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SE8305128L - triazole - Google Patents

triazole

Info

Publication number
SE8305128L
SE8305128L SE8305128A SE8305128A SE8305128L SE 8305128 L SE8305128 L SE 8305128L SE 8305128 A SE8305128 A SE 8305128A SE 8305128 A SE8305128 A SE 8305128A SE 8305128 L SE8305128 L SE 8305128L
Authority
SE
Sweden
Prior art keywords
formula
compound
denotes
acid addition
addition salts
Prior art date
Application number
SE8305128A
Other languages
Swedish (sv)
Other versions
SE433496B (en
SE8305128D0 (en
Inventor
Reet G Van
J Heeres
L Wals
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/620,989 external-priority patent/US4079062A/en
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of SE8305128D0 publication Critical patent/SE8305128D0/en
Publication of SE8305128L publication Critical patent/SE8305128L/en
Publication of SE433496B publication Critical patent/SE433496B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D317/00—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms
    • C07D317/08—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3
    • C07D317/10—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings
    • C07D317/14—Heterocyclic compounds containing five-membered rings having two oxygen atoms as the only ring hetero atoms having the hetero atoms in positions 1 and 3 not condensed with other rings with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D317/16—Radicals substituted by halogen atoms or nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Novel 1-(ss-aryl)-ethyl-1H-1,2,4-triazol ketals of the formula <IMAGE> in which Z and Ar are as defined in Claim 1, are obtained by reacting a metal salt of 1H-1,2,4-triazol with a halide carrying the radical <IMAGE> The novel compounds are used as fungicides.

Claims (1)

PatentkravPatent claims 1. FOrfarando fOr framstallning iv en hernial: forenIng med fungicid och/eller baktericid verkan till medicinsk anvdndning, vilken forening bestar as 1-(2-ary1)ety1-1H-1,2,4-triakolketa1 med formeln C112 Ar slier terapeutiskt aktiva syraadditionssalter dArav, earl Z betecknar alkylen floor utgores an -CH2-C112-, -CH(C1-13)-CH(CH3)- eller -C1J2-CH(alkyl)-, sari alkylgruppen her 1 till 10 kolatomer och Ar betecknar 2,4-dihalofenyl, kannetecknat ddrav, att ett metallsalt ay en fore-fling med formeln JO bringas att reagera med en forening med formeln Ar (29 van i Y betecknar halogen, foretrAdesvis i ett ldmpligt poldrt reaktionsinert losningsmedel vid fOrhOjda temperaturer cant att eventuellt terapeutiskt aktiva syraadditianssadter av dessa produkter framstdlles.A process for the preparation of a hernial: compound having a fungicidal and / or bactericidal action for medicinal use, which compound consists of 1- (2-aryl) ethyl-1H-1,2,4-triacolketal of the formula C112 Ar is therapeutically active. acid addition salts dArav, earl Z denotes the alkylene floor consists of -CH2-C112-, -CH (C1-13) -CH (CH3) - or -C1J2-CH (alkyl) -, sari alkyl group her 1 to 10 carbon atoms and Ar denotes 2 4-Dihalophenyl, which may be used to react a metal salt of a precursor of the formula IO with a compound of the formula Ar Active acid addition salts of these products are prepared.
SE8305128A 1974-11-18 1983-09-22 PROCEDURE FOR PREPARING A 1- (BETA-ARYL) ETHYL-1H-1,2,4-TRIAZOLKETAL SE433496B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US52458774A 1974-11-18 1974-11-18
US05/620,989 US4079062A (en) 1974-11-18 1975-10-09 Triazole derivatives

Publications (3)

Publication Number Publication Date
SE8305128D0 SE8305128D0 (en) 1983-09-22
SE8305128L true SE8305128L (en) 1983-09-23
SE433496B SE433496B (en) 1984-05-28

Family

ID=27061544

Family Applications (2)

Application Number Title Priority Date Filing Date
SE7512643A SE433495B (en) 1974-11-18 1975-11-11 TRIAZOLD DERIVATIVES WITH FUNGICID, BACTERICID OR EXTRACTIVE EFFECTS FOR AGRICULTURAL USE
SE8305128A SE433496B (en) 1974-11-18 1983-09-22 PROCEDURE FOR PREPARING A 1- (BETA-ARYL) ETHYL-1H-1,2,4-TRIAZOLKETAL

