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IE44230L - 1, 3-diaza-bicyclo [3,2, 0] heptane derivatives - Google Patents

1, 3-diaza-bicyclo [3,2, 0] heptane derivatives

Info

Publication number
IE44230L
IE44230L IE761953A IE195376A IE44230L IE 44230 L IE44230 L IE 44230L IE 761953 A IE761953 A IE 761953A IE 195376 A IE195376 A IE 195376A IE 44230 L IE44230 L IE 44230L
Authority
IE
Ireland
Prior art keywords
diaza
bicyclo
heptane derivatives
general formula
heptane
Prior art date
Application number
IE761953A
Other versions
IE44230B1 (en
Original Assignee
Smithkline Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/610,517 external-priority patent/US4000154A/en
Application filed by Smithkline Corp filed Critical Smithkline Corp
Priority to IE1921/80A priority Critical patent/IE44231B1/en
Publication of IE44230L publication Critical patent/IE44230L/en
Publication of IE44230B1 publication Critical patent/IE44230B1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/36—One oxygen atom
    • C07D263/38—One oxygen atom attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

The novel compounds of the general formula I, in which R<2> and R<4> have the meaning given in Claim 1, are valuable antibiotics. In order to prepare them, a compound of the general formula VIII is reacted with an acyl halide of the formula R<4>-Hal. <IMAGE> [GB1566261A]
IE1953/76A 1975-09-03 1976-09-01 1,3-diaza-bicyclo/3,2,0/ heptane derivatives IE44230B1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IE1921/80A IE44231B1 (en) 1975-09-03 1976-09-01 3-amino-4-oxazetidine derivatives

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/610,517 US4000154A (en) 1975-09-03 1975-09-03 3-Substituted-6β-(amino- and acylamino)-7-oxo-1,3-diazabicyclo[3.2.0]-h
US68780576A 1976-05-19 1976-05-19

Publications (2)

Publication Number Publication Date
IE44230L true IE44230L (en) 1977-03-03
IE44230B1 IE44230B1 (en) 1981-09-23

Family

ID=27086273

Family Applications (1)

Application Number Title Priority Date Filing Date
IE1953/76A IE44230B1 (en) 1975-09-03 1976-09-01 1,3-diaza-bicyclo/3,2,0/ heptane derivatives

Country Status (7)

Country Link
JP (1) JPS6055507B2 (en)
CH (1) CH633290A5 (en)
DE (1) DE2639397A1 (en)
FR (2) FR2361885A1 (en)
GB (2) GB1566262A (en)
IE (1) IE44230B1 (en)
NL (1) NL7609838A (en)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3108089C2 (en) * 1981-03-04 1987-01-15 Focke & Co, 2810 Verden Device for applying glue to packaging rags
FR2515182B1 (en) * 1981-10-23 1986-05-09 Roussel Uclaf NOVEL PRODUCTS DERIVED FROM 3-AMINO 2-OXO AZETIDINE 1-SULFAMIC ACID, THEIR PREPARATION PROCESS, THEIR APPLICATION AS MEDICAMENTS AND THE INTERMEDIATE PRODUCTS NECESSARY FOR THEIR PREPARATION
GB2151628B (en) * 1981-10-23 1986-05-21 Roussel Uclaf Azetidine intermediates
JPS6316908U (en) * 1986-07-19 1988-02-04

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2219601A1 (en) * 1971-04-27 1972-11-16 Astra Läkemedel AB, Södertälje (Schweden) beta-lactams and processes for their preparation
SE417206B (en) * 1973-03-13 1981-03-02 Merck & Co Inc PROCEDURE FOR THE PREPARATION OF SOCIETIES WITH AUTIBIOTIC ACTION
DE2356862A1 (en) * 1973-11-14 1975-05-15 Univ Kingston 1-Oxa 6-amino-penicillanic acid deriv. analogues - including antibacterials, prepd. in several stages starting with anhydropenicillin

Also Published As

Publication number Publication date
FR2344534A1 (en) 1977-10-14
JPS5239695A (en) 1977-03-28
FR2361885A1 (en) 1978-03-17
NL7609838A (en) 1977-03-07
GB1566261A (en) 1980-04-30
IE44230B1 (en) 1981-09-23
FR2361885B1 (en) 1980-03-14
JPS6055507B2 (en) 1985-12-05
DE2639397A1 (en) 1977-03-10
GB1566262A (en) 1980-04-30
CH633290A5 (en) 1982-11-30
FR2344534B1 (en) 1980-07-04

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