SG11201508912YA - 2-PHENYL OR 2-HETARYL IMIDAZOL[1,2-a]PYRIDINE DERIVATIVES - Google Patents
2-PHENYL OR 2-HETARYL IMIDAZOL[1,2-a]PYRIDINE DERIVATIVESInfo
- Publication number
- SG11201508912YA SG11201508912YA SG11201508912YA SG11201508912YA SG11201508912YA SG 11201508912Y A SG11201508912Y A SG 11201508912YA SG 11201508912Y A SG11201508912Y A SG 11201508912YA SG 11201508912Y A SG11201508912Y A SG 11201508912YA SG 11201508912Y A SG11201508912Y A SG 11201508912YA
- Authority
- SG
- Singapore
- Prior art keywords
- hetaryl
- imidazol
- phenyl
- pyridine derivatives
- pyridine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
- A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K49/00—Preparations for testing in vivo
- A61K49/0002—General or multifunctional contrast agents, e.g. chelated agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Psychiatry (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Medicinal Preparation (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13165676 | 2013-04-29 | ||
| PCT/EP2014/058415 WO2014177458A1 (en) | 2013-04-29 | 2014-04-25 | 2-PHENYL OR 2-HETARYL IMIDAZOL[1,2-a]PYRIDINE DERIVATIVES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG11201508912YA true SG11201508912YA (en) | 2015-11-27 |
Family
ID=48190297
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG11201508912YA SG11201508912YA (en) | 2013-04-29 | 2014-04-25 | 2-PHENYL OR 2-HETARYL IMIDAZOL[1,2-a]PYRIDINE DERIVATIVES |
Country Status (19)
| Country | Link |
|---|---|
| US (3) | US10138234B2 (en) |
| EP (1) | EP2991983B1 (en) |
| JP (1) | JP6212628B2 (en) |
| KR (2) | KR20160003173A (en) |
| CN (1) | CN105164125B (en) |
| AR (1) | AR096119A1 (en) |
| AU (1) | AU2014261628A1 (en) |
| BR (1) | BR112015027015A2 (en) |
| CA (1) | CA2910368A1 (en) |
| DK (1) | DK2991983T3 (en) |
| ES (1) | ES2624453T3 (en) |
| HK (1) | HK1213555A1 (en) |
| MX (1) | MX2015014353A (en) |
| PL (1) | PL2991983T3 (en) |
| RU (1) | RU2015147450A (en) |
| SG (1) | SG11201508912YA (en) |
| SI (1) | SI2991983T1 (en) |
| WO (1) | WO2014177458A1 (en) |
| ZA (1) | ZA201507389B (en) |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2991983B1 (en) * | 2013-04-29 | 2017-03-01 | F. Hoffmann-La Roche AG | 2-phenyl or 2-hetaryl imidazol[1,2-a]pyridine derivatives |
| CA2907605A1 (en) * | 2013-05-23 | 2014-11-27 | F. Hoffmann-La Roche Ag | 2-phenylimidazo[1,2-a]pyrimidines as imaging agents |
| RU2671506C2 (en) | 2013-09-26 | 2018-11-01 | Ф. Хоффманн-Ля Рош Аг | Imidazo[1,2-a]pyridin-7-amines as imaging tools |
| EP3355699B1 (en) * | 2015-09-29 | 2021-03-31 | OncoTherapy Science, Inc. | Bicyclic compound and use thereof for inhibiting suv39h2 |
| JP7059270B2 (en) | 2016-07-22 | 2022-04-25 | エーシー・イミューン・エス・アー | Compounds for imaging tau protein aggregates |
| SG11201811311VA (en) | 2016-07-22 | 2019-01-30 | Ac Immune Sa | Compounds for imaging tau protein aggregates |
| WO2018165112A1 (en) * | 2017-03-09 | 2018-09-13 | Oncotherapy Science, Inc. | Bicyclic compound and use thereof for inhibiting histone methyltransferase |
| EP3743426A1 (en) | 2018-01-24 | 2020-12-02 | AC Immune SA | Azacarboline compounds for the detection of tau aggregates |
| EP3743423A1 (en) | 2018-01-24 | 2020-12-02 | AC Immune SA | Gamma-carboline compounds for the detection of tau aggregates |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5654436A (en) * | 1995-06-07 | 1997-08-05 | American Home Products Corporation | 2-substituted benzimidazole derivatives |
| US6696039B2 (en) * | 2001-04-23 | 2004-02-24 | Trustees Of The University Of Pennsylvania | Amyloid plaque aggregation inhibitors and diagnostic imaging agents |
| ES2435070T3 (en) | 2001-08-27 | 2013-12-18 | The Trustees Of The University Of Pennsylvania | Stilbene derivatives and their use for binding and imaging of amyloid plaques |
| JP4738419B2 (en) * | 2005-11-30 | 2011-08-03 | 富士フイルムＲｉファーマ株式会社 | Diagnostic and therapeutic agents for diseases caused by amyloid aggregation and / or deposition |
| JP4913157B2 (en) * | 2006-01-17 | 2012-04-11 | エフ．ホフマン−ラ ロシュ アーゲー | Aryl-isoxazol-4-yl-imidazo [1,2-a] pyridine derivatives useful for the treatment of Alzheimer's disease via GABA receptors |