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SE7512643A SE433495B (en) 1974-11-18 1975-11-11 TRIAZOLD DERIVATIVES WITH FUNGICID, BACTERICID OR EXTRACTIVE EFFECTS FOR AGRICULTURAL USE

Country Status (28)

Country Link
JP (1) JPS5175073A (en)
AT (1) AT351861B (en)
AU (1) AU503503B2 (en)
BR (1) BR7507608A (en)
CA (1) CA1094079A (en)
CH (2) CH615676A5 (en)
CS (1) CS203098B2 (en)
CY (1) CY1064A (en)
DD (1) DD124250A5 (en)
DE (1) DE2551560C3 (en)
DK (1) DK143751C (en)
EG (1) EG11999A (en)
ES (1) ES442656A1 (en)
FI (1) FI62080C (en)
FR (1) FR2290898A1 (en)
GB (1) GB1522657A (en)
HK (1) HK39280A (en)
HU (1) HU177329B (en)
IE (1) IE42064B1 (en)
IL (1) IL48481A (en)
IT (1) IT1052304B (en)
KE (1) KE3058A (en)
NL (1) NL162650C (en)
NZ (1) NZ179111A (en)
SE (2) SE433495B (en)
SU (1) SU649316A3 (en)
TR (1) TR18704A (en)
YU (1) YU40269B (en)

Families Citing this family (54)

* Cited by examiner, † Cited by third party
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US4160838A (en) * 1977-06-02 1979-07-10 Janssen Pharmaceutica N.V. Antimicrobial and plant-growth-regulating triazole derivatives
US4218458A (en) * 1978-06-23 1980-08-19 Janssen Pharmaceutica, N.V. Heterocyclic derivatives of (4-aryloxy-methyl-1,3-dioxolan-2-yl)methyl-1H-imidazoles and 1H-1,2,4-triazoles
EP0006722B1 (en) * 1978-07-03 1984-09-05 Janssen Pharmaceutica N.V. Derivatives of (4-(piperazin-1-yl-phenyloxymethyl)-1.3-dioxolan-2-ylmethyl)-1h-imidazoles and -1h-1.2.4-triazoles, their preparation and use as fungicides and bactericides
US4287195A (en) * 1978-07-14 1981-09-01 Janssen Pharmaceutica, N.V. Heterocyclic derivatives of [4-(piperazin-1-yl-phenyloxymethyl)-1,3-dioxolan-2-ylmethyl]-1H-imidazoles and 1H-1,2,4-triazoles
CH637392A5 (en) * 1978-07-24 1983-07-29 Janssen Pharmaceutica Nv 2-Phenyl-2-azolylmethyl-cyclohexa(d)-1,3-dioxolane derivatives, processes for their preparation, compositions containing these active substances as microbicides, and their use
CH634842A5 (en) * 1978-07-25 1983-02-28 Janssen Pharmaceutica Nv 2-Phenyl-2-(1(H)-imidazolylmethyl)-1,3-dioxane derivatives, processes for their preparation, microbicides containing these active substances, and their use
FR2440367A1 (en) * 1978-11-01 1980-05-30 Ciba Geigy Ag AZOLYLACETALS, THEIR PREPARATION AND THEIR USE AS MICROBICIDAL AGENTS
CA1173449A (en) * 1979-11-16 1984-08-28 Adolf Hubele 1-¬2-(4-diphenyl)ethyl|-1h-azolylketals
NZ196075A (en) * 1980-02-04 1982-12-07 Janssen Pharmaceutica Nv Agent to protect wood coatings and detergents from micro-organisms using a triazole
US4259505A (en) * 1980-03-04 1981-03-31 Ciba-Geigy Corporation Process for the preparation of 1H-azole derivatives
DE3025879A1 (en) * 1980-07-09 1982-02-11 Basf Ag, 6700 Ludwigshafen 1,3-DIOXAN-5-YL-ALKYLTRIAZOLE, THEIR PRODUCTION, THEIR USE FOR REGULATING THE PLANT GROWTH AND MEANS THEREFOR
DE3026140A1 (en) * 1980-07-10 1982-02-18 Basf Ag, 6700 Ludwigshafen 1,3-DIOXAN-5-YL-ALKENYLTRIAZOLE, THEIR PRODUCTION, THEIR USE FOR REGULATING THE PLANT GROWTH AND MEANS THEREFOR
DE3040499A1 (en) * 1980-10-28 1982-06-03 Basf Ag, 6700 Ludwigshafen WOOD PRESERVATIVES
ZA823225B (en) * 1981-05-12 1983-03-30 Ciba Geigy Novel microbicidal arylphenyl ether derivatives,production thereof and the use thereof
DE3232737A1 (en) * 1982-09-03 1984-03-08 Bayer Ag, 5090 Leverkusen 2-ARYL-2-AZOLYLMETHYL-1,3-DIOXEPINE
GB2176106A (en) * 1985-06-05 1986-12-17 Uniroyal Ltd Fungicides comprising carboxamidothiazoles
LT2595B (en) * 1986-02-14 1994-03-25 Ciba Geigy Ag FUNGICIDE PREPARATION IN THE FORM OF SUSPENSION CONCENTRATE AND FIGHT AGAINST BRAINS
ES2009852B3 (en) * 1986-02-14 1989-10-16 Ciba-Geigy Ag FUNGICIDE MIXTURES.
LT2604B (en) * 1986-03-06 1994-03-25 Ciba Geigy Ag FUNGICIDE PREPARATION AND FIGHT AGAINST FLEXIBLE
JPS62212307A (en) * 1986-03-06 1987-09-18 チバ−ガイギ−　アクチエンゲゼルシヤフト Fungicidal composition and use
GB8613913D0 (en) * 1986-06-07 1986-07-09 Ciba Geigy Ag Microbicidal agrochemical compositions
DE3641554C2 (en) * 1986-12-05 1995-04-06 Solvay Werke Gmbh Wood preservatives
DE3641555A1 (en) * 1986-12-05 1988-06-16 Solvay Werke Gmbh MEDIUM OR CONCENTRATE FOR PRESERVATING WOOD AND WOOD MATERIALS
US4940799A (en) * 1987-07-20 1990-07-10 Ciba-Geigy Corporation Preparation of the diastereomeric mixture 2R,4S-1-[2-(2,4-dichlorophenyl)-4-n-propyl-1,3-dioxolan-2-ylmethyl]-1H-1,2,4-triazole
US5250559A (en) * 1988-11-18 1993-10-05 Ciba-Geigy Corporation Microbicidal compositions
DE3927806A1 (en) * 1989-08-23 1991-04-11 Desowag Materialschutz Gmbh MEDIUM OR CONCENTRATE FOR PRESERVING WOOD OR WOOD MATERIALS
DE4013723A1 (en) * 1990-04-28 1991-10-31 Basf Ag 5- (1,2,4-TRIAZOL-1-YLMETHYL) -ISOXAZOLINE
MD24C2 (en) * 1991-07-09 1994-05-31 Fabrica De Parfumerii Si Cosmetica "Viorica" Composition of odoriderous substances
ATE136728T1 (en) * 1991-12-19 1996-05-15 Ciba Geigy Ag MICROBICIDES
EP0556157B1 (en) * 1992-02-13 1997-11-26 Novartis AG Fungicidal mixtures based on triazole fungicides and 4,6-dimethyl-N-phenyl-2-pyrimidinamine
US5342980A (en) 1992-12-30 1994-08-30 American Cyanamid Company Fungicidal agents
DE59400216D1 (en) * 1993-09-24 1996-05-23 Basf Ag Fungicidal mixtures
TW286264B (en) * 1994-05-20 1996-09-21 Ciba Geigy Ag
DE19829113A1 (en) 1998-06-10 1999-12-16 Bayer Ag Means for controlling plant pests
NZ519460A (en) * 1999-12-13 2003-11-28 Bayer Ag Fungicidal combinations of novel fluoro-benzothiazole active substances with other known fungicidal agents
DE50310332D1 (en) 2002-11-12 2008-09-25 Basf Se PROCESS FOR INCREASING INCREASE IN GLYPHOSATE RESISTANT LEGUMINOSES
DE10347090A1 (en) 2003-10-10 2005-05-04 Bayer Cropscience Ag Synergistic fungicidal drug combinations
DE10349501A1 (en) 2003-10-23 2005-05-25 Bayer Cropscience Ag Synergistic fungicidal drug combinations
DE102005026482A1 (en) 2005-06-09 2006-12-14 Bayer Cropscience Ag Active substance combination, useful e.g. for combating unwanted phytopathogenic fungus, comprises herbicides e.g. glyphosate and active substances e.g. strobilurin, triazoles, valinamide and carboxamide
DE502006008090D1 (en) 2005-06-09 2010-11-25 Bayer Cropscience Ag ACTIVE COMBINATIONS
DE102005035300A1 (en) 2005-07-28 2007-02-01 Bayer Cropscience Ag Synergistic fungicidal composition containing a carboxamide, azole and optionally strobilurin, for control of e.g. Puccinia or Erysiphe by treatment of plants, seeds or soil
DE102006023263A1 (en) 2006-05-18 2007-11-22 Bayer Cropscience Ag Synergistic drug combinations
US8318789B2 (en) 2007-03-23 2012-11-27 Syngenta Limited Co-crystals of propiconazole
EP2000028A1 (en) 2007-06-06 2008-12-10 Bayer CropScience Aktiengesellschaft Fungicidal active agent compounds
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WO2010149758A1 (en) 2009-06-25 2010-12-29 Basf Se Antifungal 1, 2, 4-triazolyl derivatives
BR112012001001A2 (en) 2009-07-14 2016-11-16 Basf Se azole compounds of formulas i and ii, compounds of formulas i and i, compounds of formula ix, agricultural composition, use of a pharmaceutical compound, method for treating cancer or virus infections to combat zoopathogenic or humanopathogenic fungi
CN104430378A (en) 2009-07-16 2015-03-25 拜尔农作物科学股份公司 Synergistic active substance combinations containing phenyl triazoles
CN102060850B (en) * 2011-01-12 2012-12-05 周保东 Preparing and refining methods of difenoconazole
JP5958905B2 (en) * 2011-10-20 2016-08-02 公立大学法人秋田県立大学 Plant growth regulator
AR093996A1 (en) 2012-12-18 2015-07-01 Bayer Cropscience Ag BACTERICIDAL COMBINATIONS AND BINARY FUNGICIDES
CN104119322B (en) * 2014-07-11 2016-05-18 北京迪尔乐农业高新技术研发中心 A kind of triazole class compounds for sterilization and its preparation method and application
EP2910126A1 (en) 2015-05-05 2015-08-26 Bayer CropScience AG Active compound combinations having insecticidal properties

