KR950702992A - 살절지동물성 테트라히드로피리미딘(arthropodicidal tetrahydropyrimidines) - Google Patents
살절지동물성 테트라히드로피리미딘(arthropodicidal tetrahydropyrimidines) Download PDFInfo
- Publication number
- KR950702992A KR950702992A KR1019950700807A KR19950700807A KR950702992A KR 950702992 A KR950702992 A KR 950702992A KR 1019950700807 A KR1019950700807 A KR 1019950700807A KR 19950700807 A KR19950700807 A KR 19950700807A KR 950702992 A KR950702992 A KR 950702992A
- Authority
- KR
- South Korea
- Prior art keywords
- alkyl
- compound
- substituted
- haloalkyl
- alkoxy
- Prior art date
Links
- 150000005326 tetrahydropyrimidines Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims abstract 9
- 241000238421 Arthropoda Species 0.000 claims abstract 6
- 229910052799 carbon Inorganic materials 0.000 claims 5
- 229910052736 halogen Inorganic materials 0.000 claims 5
- 150000002367 halogens Chemical class 0.000 claims 4
- 125000001424 substituent group Chemical group 0.000 claims 4
- 125000006552 (C3-C8) cycloalkyl group Chemical group 0.000 claims 3
- 125000000217 alkyl group Chemical group 0.000 claims 3
- 125000004663 dialkyl amino group Chemical group 0.000 claims 3
- 125000001188 haloalkyl group Chemical group 0.000 claims 3
- IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 claims 3
- 125000004767 (C1-C4) haloalkoxy group Chemical group 0.000 claims 2
- 229910052739 hydrogen Inorganic materials 0.000 claims 2
- 229910052757 nitrogen Inorganic materials 0.000 claims 2
- 125000004765 (C1-C4) haloalkyl group Chemical group 0.000 claims 1
- 125000006700 (C1-C6) alkylthio group Chemical group 0.000 claims 1
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 claims 1
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 claims 1
- BRYAHCCROQPDGU-UHFFFAOYSA-N 1-[(6-chloropyridin-3-yl)methyl]-2,6-dimethyl-8-nitro-2,3,5,7-tetrahydroimidazo[1,2-c]pyrimidine Chemical compound CC1CN2CN(C)CC([N+]([O-])=O)=C2N1CC1=CC=C(Cl)N=C1 BRYAHCCROQPDGU-UHFFFAOYSA-N 0.000 claims 1
- NYDMOBMRJZOSGF-UHFFFAOYSA-N 2,6-dimethyl-1-(2-methylsulfanylethyl)-8-nitro-2,3,5,7-tetrahydroimidazo[1,2-c]pyrimidine Chemical compound C1N(C)CC([N+]([O-])=O)=C2N(CCSC)C(C)CN21 NYDMOBMRJZOSGF-UHFFFAOYSA-N 0.000 claims 1
- 125000000882 C2-C6 alkenyl group Chemical group 0.000 claims 1
- 125000003320 C2-C6 alkenyloxy group Chemical group 0.000 claims 1
- 125000003601 C2-C6 alkynyl group Chemical group 0.000 claims 1
- 125000004648 C2-C8 alkenyl group Chemical group 0.000 claims 1
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 claims 1
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 1
- 125000003710 aryl alkyl group Chemical group 0.000 claims 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 1
- 125000004432 carbon atom Chemical group C* 0.000 claims 1
- 125000004438 haloalkoxy group Chemical group 0.000 claims 1
- 125000004995 haloalkylthio group Chemical group 0.000 claims 1
- 125000005843 halogen group Chemical group 0.000 claims 1
- 125000005842 heteroatom Chemical group 0.000 claims 1
- 125000000623 heterocyclic group Chemical group 0.000 claims 1
- QJGQUHMNIGDVPM-UHFFFAOYSA-N nitrogen group Chemical group [N] QJGQUHMNIGDVPM-UHFFFAOYSA-N 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 239000001301 oxygen Chemical group 0.000 claims 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 claims 1
- 229920006395 saturated elastomer Polymers 0.000 claims 1
- 125000000446 sulfanediyl group Chemical group *S* 0.000 claims 1
- 229910052717 sulfur Chemical group 0.000 claims 1
- 239000011593 sulfur Chemical group 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
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- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Dentistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Plant Pathology (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
하기 일반식(I)의 살절지동물성 화합물, 조성물 및 절지동물 방제용 용도에 관한 것이다.
