IS7507A - Ný efnasambönd - Google Patents

Ný efnasambönd

Info

Publication number: IS7507A
Authority: IS; Iceland
Prior art keywords: new compounds; compounds; csbp; trisubstituted; pyrido
Prior art date: 2002-04-19

Application number

IS7507A

Other languages

English (en)

Inventor

C. Boehm Jeffrey

L. Widdowson Katherine

F Callahan James

Wan Zehong

Original Assignee

Smithkline Beecham Corporation

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-04-19

Filing date

2004-10-15

Publication date

2004-10-15

2004-10-15 Application filed by Smithkline Beecham Corporation filed Critical Smithkline Beecham Corporation

2004-10-15 Publication of IS7507A publication Critical patent/IS7507A/is

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
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- A—HUMAN NECESSITIES
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- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Physical Education & Sports Medicine (AREA)
Virology (AREA)
Rheumatology (AREA)
Oncology (AREA)
Orthopedic Medicine & Surgery (AREA)
Immunology (AREA)
Pulmonology (AREA)
Communicable Diseases (AREA)
Heart & Thoracic Surgery (AREA)
Diabetes (AREA)
Dermatology (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Neurology (AREA)
Molecular Biology (AREA)
Neurosurgery (AREA)
Hematology (AREA)
Tropical Medicine & Parasitology (AREA)
Biomedical Technology (AREA)
Pain & Pain Management (AREA)
Endocrinology (AREA)
Vascular Medicine (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Biotechnology (AREA)

IS7507A 2002-04-19 2004-10-15 Ný efnasambönd IS7507A (is)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US37421902P	2002-04-19	2002-04-19
US38855702P	2002-06-13	2002-06-13
PCT/US2003/012127 WO2003088972A1 (en)	2002-04-19	2003-04-18	Novel compounds

Publications (1)

Publication Number	Publication Date
IS7507A true IS7507A (is)	2004-10-15

Family

ID=29254549

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IS7507A IS7507A (is)	2002-04-19	2004-10-15	Ný efnasambönd

Country Status (18)

Country	Link
US (1)	US7629350B2 (is)
EP (1)	EP1499320B1 (is)
JP (1)	JP4603268B2 (is)
KR (1)	KR20040103972A (is)
CN (1)	CN1646131A (is)
AT (1)	ATE370952T1 (is)
AU (1)	AU2003225072A1 (is)
BR (1)	BR0309053A (is)
CA (1)	CA2482022A1 (is)
DE (1)	DE60315826T2 (is)
ES (1)	ES2291630T3 (is)
IL (1)	IL164606A0 (is)
IS (1)	IS7507A (is)
MX (1)	MXPA04010267A (is)
NO (1)	NO20045025L (is)
PL (1)	PL373339A1 (is)
RU (1)	RU2004133811A (is)
WO (1)	WO2003088972A1 (is)

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2003
- 2003-04-18 JP JP2003585724A patent/JP4603268B2/ja not_active Expired - Fee Related
- 2003-04-18 EP EP03721779A patent/EP1499320B1/en not_active Expired - Lifetime
- 2003-04-18 MX MXPA04010267A patent/MXPA04010267A/es unknown
- 2003-04-18 BR BR0309053-1A patent/BR0309053A/pt not_active IP Right Cessation
- 2003-04-18 KR KR10-2004-7016716A patent/KR20040103972A/ko not_active Application Discontinuation
- 2003-04-18 ES ES03721779T patent/ES2291630T3/es not_active Expired - Lifetime
- 2003-04-18 CA CA002482022A patent/CA2482022A1/en not_active Abandoned
- 2003-04-18 AU AU2003225072A patent/AU2003225072A1/en not_active Abandoned
- 2003-04-18 CN CNA038087936A patent/CN1646131A/zh active Pending
- 2003-04-18 PL PL03373339A patent/PL373339A1/xx unknown
- 2003-04-18 AT AT03721779T patent/ATE370952T1/de not_active IP Right Cessation
- 2003-04-18 US US10/511,770 patent/US7629350B2/en not_active Expired - Fee Related
- 2003-04-18 DE DE60315826T patent/DE60315826T2/de not_active Expired - Lifetime
- 2003-04-18 WO PCT/US2003/012127 patent/WO2003088972A1/en active IP Right Grant
- 2003-04-18 RU RU2004133811/04A patent/RU2004133811A/ru not_active Application Discontinuation
2004
- 2004-10-14 IL IL16460604A patent/IL164606A0/xx unknown
- 2004-10-15 IS IS7507A patent/IS7507A/is unknown
- 2004-11-18 NO NO20045025A patent/NO20045025L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
WO2003088972A1 (en)	2003-10-30
KR20040103972A (ko)	2004-12-09
JP2005529877A (ja)	2005-10-06
JP4603268B2 (ja)	2010-12-22
NO20045025L (no)	2004-11-18
AU2003225072A1 (en)	2003-11-03
ES2291630T3 (es)	2008-03-01
EP1499320B1 (en)	2007-08-22
PL373339A1 (en)	2005-08-22
US20060293348A1 (en)	2006-12-28
EP1499320A1 (en)	2005-01-26
BR0309053A (pt)	2005-02-22
RU2004133811A (ru)	2005-04-20
MXPA04010267A (es)	2005-02-03
US7629350B2 (en)	2009-12-08
CN1646131A (zh)	2005-07-27
ATE370952T1 (de)	2007-09-15
EP1499320A4 (en)	2006-05-17
IL164606A0 (en)	2005-12-18
DE60315826D1 (de)	2007-10-04
DE60315826T2 (de)	2008-05-21
CA2482022A1 (en)	2003-10-30

Publication	Publication Date	Title
NO20031794D0 (no)	2003-04-22	Nye forbindelser
EA200702071A1 (ru)	2008-02-28	Новые соединения
DE69917296D1 (de)	2004-06-17	Neue substituierte triazolverbindungen
UA81453C2 (en)	2008-01-10	Pyrazolopyridine derivates
IS7507A (is)	2004-10-15	Ný efnasambönd
MY141144A (en)	2010-03-15	1, 5-disubstituted-3,4-dihydro-1h-pyrimido 4,5-dipyrimidin-2-one compounds and their use in treating csbp/p38 kinase mediated diseases
PL372926A1 (en)	2005-08-08	Piperidine-pyridazones and phthalazones as pde4 inhibitors
TW200724142A (en)	2007-07-01	Novel compounds
BR9810342A (pt)	2000-09-05	Novos compostos imidazola substituìdos
WO2007147103A3 (en)	2008-11-13	Novel compounds
DE60020595D1 (de)	2005-07-07	3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p38-kinase-inhibitoren
TNSN05133A1 (en)	2007-05-14	Imidazoquinoline derivatives as adenosine a3 receptor ligands
ATE281439T1 (de)	2004-11-15	3,4-dihydro-(1h)chinazolin-2-on-verbindungen als csbp/p38-kinase-inhibitoren
UY26980A1 (es)	2002-06-20	Nuevos compuestos
EP1842851A3 (en)	2008-02-27	Novel compounds