SE435516B - Sett att framstella nya 11beta-substituerade 1,3,5(10)-triensteroidderivat - Google Patents

Sett att framstella nya 11beta-substituerade 1,3,5(10)-triensteroidderivat

Info

Publication number: SE435516B
Authority: SE; Sweden
Prior art keywords: compound; formula; preparation; ethynyl; mixture
Prior art date: 1977-01-13

Application number

SE7714614A

Other languages

English (en)

Swedish (sv)

Other versions

SE7714614L (sv

Inventor

J G Teutsch

D Philibert

Original Assignee

Roussel Uclaf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1977-01-13

Filing date

1977-12-21

Publication date

1984-10-01

1977-12-21 Application filed by Roussel Uclaf filed Critical Roussel Uclaf

1978-07-14 Publication of SE7714614L publication Critical patent/SE7714614L/xx

1984-10-01 Publication of SE435516B publication Critical patent/SE435516B/sv

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J51/00—Normal steroids with unmodified cyclopenta(a)hydrophenanthrene skeleton not provided for in groups C07J1/00 - C07J43/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J21/00—Normal steroids containing carbon, hydrogen, halogen or oxygen having an oxygen-containing hetero ring spiro-condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J21/005—Ketals
- C07J21/006—Ketals at position 3
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J33/00—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- C07J33/002—Normal steroids having a sulfur-containing hetero ring spiro-condensed or not condensed with the cyclopenta(a)hydrophenanthrene skeleton not condensed
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J7/00—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms
- C07J7/0005—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21
- C07J7/001—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group
- C07J7/004—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa
- C07J7/0045—Normal steroids containing carbon, hydrogen, halogen or oxygen substituted in position 17 beta by a chain of two carbon atoms not substituted in position 21 substituted in position 20 by a keto group substituted in position 17 alfa not substituted in position 16
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
- C07J71/0005—Oxygen-containing hetero ring
- C07J71/001—Oxiranes

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

SE7714614A 1977-01-13 1977-12-21 Sett att framstella nya 11beta-substituerade 1,3,5(10)-triensteroidderivat SE435516B (sv)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
FR7700859A FR2377419A1 (fr)	1977-01-13	1977-01-13	Nouveaux derives steroides 11b-substitues 1,3,5 (10) trieniques, leur procede de preparation et leur application comme medicament

Publications (2)

Publication Number	Publication Date
SE7714614L SE7714614L (sv)	1978-07-14
SE435516B true SE435516B (sv)	1984-10-01

Family

ID=9185438

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SE7714614A SE435516B (sv)	1977-01-13	1977-12-21	Sett att framstella nya 11beta-substituerade 1,3,5(10)-triensteroidderivat

Country Status (14)

Country	Link
US (1)	US4272530A (fr)
JP (1)	JPS5390254A (fr)
BE (1)	BE862870A (fr)
CA (1)	CA1121339A (fr)
CH (1)	CH630646A5 (fr)
DE (1)	DE2801417A1 (fr)
DK (1)	DK161334C (fr)
FR (1)	FR2377419A1 (fr)
GB (1)	GB1595133A (fr)
HU (1)	HU176154B (fr)
IE (1)	IE46302B1 (fr)
LU (1)	LU78859A1 (fr)
NL (1)	NL7800364A (fr)
SE (1)	SE435516B (fr)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
NL7701384A (nl) *	1977-02-10	1978-08-14	Akzo Nv	Werkwijze voor het bereiden van nieuwe steroiden van de oestraanreeks.
FR2528434B1 (fr)	1982-06-11	1985-07-19	Roussel Uclaf	Nouveaux 19-nor steroides substitues en 11b et eventuellement en 2, leur procede de preparation et leur application comme medicament
FR2522328B1 (fr) *	1982-03-01	1986-02-14	Roussel Uclaf	Nouveaux produits derives de la structure 3-ceto 4,9 19-nor steroides, leur procede de preparation et leur application comme medicaments
FR2640977A2 (en) *	1982-06-11	1990-06-29	Roussel Uclaf	New position-11 substituted 19-norsteroids and their application as medicinal products.
DE3625315A1 (de) *	1986-07-25	1988-01-28	Schering Ag	11ss-(4-isopropenylphenyl)-estra-4,9-diene, deren herstellung und diese enthaltende pharmazeutische praeparate
DE3925179C2 (de) *	1988-08-22	1996-07-18	Volkswagen Ag	Ansaugluftsteuersystem zum Betreiben einer Brennkraftmaschine mit Leerlaufdrehzahlregelung
DE4018168A1 (de) *	1990-06-01	1991-12-05	Schering Ag	Ausgangsverbindungen fuer die herstellung von 10ss-h-steroiden und ein verfahren zur herstellung dieser ausgangsverbindungen
DE4132182A1 (de) *	1991-09-24	1993-03-25	Schering Ag	11(beta)-substituierte 14, 17-ethanoestratriene, verfahren zur herstellung dieser verbindungen, sowie ihre verwendung zur herstellung von arzneimitteln
US5427766A (en) *	1993-11-15	1995-06-27	The Dow Chemical Company	Radiolabeled steroids for use in radiochemical-guided surgery
AU8201601A (en) *	2000-07-28	2002-02-13	Akzo Nobel Nv	16alpha-methyl or ethyl substituted estrogens
FR2826004B1 (fr) *	2001-06-13	2008-03-28	Aventis Pharma Sa	Procede de preparation de derives estrogenes
PT1624878E (pt) *	2003-05-22	2007-01-31	Pantarhei Bioscience Bv	Utilização de composições que compreendem um componente estrogénico para o tratamento e prevenção da dor musculoesquelética
UA89964C2 (ru)	2004-09-08	2010-03-25	Н.В. Органон	15β-ЗАМЕЩЕННЫЕ СТЕРОИДЫ, КОТОРЫЕ ИМЕЮТ СЕЛЕКТИВНУЮ ЭСТРОГЕННУЮ АКТИВНОСТЬ
JPWO2022080271A1 (fr)	2020-10-15	2022-04-21
EP4231334A4 (fr)	2020-10-15	2024-11-13	Resonac Corporation	Gaz de gravure, son procédé de production, procédé de gravure et procédé de production d'un élément semi-conducteur

