
- 2008-12-31 EA EA201070813A patent/EA201070813A1/ru unknown
- 2008-12-31 MX MX2010007349A patent/MX2010007349A/es not_active Application Discontinuation
- 2008-12-31 AU AU2008351927A patent/AU2008351927A1/en not_active Abandoned
- 2008-12-31 CN CN2008801238170A patent/CN101910172A/zh active Pending
- 2008-12-31 BR BRPI0821992-3A patent/BRPI0821992A2/pt not_active IP Right Cessation
- 2008-12-31 EP EP08872909A patent/EP2225242A2/fr not_active Withdrawn
- 2008-12-31 WO PCT/FR2008/001834 patent/WO2009106749A2/fr active Application Filing
- 2008-12-31 TW TW097151676A patent/TW200934777A/zh unknown
-
2010
- 2010-06-28 IL IL206671A patent/IL206671A0/en unknown
- 2010-07-01 US US12/828,370 patent/US20100317673A1/en not_active Abandoned
- 2010-07-01 ZA ZA2010/04643A patent/ZA201004643B/en unknown
- 2010-07-02 CO CO10080861A patent/CO6331306A2/es not_active Application Discontinuation
- 2010-08-02 MA MA33057A patent/MA32059B1/fr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2009106749A3 (fr) | 2010-05-06 |
| FR2925901A1 (fr) | 2009-07-03 |
| UY3816Q (es) | 2008-09-30 |
| CO6331306A2 (es) | 2011-10-20 |
| BRPI0821992A2 (pt) | 2015-06-23 |
| MA32059B1 (fr) | 2011-02-01 |
| TW200934777A (en) | 2009-08-16 |
| CN101910172A (zh) | 2010-12-08 |
| CL2008003933A1 (es) | 2010-02-12 |
| EA201070813A1 (ru) | 2010-12-30 |
| MX2010007349A (es) | 2010-08-18 |
| AR070072A1 (es) | 2010-03-10 |
| AU2008351927A1 (en) | 2009-09-03 |
| EP2225242A2 (fr) | 2010-09-08 |
| FR2925901B1 (fr) | 2011-03-04 |
| US20100317673A1 (en) | 2010-12-16 |
| CA2710860A1 (fr) | 2009-09-03 |
| ZA201004643B (en) | 2011-09-28 |
| KR20100099244A (ko) | 2010-09-10 |
| WO2009106749A2 (fr) | 2009-09-03 |
| JP2011509250A (ja) | 2011-03-24 |
| IL206671A0 (en) | 2010-12-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20130118 |