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SI3013826T1 - Inhibitorji kristalinične bromodomene - Google Patents

Inhibitorji kristalinične bromodomene

Info

Publication number
SI3013826T1
SI3013826T1 SI201430310T SI201430310T SI3013826T1 SI 3013826 T1 SI3013826 T1 SI 3013826T1 SI 201430310 T SI201430310 T SI 201430310T SI 201430310 T SI201430310 T SI 201430310T SI 3013826 T1 SI3013826 T1 SI 3013826T1
Authority
SI
Slovenia
Prior art keywords
crystalline
bromodomain inhibitors
bromodomain
inhibitors
crystalline bromodomain
Prior art date
Application number
SI201430310T
Other languages
English (en)
Inventor
Yuchuan Gong
Original Assignee
Abbvie Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbvie Inc. filed Critical Abbvie Inc.
Publication of SI3013826T1 publication Critical patent/SI3013826T1/sl

Links

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
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  • Diabetes (AREA)
  • Immunology (AREA)
  • Virology (AREA)
  • Endocrinology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Hematology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Reproductive Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Rheumatology (AREA)
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  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Pain & Pain Management (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Transplantation (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
SI201430310T 2013-06-28 2014-06-27 Inhibitorji kristalinične bromodomene SI3013826T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361840777P 2013-06-28 2013-06-28
PCT/US2014/044513 WO2014210425A1 (en) 2013-06-28 2014-06-27 Crystalline bromodomain inhibitors
EP14745267.6A EP3013826B1 (en) 2013-06-28 2014-06-27 Crystalline bromodomain inhibitors

Publications (1)

Publication Number Publication Date
SI3013826T1 true SI3013826T1 (sl) 2017-10-30

Family

ID=51261220

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Application Number Title Priority Date Filing Date
SI201430310T SI3013826T1 (sl) 2013-06-28 2014-06-27 Inhibitorji kristalinične bromodomene

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US (3) US9321765B2 (sl)
EP (1) EP3013826B1 (sl)
JP (1) JP6423425B2 (sl)
KR (1) KR102323829B1 (sl)
CN (1) CN105473586B (sl)
AR (1) AR096758A1 (sl)
AU (2) AU2014302252B2 (sl)
BR (1) BR112015032736A2 (sl)
CA (1) CA2916221C (sl)
CL (1) CL2015003722A1 (sl)
CR (1) CR20160036A (sl)
CY (1) CY1119066T1 (sl)
DK (1) DK3013826T3 (sl)
DO (1) DOP2015000304A (sl)
ES (1) ES2636939T3 (sl)
HK (2) HK1223354A1 (sl)
HR (1) HRP20171154T1 (sl)
IL (1) IL243202B (sl)
LT (1) LT3013826T (sl)
ME (1) ME02801B (sl)
MX (1) MX360065B (sl)
NZ (1) NZ631112A (sl)
PE (1) PE20160287A1 (sl)
PH (1) PH12015502792A1 (sl)
PL (1) PL3013826T3 (sl)
PT (1) PT3013826T (sl)
RS (1) RS56318B1 (sl)
RU (1) RU2675268C2 (sl)
SG (1) SG11201510692TA (sl)
SI (1) SI3013826T1 (sl)
TW (1) TWI639594B (sl)
UY (1) UY35632A (sl)
WO (1) WO2014210425A1 (sl)

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CN110964691B (zh) * 2019-12-31 2020-10-30 深圳新赛尔生物科技有限公司 子宫内膜干细胞的定向成脂分化培养
JP2023510610A (ja) * 2020-01-19 2023-03-14 チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド ブロモドメインタンパク質阻害剤の結晶形、塩形態及びその製造方法
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HK1223354A1 (zh) 2017-07-28
CA2916221A1 (en) 2014-12-31
IL243202B (en) 2019-07-31
PT3013826T (pt) 2017-08-11
US20150005340A1 (en) 2015-01-01
AU2014302252B2 (en) 2018-03-22
AR096758A1 (es) 2016-02-03
ME02801B (me) 2018-01-20
MX2015017435A (es) 2016-08-12
US9321765B2 (en) 2016-04-26
WO2014210425A1 (en) 2014-12-31
EP3013826A1 (en) 2016-05-04
CR20160036A (es) 2016-05-17
KR20160025021A (ko) 2016-03-07
SG11201510692TA (en) 2016-01-28
TW201534608A (zh) 2015-09-16
PH12015502792A1 (en) 2016-03-21
RS56318B1 (sr) 2017-12-29
CN105473586B (zh) 2019-11-05
PE20160287A1 (es) 2016-05-22
IL243202A0 (en) 2016-02-29
KR102323829B1 (ko) 2021-11-09
US20170066765A1 (en) 2017-03-09
EP3013826B1 (en) 2017-05-10
AU2014302252A1 (en) 2015-12-24
UY35632A (es) 2015-01-30
RU2016102591A (ru) 2017-08-03
LT3013826T (lt) 2017-08-10
CN105473586A (zh) 2016-04-06
US20160237085A1 (en) 2016-08-18
CY1119066T1 (el) 2018-01-10
CL2015003722A1 (es) 2016-07-29
DK3013826T3 (en) 2017-08-28
HRP20171154T1 (hr) 2017-10-20
JP2016525090A (ja) 2016-08-22
BR112015032736A2 (pt) 2017-07-25
MX360065B (es) 2018-10-22
JP6423425B2 (ja) 2018-11-14
RU2675268C2 (ru) 2018-12-18
PL3013826T3 (pl) 2017-10-31
RU2016102591A3 (sl) 2018-04-25
DOP2015000304A (es) 2016-02-29
TWI639594B (zh) 2018-11-01
NZ631112A (en) 2018-03-23
ES2636939T3 (es) 2017-10-10
AU2018201986A1 (en) 2018-04-12
CA2916221C (en) 2022-08-30
HK1224298A1 (zh) 2017-08-18

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