식 중, R1, R2및 n은 명세서에 정의된 바와 같다.
Description
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음
Claims (9)
- 하기 일반식(I)의 화합물,식중, R1은 CH3SCH2CH2-,중에서 선택되고, R2는 H; 경우에 따라 CN, C(O)R3, NO2, OH, SH, C1-C4알콕시, C1-C4알킬티오, C1-C4할로알콕시, N(R5)(R6)R7X, C1-C4알킬아미노, C2-C8디알킬아미노 및 C3-C8시클로알킬에서 독립적으로 선택된 1 또는 2개의 치환체로 치환된C1-C20알킬; C1-C20할로알킬; C1-C6알콕시; C1-C6알킬티오; C2-C6알케닐; C2-C6알케닐옥시; C7-C10아르알콕시; C2-C6알키닐; C(O)R3; N(R5)R6; 경우에 따라 할로겐, C1-C2알킬 및 C1-C2할로알킬에서 독립적으로 선택된 1 내지 3개의 치환체로 치환된 C3-C8시클로알킬; 각 고리가 경우에 따라 할로겐, NO2, CN, C1-C4알킬, C1-C4알콕시, C1-C4알킬티오, C1-C2할로알킬, C1-C2할로알콕시 및 C1-C2할로알킬티오에서 선택된 치환체로 치환된 페닐 및 C7-C10아르알킬; 할로겐, NO2, NH2, CN, C1-C4알킬, C1-C4알콕시, C1-C4알킬티오, C1-C4할로알킬, C1-C4할로알콕시, C1-C4로알킬티오, C1-C4알킬아미노 및 C2-C8디알킬아미노에서 선택된 기로 경우에 따라 치환된 헤테로방향족 고리로 치환된 C1-C3알킬; 2 내지 7개의 탄소원자, 및 질소, 산소 및 황에서 선택된 1 내지 4개의 헤테로원자를 함유하고 탄소 또는 질소를 통해 부착된, 완전 불포화, 부분 불포화 또는 완전 포화된 3 내지 8원 헤테로고리; 및 (CH2CH2O)qR4기 중에서 선택되고, R3은 H, NH2C1-C6알킬, OH, C1-C6알콕시, C1-C4알킬아미노 및 C2-C8디알킬아미노 중에서 선택되고, R4는 H 및 C1-C5알킬 중에서 선택되고, R5및 R6은 H; C1-C6알킬; 및 할로겐, C1-C6알킬 및 C1-C6할로알킬에서 선택된 치환체에 의해 경우에 따라 치환된 페닐 중에서 독립적으로 선택되고, R7은 C1-C6알킬 중에서 선택되고, X는 할로겐 및 OH 중에서 선택되고, n은 1 또는 2이며, q는 1,2,3,4 또는 5이다.
- 제1항에 있어서, R1은 CH3SCH2CH2-,중에서 선택되고, R2는 C1-C6알킬; C3-C8시클로알킬; C2-C8알케닐,; N(R5)R6; C3-C6시클로 알킬, C2-C8디알킬아미노 및 N(R5)(R6)R7X에서 선택된 기로 치환된 C1-C5알킬; 및 (CH2CH2O)qR4기 중에서 선택되고, n은 1인 화합물.
- 제2항에 있어서, R1은 CH3SCH2CH2-이고, R2는 C1-C6알킬인 화합물.
- 제2항에 있어서, R1은R2는 C1-C6알킬인 화합물.
- 제2항에 있어서, R1은R2는 C1-C6알킬인 화합물.
- 제3항에 있어서, 1,2,3,5,6,7-헥사히드로-2, 6-디메틸-1-[2-(메틸티오)에틸]-8-니트로이미다조[1,2-c]피리미딘인 화합물.
