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SMT201500070B - Derivati di pirazolo piridina come inibitori di nadph ossidasi - Google Patents

Derivati di pirazolo piridina come inibitori di nadph ossidasi

Info

Publication number
SMT201500070B
SMT201500070B SM201500070T SM201500070T SMT201500070B SM T201500070 B SMT201500070 B SM T201500070B SM 201500070 T SM201500070 T SM 201500070T SM 201500070 T SM201500070 T SM 201500070T SM T201500070 B SMT201500070 B SM T201500070B
Authority
SM
San Marino
Prior art keywords
pyridine derivatives
oxidase inhibitors
nadph oxidase
pyrazole pyridine
pyrazole
Prior art date
Application number
SM201500070T
Other languages
English (en)
Italian (it)
Inventor
Patrick Page
Mike Orchard
Benoit Laleu
Francesca Gaggini
Original Assignee
Genkyo Tex Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Genkyo Tex Sa filed Critical Genkyo Tex Sa
Publication of SMT201500070B publication Critical patent/SMT201500070B/xx

Links

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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SM201500070T 2008-09-23 2015-03-18 Derivati di pirazolo piridina come inibitori di nadph ossidasi SMT201500070B (it)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08164857A EP2166010A1 (en) 2008-09-23 2008-09-23 Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
PCT/IB2009/054156 WO2010035221A1 (en) 2008-09-23 2009-09-22 Pyrazolo pyridine derivatives as nadph oxidase inhibitors

Publications (1)

Publication Number Publication Date
SMT201500070B true SMT201500070B (it) 2015-05-05

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
SM201500070T SMT201500070B (it) 2008-09-23 2015-03-18 Derivati di pirazolo piridina come inibitori di nadph ossidasi

Country Status (22)

Country Link
US (3) US9096588B2 (xx)
EP (3) EP2166010A1 (xx)
JP (2) JP5700837B2 (xx)
KR (3) KR101763096B1 (xx)
CN (1) CN102159573B (xx)
AU (1) AU2009298008B2 (xx)
BR (1) BRPI0919330A2 (xx)
CA (1) CA2737550C (xx)
CY (1) CY1115952T1 (xx)
DK (2) DK2344492T3 (xx)
ES (2) ES2673405T3 (xx)
HK (2) HK1159107A1 (xx)
HR (1) HRP20150082T1 (xx)
IL (1) IL211892A0 (xx)
PL (2) PL2860179T3 (xx)
PT (2) PT2860179T (xx)
RS (1) RS53781B1 (xx)
RU (1) RU2538041C2 (xx)
SI (1) SI2344492T1 (xx)
SM (1) SMT201500070B (xx)
TR (1) TR201808380T4 (xx)
WO (1) WO2010035221A1 (xx)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2002835A1 (en) 2007-06-04 2008-12-17 GenKyo Tex Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
EP2000176A1 (en) 2007-06-04 2008-12-10 GenKyo Tex Tetrahydroindole derivatives as NADPH Oxidase inhibitors
EP2166009A1 (en) * 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as nadph oxidase inhibitors
EP2165707A1 (en) 2008-09-23 2010-03-24 Genkyo Tex Sa Pyrazolo pyridine derivatives as NADPH oxidase inhibitors
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