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3337365A (en) *	1963-03-25	1967-08-22	Ibm	Electrical resistance composition and method of using the same to form a resistor
US3299108A (en) *	1965-10-18	1967-01-17	Searle & Co	17alpha-alkynyl/alkenyl-13beta-alkyl-11-alkylgona-1, 3, 5 (10)-triene-3, 17beta-diols, ethers and esters thereof and intermediates thereto
US3346602A (en) *	1966-10-12	1967-10-10	Searle & Co	13beta-alkyl-11-alkylgona-1, 3, 5 (10)-trien-17-ones, ethers and esters thereof
US3465010A (en) *	1966-11-22	1969-09-02	Searle & Co	17 - (unsaturated hydrocarbon - substituted) 11,13beta - dialkylgon -4 - ene - 3,17beta-diols and esters thereof
US3629304A (en) *	1969-06-16	1971-12-21	Searle & Co	17alpha-alkynyl - 11beta 13beta - dialkylgona-1 3 5 (10)-triene - 3 17beta-diol 3-cycloalkyl ethers compositions and method
GB1255345A (en) *	1969-08-15	1971-12-01	Searle & Co	3-(3-OXO-11beta13beta-DIALKYL-17beta-HYDROXYGON-4-EN-17alpha-YL) PROPIONIC ACID gamma-LACTONE
US3755301A (en) *	1972-06-23	1973-08-28	Searle & Co	Manufacture of 11-alkyl steroids
US3927046A (en) *	1972-12-09	1975-12-16	Akzona Inc	Novel 11,11-alkylidene steroids
FR2235949B1 (fr) *	1973-06-18	1978-03-17	Roussel Uclaf
NL7317358A (nl) *	1973-12-19	1975-06-23	Akzo Nv	Nieuwe 11(beta)-alkylsteroiden van de oestraanreeks.

1977
- 1977-01-13 FR FR7700859A patent/FR2377419A1/fr active Granted
- 1977-12-21 SE SE7714614A patent/SE435516B/sv not_active IP Right Cessation
1978
- 1978-01-06 US US05/867,486 patent/US4272530A/en not_active Expired - Lifetime
- 1978-01-12 HU HU78RO955A patent/HU176154B/hu unknown
- 1978-01-12 CA CA000294815A patent/CA1121339A/fr not_active Expired
- 1978-01-12 LU LU78859A patent/LU78859A1/fr unknown
- 1978-01-12 DK DK013978A patent/DK161334C/da not_active IP Right Cessation
- 1978-01-12 NL NL7800364A patent/NL7800364A/xx not_active Application Discontinuation
- 1978-01-12 BE BE184285A patent/BE862870A/fr not_active IP Right Cessation
- 1978-01-13 JP JP206778A patent/JPS5390254A/ja active Granted
- 1978-01-13 CH CH39178A patent/CH630646A5/fr not_active IP Right Cessation
- 1978-01-13 GB GB1377/78A patent/GB1595133A/en not_active Expired
- 1978-01-13 DE DE19782801417 patent/DE2801417A1/de active Granted
- 1978-01-13 IE IE79/78A patent/IE46302B1/en not_active IP Right Cessation

Also Published As

Publication number	Publication date
JPS5390254A (en)	1978-08-08
JPS6257638B2 (fr)	1987-12-02
CA1121339A (fr)	1982-04-06
LU78859A1 (fr)	1978-09-18
CH630646A5 (fr)	1982-06-30
BE862870A (fr)	1978-07-12
IE780079L (en)	1978-07-13
FR2377419A1 (fr)	1978-08-11
US4272530A (en)	1981-06-09
HU176154B (en)	1980-12-28
DK161334C (da)	1991-12-09
FR2377419B1 (fr)	1979-04-20
DK161334B (da)	1991-06-24
SE7714614L (sv)	1978-07-14
IE46302B1 (en)	1983-04-20
DE2801417C2 (fr)	1992-09-17
DE2801417A1 (de)	1978-07-20
GB1595133A (en)	1981-08-05
NL7800364A (nl)	1978-07-17
DK13978A (da)	1978-07-14

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