- 제4항에 있어서, 1-[(6-클로로-3-피리디닐)메틸]-1,2,3,5,6,7-헥사히드로-2, 6-디메틸-8-니트로이미다조[1,2-C]피리미딘인 화합물.
- 살절지동물 유효량의 제1항 내지 제7항 중 어느 한 항에 따른 화합물과 그에 대한 담체로 이루어진 살절지동물 조성물.
- 절지동물 또는 그의 서식지를 살절지동물 유효량의 제1항 내지 제7항 중 어느 한 항에 따른 화합물에 접촉시키는 것으로 이루어지는 절지동물 방제 방법.※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US07/938808 | 1992-09-01 | ||
| US07/938,808 US5393914A (en) | 1992-09-01 | 1992-09-01 | Motor fuel detergent additives-hydrocarbyloxypolyether allophonate esters of 2-hydroxy ethane |
| US4870493A | 1993-04-15 | 1993-04-15 | |
| US08/048,704 | 1993-04-15 | ||
| PCT/US1993/007926 WO1994005670A1 (en) | 1992-09-01 | 1993-08-26 | Arthropodicidal tetrahydropyrimidines |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR950702992A true KR950702992A (ko) | 1995-08-23 |
Family
ID=26726433
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019950700807A KR950702992A (ko) | 1992-09-01 | 1993-08-26 | 살절지동물성 테트라히드로피리미딘(arthropodicidal tetrahydropyrimidines) |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP0658163A1 (ko) |
| JP (1) | JPH08500605A (ko) |
| KR (1) | KR950702992A (ko) |
| CN (1) | CN1087636A (ko) |
| AU (1) | AU5087793A (ko) |
| BR (1) | BR9307144A (ko) |
| CA (1) | CA2143625A1 (ko) |
| TW (1) | TW242626B (ko) |
| WO (1) | WO1994005670A1 (ko) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4401635A1 (de) * | 1994-01-21 | 1995-07-27 | Bayer Ag | Substituierte 1,2,3,4-Tetrahydro-5-nitro-pyrimidine |
| DE19529411A1 (de) * | 1995-08-10 | 1997-02-13 | Bayer Ag | Substituierte Tetrahydro-5-nitro-pyrimidine |
| CN116806837B (zh) * | 2023-07-03 | 2024-01-23 | 山东福瑞达生物科技有限公司 | 四氢嘧啶在降低虫害对禾本科植物侵害上的应用 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3638121A1 (de) * | 1986-05-30 | 1987-12-03 | Bayer Ag | 1,2,3,6-tetrahydro-5-nitro-pyrimidin-derivate |
-
1993
- 1993-08-24 TW TW082106824A patent/TW242626B/zh active
- 1993-08-26 BR BR9307144A patent/BR9307144A/pt not_active Application Discontinuation
- 1993-08-26 AU AU50877/93A patent/AU5087793A/en not_active Abandoned
- 1993-08-26 JP JP6507257A patent/JPH08500605A/ja active Pending
- 1993-08-26 EP EP93920277A patent/EP0658163A1/en not_active Withdrawn
- 1993-08-26 KR KR1019950700807A patent/KR950702992A/ko not_active Application Discontinuation
- 1993-08-26 WO PCT/US1993/007926 patent/WO1994005670A1/en not_active Application Discontinuation
- 1993-08-26 CA CA002143625A patent/CA2143625A1/en not_active Abandoned
- 1993-09-01 CN CN93118837A patent/CN1087636A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AU5087793A (en) | 1994-03-29 |
| CA2143625A1 (en) | 1994-03-17 |
| EP0658163A1 (en) | 1995-06-21 |
| WO1994005670A1 (en) | 1994-03-17 |
| JPH08500605A (ja) | 1996-01-23 |
| TW242626B (ko) | 1995-03-11 |
| BR9307144A (pt) | 1999-03-30 |
| CN1087636A (zh) | 1994-06-08 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0105 | International application |
Patent event date: 19950228 Patent event code: PA01051R01D Comment text: International Patent Application |
|
| PG1501 | Laying open of application | ||
| PC1203 | Withdrawal of no request for examination | ||
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |