SI0946585T1 - Steroids substituted in position 11, method of preparation, application as medicines and pharmaceutical compositions containing them - Google Patents

Steroids substituted in position 11, method of preparation, application as medicines and pharmaceutical compositions containing them

Info

Publication number: SI0946585T1
Authority: SI; Slovenia
Prior art keywords: medicines; preparation; application; pharmaceutical compositions; compositions containing
Prior art date: 1996-12-23

Application number

SI9730353T

Other languages

English (en)

Slovenian (sl)

Inventor

Yamina Bouali

Francois Nique

Jean-Georges Teutsch

De Velde Patrick Van

Original Assignee

Aventis Pharma S.A.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-12-23

Filing date

1997-12-22

Publication date

2002-10-31

1997-12-22 Application filed by Aventis Pharma S.A. filed Critical Aventis Pharma S.A.

2002-10-31 Publication of SI0946585T1 publication Critical patent/SI0946585T1/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
- C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/32—Antioestrogens

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Veterinary Medicine (AREA)
Physical Education & Sports Medicine (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Diabetes (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SI9730353T 1996-12-23 1997-12-22 Steroids substituted in position 11, method of preparation, application as medicines and pharmaceutical compositions containing them SI0946585T1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
FR9615829A FR2757519B1 (fr)	1996-12-23	1996-12-23	Steroides substitues en position 11, leur procede de preparation, leur application comme medicament et les compositions pharmaceutiques les renfermant
PCT/FR1997/002379 WO1998028324A1 (fr)	1996-12-23	1997-12-22	Steroides substitues en position 11, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
EP97952972A EP0946585B1 (fr)	1996-12-23	1997-12-22	Steroides substitues en position 11, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant

Publications (1)

Publication Number	Publication Date
SI0946585T1 true SI0946585T1 (en)	2002-10-31

Family

ID=9498983

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SI9730353T SI0946585T1 (en)	1996-12-23	1997-12-22	Steroids substituted in position 11, method of preparation, application as medicines and pharmaceutical compositions containing them

Country Status (33)

Country	Link
US (3)	US6207657B1 (xx)
EP (1)	EP0946585B1 (xx)
JP (1)	JP4376319B2 (xx)
KR (1)	KR20000062288A (xx)
CN (1)	CN1247541A (xx)
AP (1)	AP9901567A0 (xx)
AR (1)	AR010857A1 (xx)
AT (1)	ATE216396T1 (xx)
AU (1)	AU726350B2 (xx)
BR (1)	BR9714433A (xx)
CA (1)	CA2275955A1 (xx)
CZ (1)	CZ227899A3 (xx)
DE (1)	DE69712095T2 (xx)
DK (1)	DK0946585T3 (xx)
EA (1)	EA001868B1 (xx)
ES (1)	ES2174329T3 (xx)
FR (1)	FR2757519B1 (xx)
HR (1)	HRP970711B1 (xx)
HU (1)	HUP0001447A3 (xx)
ID (1)	ID22627A (xx)
IL (1)	IL130509A0 (xx)
NO (1)	NO313333B1 (xx)
NZ (1)	NZ336224A (xx)
PL (1)	PL334124A1 (xx)
PT (1)	PT946585E (xx)
SI (1)	SI0946585T1 (xx)
SK (1)	SK83099A3 (xx)
TR (1)	TR199901453T2 (xx)
TW (1)	TW492974B (xx)
UA (1)	UA54483C2 (xx)
WO (1)	WO1998028324A1 (xx)
YU (1)	YU29299A (xx)
ZA (1)	ZA9711324B (xx)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2757519B1 (fr) *	1996-12-23	1999-06-11	Hoechst Marion Roussel Inc	Steroides substitues en position 11, leur procede de preparation, leur application comme medicament et les compositions pharmaceutiques les renfermant
FR2780060B1 (fr) *	1998-06-23	2000-08-04	Hoechst Marion Roussel Inc	Nouveaux 19-nor steroides 17-halogenes, procede et intermediaires de preparation, application comme medicaments et compositions pharmaceutiques les renfermant
DE19929715A1 (de) *	1999-06-24	2000-12-28	Schering Ag	11ß-langkettig-substituierte Estratriene, Verfahren zur Herstellung , pharmazeutische Präparate, die diese 11ß-langkettig-substituierten Estratriene enthalten, sowie deren Verwendung zur Herstellung von Arzneimitteln
FR2826004B1 (fr) *	2001-06-13	2008-03-28	Aventis Pharma Sa	Procede de preparation de derives estrogenes
FR2854402B1 (fr) *	2003-04-29	2008-07-04	Aventis Pharma Sa	Nouveau procede et intermediaires de preparation de composes 19-nor-steroides

