JPS5668680A - Novel piperidine derivative and hypotensive agent containing the same - Google Patents
Novel piperidine derivative and hypotensive agent containing the sameInfo
- Publication number
- JPS5668680A JPS5668680A JP14284979A JP14284979A JPS5668680A JP S5668680 A JPS5668680 A JP S5668680A JP 14284979 A JP14284979 A JP 14284979A JP 14284979 A JP14284979 A JP 14284979A JP S5668680 A JPS5668680 A JP S5668680A
- Authority
- JP
- Japan
- Prior art keywords
- formula
- alkyl
- compound
- hypotensive agent
- same
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Landscapes
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:A compound of formula I [Ar is naphthyl, phenyl, etc.; Q is CO, CH2, CH(OR1) (R1 is H, alkyl, etc.); R is H, alkyl or cycloalkyl; Z is group of formula II (R2 is H, alkyl or alkoxycarbonyl, etc.) or formula III (R3 is alkyl)] and an acid addition salt thereof.
EXAMPLE: 1-[ 2-Oxo-2-( 3, 4-dimethoxyphenyl )-1-ethyl ]-4-( 2-keto-1-benzimidazolinyl )-piperidine.
USE: A hypotensive agent.
PROCESS: The compound of formula I in which Q is CO is obtained by the reaction shown in the reaction scheme (X is a releasing group, e.g. halogen, OSO2CH3, etc.), and the resultant compound is reduced and acylated or alkylated to afford the compound of formula I in which Q is CH(OR1).
COPYRIGHT: (C)1981,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP14284979A JPS5668680A (en) | 1979-11-06 | 1979-11-06 | Novel piperidine derivative and hypotensive agent containing the same |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP14284979A JPS5668680A (en) | 1979-11-06 | 1979-11-06 | Novel piperidine derivative and hypotensive agent containing the same |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5668680A true JPS5668680A (en) | 1981-06-09 |
Family
ID=15325039
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP14284979A Pending JPS5668680A (en) | 1979-11-06 | 1979-11-06 | Novel piperidine derivative and hypotensive agent containing the same |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5668680A (en) |
Citations (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS4867283A (en) * | 1971-12-18 | 1973-09-13 | ||
JPS4941381A (en) * | 1972-04-12 | 1974-04-18 | ||
JPS4995980A (en) * | 1973-01-04 | 1974-09-11 | ||
JPS54160371A (en) * | 1978-06-02 | 1979-12-19 | Kyowa Hakko Kogyo Co Ltd | Novel piperidine derivative and hypotensive agents comprising it |
JPS5517385A (en) * | 1978-07-20 | 1980-02-06 | Science Union & Cie | Benzimidazolinone derivative and medical composition containing it |
JPS5585585A (en) * | 1978-12-25 | 1980-06-27 | Kyowa Hakko Kogyo Co Ltd | Novel piperidine derivative and hypotensor containing the same |
-
1979
- 1979-11-06 JP JP14284979A patent/JPS5668680A/en active Pending
Patent Citations (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS4867283A (en) * | 1971-12-18 | 1973-09-13 | ||
JPS4941381A (en) * | 1972-04-12 | 1974-04-18 | ||
JPS4995980A (en) * | 1973-01-04 | 1974-09-11 | ||
JPS54160371A (en) * | 1978-06-02 | 1979-12-19 | Kyowa Hakko Kogyo Co Ltd | Novel piperidine derivative and hypotensive agents comprising it |
JPS5517385A (en) * | 1978-07-20 | 1980-02-06 | Science Union & Cie | Benzimidazolinone derivative and medical composition containing it |
JPS5585585A (en) * | 1978-12-25 | 1980-06-27 | Kyowa Hakko Kogyo Co Ltd | Novel piperidine derivative and hypotensor containing the same |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
PH23739A (en) | Piperidine derivative and pharmaceutical composition | |
EP0282959A3 (en) | Substituted 9-amino-tetrahydro-acridines and related compounds, a process for their preparation and their use as medicaments | |
NO20005714D0 (en) | Novel substituted cyclic compounds, process for their preparation and pharmaceutical compositions containing them | |
IE883391L (en) | Novel compounds | |
KR880001583A (en) | Method for preparing optically active benzenesulfonamide derivatives | |
HUT37794A (en) | Process for producing new beta-carbolina-3-oxa-diazolyl derivatives and pharmaceutical compositions containing them | |
EP0300882A3 (en) | Novel 5-aminomethylene-2,4-imidazolidinediones and 5-aminomethylene-2-thionoimidazolidine-4-ones | |
IL75116A (en) | Ethyl substituted-beta-carboxylates,process for the preparation thereof and pharmaceutical compositions containing the same | |
JPS54160371A (en) | Novel piperidine derivative and hypotensive agents comprising it | |
JPS5668680A (en) | Novel piperidine derivative and hypotensive agent containing the same | |
NO832667L (en) | PROCEDURE FOR PREPARING 7ALFA-ACYLTHIO-15,16-METHYLENE-3-OXO-17ALFA-PREGNA-1,4-DIEN-21,17-CARBOLACTONES | |
BR8603787A (en) | HETEROCYCLICAL COMPOUNDS, AND, THE PROCESS OF ITS PREPARATION AND APPLICATION | |
ATE168688T1 (en) | METHOD FOR PRODUCING SULFONYL UREA DERIVATIVES | |
JPS56164184A (en) | Novel piperidine derivative | |
IE801382L (en) | Piperidines. | |
ATE34740T1 (en) | (BIS(HYDROXYMETHYL)METHYL)-ISOCHINOLINE DERIVATIVES, PROCESSES FOR THEIR MANUFACTURE AND PHARMACEUTICAL PREPARATIONS CONTAINING THEM. | |
JPS56164183A (en) | Novel piperidine derivative | |
JPS5585585A (en) | Novel piperidine derivative and hypotensor containing the same | |
HU9701295D0 (en) | New process for making intermediers | |
EP0261073A3 (en) | Insecticidal and acaricidal alkane and alkoxy alkane derivatives | |
ATE135693T1 (en) | HALOGENO-4-METHYLPYRAZOLES AND METHOD FOR THE PRODUCTION THEREOF | |
JPS56125385A (en) | Novel piperidine derivative | |
DE3067896D1 (en) | Process for the production of azo compounds | |
MY101628A (en) | Sulfonamide compounds and salts thereof, herbicidal compositions containing them, and process for producing them. | |
JPS5639086A (en) | Novel piperidine derivative and hypotensive agent containing the same |