UA84714C2 - Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION - Google Patents
Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATIONInfo
- Publication number
- UA84714C2 UA84714C2 UAA200603711A UAA200603711A UA84714C2 UA 84714 C2 UA84714 C2 UA 84714C2 UA A200603711 A UAA200603711 A UA A200603711A UA A200603711 A UAA200603711 A UA A200603711A UA 84714 C2 UA84714 C2 UA 84714C2
- Authority
- UA
- Ukraine
- Prior art keywords
- heading
- treatment
- hiv
- inflammation
- normal
- Prior art date
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
The present invention provides compounds of formula (I) wherein Rand Rare as defined hereinabove. The compounds of the present invention are modulators, especially antagonists, of the activity of chemokine CCR5 receptors. Modulators of the CCR5 receptor may be useful in the treatment of various inflammatory diseases and conditions, and in the treatment of infection by HIV and genetically related retroviruses.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB0323236.0A GB0323236D0 (en) | 2003-10-03 | 2003-10-03 | Chemical compounds |
Publications (1)
Publication Number | Publication Date |
---|---|
UA84714C2 true UA84714C2 (en) | 2008-11-25 |
Family
ID=29415495
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200603711A UA84714C2 (en) | 2003-10-03 | 2004-09-28 | Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION |
Country Status (5)
Country | Link |
---|---|
CN (2) | CN100526313C (en) |
GB (1) | GB0323236D0 (en) |
GT (1) | GT200400203A (en) |
UA (1) | UA84714C2 (en) |
ZA (1) | ZA200602096B (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8012956B2 (en) * | 2007-10-25 | 2011-09-06 | Exelixis, Inc. | Tropane compounds |
-
2003
- 2003-10-03 GB GBGB0323236.0A patent/GB0323236D0/en not_active Ceased
-
2004
- 2004-09-28 CN CNB2004800286836A patent/CN100526313C/en not_active Expired - Fee Related
- 2004-09-28 UA UAA200603711A patent/UA84714C2/en unknown
- 2004-09-28 CN CN200910146182A patent/CN101632664A/en active Pending
- 2004-10-01 GT GT200400203A patent/GT200400203A/en unknown
-
2006
- 2006-03-10 ZA ZA200602096A patent/ZA200602096B/en unknown
Also Published As
Publication number | Publication date |
---|---|
GB0323236D0 (en) | 2003-11-05 |
CN101632664A (en) | 2010-01-27 |
GT200400203A (en) | 2005-04-18 |
ZA200602096B (en) | 2007-05-30 |
CN1863801A (en) | 2006-11-15 |
CN100526313C (en) | 2009-08-12 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MY137609A (en) | Imidazopyridine substituted tropane derivatives with ccr5 receptor antagonist activity for the treatment of hiv and inflammation | |
AP1789A (en) | Tropane derivatives useful in therapy. | |
WO2007116313A3 (en) | Pyrrolidine derivatives as modulators of chemokine ccr5 receptors | |
TW200635897A (en) | Piperidine derivatives and their use as anti-inflammatory agents | |
GEP20084505B (en) | 3-cycloalkylaminopyrrolidine derivatives as modulators of chemokine receptors | |
NO20070137L (en) | Heterocyclic antiviral compounds | |
DK1646389T3 (en) | Pyrimidine-2,4-dione derivatives as gonadotropin-releasing hormone receptor antagonists | |
AU2003301020A1 (en) | Isoquinolinone derivatives and their use as therapeutic agents | |
DE602004020638D1 (en) | PYRIMIDIN-2,4-DION DERIVATIVES AS GONADOTROPINE RELEASING HORMONE RECEPTOR ANTAGONISTS | |
NO20080033L (en) | Quinoline derivatives as NK3 antagonists | |
UA83868C2 (en) | Benzimidazolone and quinazolinone derivatives as agonists on human orl1 receptors | |
GEP20094680B (en) | Piperazinylpiperidine derivatives as chemokine receptor antagonists | |
AU2003226765A1 (en) | Azaindolylpiperidine derivatives as antihistaminic and antiallergic agents | |
UA84714C2 (en) | Normal;heading 1;heading 2;IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV AND INFLAMMATION | |
SG158111A1 (en) | Novel spirotropane compounds and methods for the modulation of chemokine receptor activity | |
CR8323A (en) | DERIVATIVES OF TROPANO | |
DOP2004001002A (en) | DERIVATIVES OF 2-METHYL-4,5,6,7-TETRAHIDRO-1H-IMIDAZO [4,5, C] -PIRIDIN-1-IL-8-AZABICLO- [3.2.1] -OCTO-8-IL] - 1- (3-FLUOROPHENYL) PROPIL WITH ANTIGONIST ACTIVITY OF CCR5 RECEIVER | |
ECSP045344A (en) | USEFUL TROPANO DERIVATIVES IN THERAPY | |
TNSN06096A1 (en) | IMIDAZOPYRIDINE SUBSTITUTED TROPANE DERIVATIVES WITH CCR5 RECEPTOR ANTAGONIST ACTIVITY FOR THE TREATMENT OF HIV INFECTION AND INFLAMMATION | |
MY141461A (en) | N-ureidoalkyl-piperidines as modulators of chemokine receptor activity |