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2640977A2 (en) *	1982-06-11	1990-06-29	Roussel Uclaf	New position-11 substituted 19-norsteroids and their application as medicinal products.
US4859585A (en) *	1986-04-17	1989-08-22	Trustees Of Tufts College	In-vitro methods for identifying compositions which are agonists and antagonists of estrogens
FR2643638B1 (fr) *	1989-02-24	1991-06-14	Roussel Uclaf	Nouveaux 19-nor steroides ayant en position 11beta une chaine carbonee comportant une fonction amide ou carbamate, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant
EP0643071B1 (en) *	1993-03-25	2001-02-14	Iskra Industry Co., Ltd.	Compound for inhibiting bone resorption and accelerating osteogenesis
DE4329867C1 (de) *	1993-09-03	1994-09-15	Siemens Ag	Stromspiegel
FR2757519B1 (fr) *	1996-12-23	1999-06-11	Hoechst Marion Roussel Inc	Steroides substitues en position 11, leur procede de preparation, leur application comme medicament et les compositions pharmaceutiques les renfermant
FR2757399B1 (fr) *	1996-12-23	1999-12-17	Hoechst Marion Roussel Inc	Application de composes steroides substitues en 11 pour la fabrication de medicaments ayant une activite estrogene dissociee
FR2761992B1 (fr) *	1997-04-09	1999-06-11	Hoechst Marion Roussel Inc	Nouveaux steroides 4-halogenes, leur procede et intermediaires de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
FR2771096B1 (fr) *	1997-11-17	2000-08-11	Hoechst Marion Roussel Inc	Nouveaux 19-nor steroides, substitues en position 11beta, procede et intermediaires de preparation, application comme medicaments et compositions pharmaceutiques les renfermant