| WO2008118122A2 (en) * | 2006-05-08 | 2008-10-02 | Molecular Neuroimaging, Llc | Compounds and amyloid probes thereof for therapeutic and imaging uses |
| CN101501033B (en) * | 2006-06-21 | 2012-08-01 | 通用电气医疗有限公司 | Novel compound having affinity for amyloid |
| NZ577318A (en) * | 2006-11-17 | 2012-04-27 | Nihon Mediphysics Co Ltd | Novel compounds with affinity for amyloid |
| US20100092385A1 (en) | 2007-01-22 | 2010-04-15 | Astrazeneca Ab | Novel Heteroaryl Substituted Imidazo [1,2-A] Pyridine Derivatives |
| US20150377123A1 (en) | 2007-08-01 | 2015-12-31 | United Technologies Corporation | Turbine section of high bypass turbofan |
| TW200922628A (en) * | 2007-10-30 | 2009-06-01 | Nihon Mediphysics Co Ltd | Use of novel compound having affinity for amyloid, and process for production of the same |
| MX2011002647A (en) | 2008-09-23 | 2011-04-07 | Wista Lab Ltd | Ligands for aggregated tau molecules. |
| DK2480546T3 (en) * | 2009-09-24 | 2015-02-02 | Hoffmann La Roche | Imidazopyridine or imidazopyrimidinderivater as phosphodiesterase inhibitors 10A |
| US8703768B2 (en) * | 2010-06-09 | 2014-04-22 | Hoffmann-La Roche Inc. | Nitrogen containing heteroaryl compounds |
| EP2991983B1 (en) | 2013-04-29 | 2017-03-01 | F. Hoffmann-La Roche AG | 2-phenyl or 2-hetaryl imidazol[1,2-a]pyridine derivatives |
| RU2671506C2 (en) * | 2013-09-26 | 2018-11-01 | Ф. Хоффманн-Ля Рош Аг | Imidazo[1,2-a]pyridin-7-amines as imaging tools |
-
2014
- 2014-04-25 EP EP14719326.2A patent/EP2991983B1/en active Active
- 2014-04-25 WO PCT/EP2014/058415 patent/WO2014177458A1/en active Application Filing
- 2014-04-25 SG SG11201508912YA patent/SG11201508912YA/en unknown
- 2014-04-25 SI SI201430205A patent/SI2991983T1/en unknown
- 2014-04-25 BR BR112015027015A patent/BR112015027015A2/en not_active IP Right Cessation
- 2014-04-25 ES ES14719326.2T patent/ES2624453T3/en active Active
- 2014-04-25 MX MX2015014353A patent/MX2015014353A/en unknown
- 2014-04-25 CA CA2910368A patent/CA2910368A1/en not_active Abandoned
- 2014-04-25 KR KR1020157033882A patent/KR20160003173A/en active IP Right Grant
- 2014-04-25 KR KR1020177021836A patent/KR20170094001A/en not_active Application Discontinuation
- 2014-04-25 RU RU2015147450A patent/RU2015147450A/en not_active Application Discontinuation
- 2014-04-25 JP JP2016511013A patent/JP6212628B2/en active Active
- 2014-04-25 DK DK14719326.2T patent/DK2991983T3/en active
- 2014-04-25 PL PL14719326T patent/PL2991983T3/en unknown
- 2014-04-25 AU AU2014261628A patent/AU2014261628A1/en not_active Abandoned
- 2014-04-25 CN CN201480024056.9A patent/CN105164125B/en active Active
- 2014-04-28 AR ARP140101744A patent/AR096119A1/en unknown
-
2015
- 2015-10-06 ZA ZA2015/07389A patent/ZA201507389B/en unknown
- 2015-10-28 US US14/925,574 patent/US10138234B2/en active Active
-
2016
- 2016-02-11 HK HK16101486.1A patent/HK1213555A1/en unknown
-
2018
- 2018-10-16 US US16/161,299 patent/US11358962B2/en active Active
- 2018-10-16 US US16/161,306 patent/US10975073B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| KR20170094001A (en) | 2017-08-16 |
| AU2014261628A1 (en) | 2015-10-22 |
| JP2016520046A (en) | 2016-07-11 |
| HK1213555A1 (en) | 2016-07-08 |
| AR096119A1 (en) | 2015-12-09 |
| DK2991983T3 (en) | 2017-05-08 |
| WO2014177458A1 (en) | 2014-11-06 |
| RU2015147450A (en) | 2017-06-05 |
| ES2624453T3 (en) | 2017-07-14 |
| PL2991983T3 (en) | 2017-07-31 |
| US10975073B2 (en) | 2021-04-13 |
| KR20160003173A (en) | 2016-01-08 |
| EP2991983A1 (en) | 2016-03-09 |
| CN105164125B (en) | 2017-10-13 |
| CN105164125A (en) | 2015-12-16 |
| US10138234B2 (en) | 2018-11-27 |
| JP6212628B2 (en) | 2017-10-11 |
| MX2015014353A (en) | 2016-04-07 |
| EP2991983B1 (en) | 2017-03-01 |
| US20190048003A1 (en) | 2019-02-14 |
| US11358962B2 (en) | 2022-06-14 |
| CA2910368A1 (en) | 2014-11-06 |
| BR112015027015A2 (en) | 2017-07-25 |
| US20160244441A1 (en) | 2016-08-25 |
| US20190048002A1 (en) | 2019-02-14 |
| ZA201507389B (en) | 2017-01-25 |
| SI2991983T1 (en) | 2017-06-30 |
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