JPS5598163A - Cinnamylmoranoline derivative - Google Patents
Cinnamylmoranoline derivativeInfo
- Publication number
- JPS5598163A JPS5598163A JP571479A JP571479A JPS5598163A JP S5598163 A JPS5598163 A JP S5598163A JP 571479 A JP571479 A JP 571479A JP 571479 A JP571479 A JP 571479A JP S5598163 A JPS5598163 A JP S5598163A
- Authority
- JP
- Japan
- Prior art keywords
- cinnamylmoranoline
- methyl
- reaction
- formula
- carbinol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Hydrogenated Pyridines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
NEW MATERIAL:Cinnamylmoranoline derivatives of the formula (R1 is H, methyl; R2 is H, hydroxymethyl; R3 is H, methyl, ethyl, methoxyethyl).
USE: They have strong activity of preventing the excessive increase in blood sugar and low toxicity, thus being suitably used as preventive and remedy for hyperglycemia and various kinds of diseases caused by hyperglycemic conditions, e.g., diabetes, arteriosclerosis, fatness, gastrisis, gastric ulcer, duodenal ulcer.
PREPARATION: For example, the comound shown in formula is obtained by treating m-β-methoxyethoxybenzaldehyde resulting from reaction between m-hydroxybenzaldehyde and methoxyethoxybromide with vinylmagnesium bromide to form a carbinol followed by reaction of the carbinol with phosphorus tribromide.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (14)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP571479A JPS6026387B2 (en) | 1979-01-20 | 1979-01-20 | Cinnamyl moranoline derivative |
GB7909865A GB2020278B (en) | 1978-05-03 | 1979-03-21 | Moranoline dervitives |
DE2915037A DE2915037C3 (en) | 1978-05-03 | 1979-04-12 | New N-substituted moranoline derivatives |
FR7910559A FR2424910A1 (en) | 1978-05-03 | 1979-04-25 | MORANOLINE N-SUBSTITUTES DERIVATIVES AND THEIR USE, IN PARTICULAR FOR THE TREATMENT OF HYPERGLYCEMIA |
US06/033,839 US4533668A (en) | 1978-05-03 | 1979-04-27 | Antihyperglycemic moranoline derivatives |
DK178379A DK151623C (en) | 1978-05-03 | 1979-05-01 | METHOD OF ANALOGUE FOR THE PREPARATION OF N-SUBSTITUTED MORANOLINE DERIVATIVES OR PHARMACEUTICAL ACCEPTABLE ACID ADDITION SALTS. |
NLAANVRAGE7903421,A NL175820C (en) | 1978-05-03 | 1979-05-02 | N-SUBSTITUTED MORANOLINE DERIVATIVES, METHOD FOR PREPARING A MEDICINAL PRODUCT THEREFROM, AND MEDICINAL PRODUCT OBTAINED THEREFORE. |
IT48904/79A IT1116820B (en) | 1978-05-03 | 1979-05-02 | MORANOLINA DERIVATIVES WITH PHARMACOLOGICAL PROPERTIES |
SE7903817A SE436874B (en) | 1978-05-03 | 1979-05-02 | N-SUBSTITUTED MORANOLINE DERIVATIVES |
CH415879A CH642629A5 (en) | 1978-05-03 | 1979-05-03 | MORANOLINE DERIVATIVES SUBSTITUTED ON NITROGEN ATOM. |
AT278781A AT371441B (en) | 1979-01-20 | 1981-06-23 | METHOD FOR PRODUCING NEW N-SUBSTITUTED MORANOLINE DERIVATIVES AND THEIR ACID ADDITION SALTS |
SE8402551A SE451017B (en) | 1978-05-03 | 1984-05-11 | CINNAMYLMORANOLIN DERIVATIVES |
SE8402550A SE451016B (en) | 1978-05-03 | 1984-05-11 | N-SUBSTITUTED MORANOLINE DERIVATIVES |
SE8402549A SE451015B (en) | 1978-05-03 | 1984-05-11 | SUBSTITUTED MORANOLINE DERIVATIVES |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP571479A JPS6026387B2 (en) | 1979-01-20 | 1979-01-20 | Cinnamyl moranoline derivative |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5598163A true JPS5598163A (en) | 1980-07-25 |
JPS6026387B2 JPS6026387B2 (en) | 1985-06-24 |
Family
ID=11618779
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP571479A Expired JPS6026387B2 (en) | 1978-05-03 | 1979-01-20 | Cinnamyl moranoline derivative |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS6026387B2 (en) |
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2626470A1 (en) * | 1987-12-09 | 1989-08-04 | Nippon Shinyaku Co Ltd | DEPRESSOR OF THE INHIBITOR OF (ALPHA) 2-PLASMINE |
EP0350012A2 (en) * | 1988-07-08 | 1990-01-10 | Meiji Seika Kaisha Ltd. | Antiviral composition |
WO1991003242A1 (en) * | 1989-09-07 | 1991-03-21 | Nippon Shinyaku Co., Ltd. | Antiviral drug |
US5252587A (en) * | 1990-04-27 | 1993-10-12 | Merrell Dow Pharmaceuticals, Inc. | N-derivatives of 1-deoxy nojirimycin |
US5536732A (en) * | 1990-04-27 | 1996-07-16 | Merrell Pharmaceuticals Inc. | N-derivatives of 1-deoxy nojirimycin |
-
1979
- 1979-01-20 JP JP571479A patent/JPS6026387B2/en not_active Expired
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2626470A1 (en) * | 1987-12-09 | 1989-08-04 | Nippon Shinyaku Co Ltd | DEPRESSOR OF THE INHIBITOR OF (ALPHA) 2-PLASMINE |
EP0350012A2 (en) * | 1988-07-08 | 1990-01-10 | Meiji Seika Kaisha Ltd. | Antiviral composition |
WO1991003242A1 (en) * | 1989-09-07 | 1991-03-21 | Nippon Shinyaku Co., Ltd. | Antiviral drug |
US5252587A (en) * | 1990-04-27 | 1993-10-12 | Merrell Dow Pharmaceuticals, Inc. | N-derivatives of 1-deoxy nojirimycin |
US5536732A (en) * | 1990-04-27 | 1996-07-16 | Merrell Pharmaceuticals Inc. | N-derivatives of 1-deoxy nojirimycin |
Also Published As
Publication number | Publication date |
---|---|
JPS6026387B2 (en) | 1985-06-24 |
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