1996
- 1996-12-23 FR FR9615829A patent/FR2757519B1/fr not_active Expired - Fee Related
1997
- 1997-12-17 ZA ZA9711324A patent/ZA9711324B/xx unknown
- 1997-12-22 ES ES97952972T patent/ES2174329T3/es not_active Expired - Lifetime
- 1997-12-22 NZ NZ336224A patent/NZ336224A/en unknown
- 1997-12-22 AU AU56678/98A patent/AU726350B2/en not_active Ceased
- 1997-12-22 YU YU29299A patent/YU29299A/sh unknown
- 1997-12-22 SI SI9730353T patent/SI0946585T1/xx unknown
- 1997-12-22 CA CA002275955A patent/CA2275955A1/fr not_active Abandoned
- 1997-12-22 KR KR1019997005685A patent/KR20000062288A/ko not_active Application Discontinuation
- 1997-12-22 BR BR9714433-9A patent/BR9714433A/pt not_active IP Right Cessation
- 1997-12-22 CZ CZ992278A patent/CZ227899A3/cs unknown
- 1997-12-22 DK DK97952972T patent/DK0946585T3/da active
- 1997-12-22 US US09/331,823 patent/US6207657B1/en not_active Expired - Lifetime
- 1997-12-22 TR TR1999/01453T patent/TR199901453T2/xx unknown
- 1997-12-22 PL PL97334124A patent/PL334124A1/xx unknown
- 1997-12-22 AT AT97952972T patent/ATE216396T1/de not_active IP Right Cessation
- 1997-12-22 ID IDW990573A patent/ID22627A/id unknown
- 1997-12-22 IL IL13050997A patent/IL130509A0/xx unknown
- 1997-12-22 WO PCT/FR1997/002379 patent/WO1998028324A1/fr not_active Application Discontinuation
- 1997-12-22 DE DE69712095T patent/DE69712095T2/de not_active Expired - Lifetime
- 1997-12-22 JP JP52847398A patent/JP4376319B2/ja not_active Expired - Fee Related
- 1997-12-22 CN CN97181921A patent/CN1247541A/zh active Pending
- 1997-12-22 EA EA199900588A patent/EA001868B1/ru not_active IP Right Cessation
- 1997-12-22 AP APAP/P/1999/001567A patent/AP9901567A0/en unknown
- 1997-12-22 PT PT97952972T patent/PT946585E/pt unknown
- 1997-12-22 SK SK830-99A patent/SK83099A3/sk unknown
- 1997-12-22 EP EP97952972A patent/EP0946585B1/fr not_active Expired - Lifetime
- 1997-12-22 UA UA99074263A patent/UA54483C2/uk unknown
- 1997-12-22 HU HU0001447A patent/HUP0001447A3/hu unknown
- 1997-12-23 AR ARP970106163A patent/AR010857A1/es unknown
- 1997-12-23 HR HR970711A patent/HRP970711B1/xx not_active IP Right Cessation
1998
- 1998-02-06 TW TW086119813A patent/TW492974B/zh active
1999
- 1999-06-23 NO NO19993125A patent/NO313333B1/no unknown
2000
- 2000-06-13 US US09/592,710 patent/US6482813B1/en not_active Expired - Lifetime
2002
- 2002-02-14 US US10/075,364 patent/US6541464B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
DE69712095T2 (de)	2002-11-14
UA54483C2 (uk)	2003-03-17
WO1998028324A1 (fr)	1998-07-02
NZ336224A (en)	2001-02-23
PL334124A1 (en)	2000-02-14
DE69712095D1 (de)	2002-05-23
HUP0001447A1 (hu)	2000-11-28
CN1247541A (zh)	2000-03-15
TW492974B (en)	2002-07-01
HUP0001447A3 (en)	2001-03-28
CA2275955A1 (fr)	1998-07-02
AU5667898A (en)	1998-07-17
CZ227899A3 (cs)	1999-09-15
US6541464B2 (en)	2003-04-01
HRP970711A2 (en)	1998-10-31
HRP970711B1 (en)	2002-04-30
IL130509A0 (en)	2000-06-01
ES2174329T3 (es)	2002-11-01
SK83099A3 (en)	2000-01-18
JP4376319B2 (ja)	2009-12-02
NO993125D0 (no)	1999-06-23
FR2757519A1 (fr)	1998-06-26
YU29299A (sh)	2001-05-28
AP9901567A0 (en)	1999-06-30
US6207657B1 (en)	2001-03-27
FR2757519B1 (fr)	1999-06-11
BR9714433A (pt)	2000-05-02
AU726350B2 (en)	2000-11-02
AR010857A1 (es)	2000-07-12
ATE216396T1 (de)	2002-05-15
EP0946585B1 (fr)	2002-04-17
EA001868B1 (ru)	2001-10-22
DK0946585T3 (da)	2002-08-05
PT946585E (pt)	2002-09-30
NO313333B1 (no)	2002-09-16
KR20000062288A (ko)	2000-10-25
ZA9711324B (en)	1999-01-19
EP0946585A1 (fr)	1999-10-06
TR199901453T2 (xx)	1999-08-23
EA199900588A1 (ru)	2000-02-28
ID22627A (id)	1999-12-02
NO993125L (no)	1999-08-20
JP2001507010A (ja)	2001-05-29
US20020198374A1 (en)	2002-12-26
US6482813B1 (en)	2002-11-19

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