Also Published As

Publication number Publication date
DE2551560A1 (en) 1976-05-20
FR2290898A1 (en) 1976-06-11
NL162650B (en) 1980-01-15
KE3058A (en) 1980-06-27
DD124250A5 (en) 1977-02-09
AT351861B (en) 1979-08-27
FI62080B (en) 1982-07-30
HU177329B (en) 1981-09-28
AU503503B2 (en) 1979-09-06
AU8671975A (en) 1977-05-26
CA1094079A (en) 1981-01-20
IT1052304B (en) 1981-06-20
HK39280A (en) 1980-08-08
EG11999A (en) 1978-09-30
YU292975A (en) 1982-02-28
CY1064A (en) 1980-10-24
FI62080C (en) 1982-11-10
FR2290898B1 (en) 1980-06-27
SE433495B (en) 1984-05-28
DK517175A (en) 1976-05-19
JPS5175073A (en) 1976-06-29
NZ179111A (en) 1978-03-06
TR18704A (en) 1977-08-10
GB1522657A (en) 1978-08-23
SE7512643L (en) 1976-05-19
SE433496B (en) 1984-05-28
CH625103A5 (en) 1981-09-15
ATA877775A (en) 1979-01-15
IE42064B1 (en) 1980-05-21
IE42064L (en) 1976-05-18
NL7513389A (en) 1976-05-20
SE425246B (en) 1982-09-13
JPS614834B2 (en) 1986-02-13
DE2551560B2 (en) 1980-07-31
BR7507608A (en) 1976-08-03
SU649316A3 (en) 1979-02-25
YU40269B (en) 1985-12-31
SE8305128D0 (en) 1983-09-22
DE2551560C3 (en) 1981-04-16
IL48481A0 (en) 1976-01-30
DK143751C (en) 1982-03-29
DK143751B (en) 1981-10-05
NL162650C (en) 1980-06-16
FI753228A (en) 1976-05-19
CH615676A5 (en) 1980-02-15
ES442656A1 (en) 1977-08-16
CS203098B2 (en) 1981-02-27
IL48481A (en) 1979-01-31

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