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HUP0200580A2 - Celecoxib polimorf kristályos formái, eljárás az előállításukra és ezeket tartalmazó gyógyszerkészítmények - Google Patents

Celecoxib polimorf kristályos formái, eljárás az előállításukra és ezeket tartalmazó gyógyszerkészítmények

Info

Publication number
HUP0200580A2
HUP0200580A2 HU0200580A HUP0200580A HUP0200580A2 HU P0200580 A2 HUP0200580 A2 HU P0200580A2 HU 0200580 A HU0200580 A HU 0200580A HU P0200580 A HUP0200580 A HU P0200580A HU P0200580 A2 HUP0200580 A2 HU P0200580A2
Authority
HU
Hungary
Prior art keywords
celecoxib
preparation
pharmaceutical compositions
compositions containing
crystalline forms
Prior art date
Application number
HU0200580A
Other languages
English (en)
Inventor
Leaonard J. Ferro
Patricia J. Miyake
Original Assignee
Pharmacia Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corporation filed Critical Pharmacia Corporation
Publication of HUP0200580A2 publication Critical patent/HUP0200580A2/hu
Publication of HUP0200580A3 publication Critical patent/HUP0200580A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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Abstract

A találmány (I) képletű celecoxib I és II kristályformájára, ezekelőállítására, az ezeket tartalmazó gyógyszerkészítményre és ezenkészítmények előállítására vonatkozik. Ó
HU0200580A 1999-12-08 2000-12-01 Polymorphic crystalline forms of celecoxib, process their preparation and pharmaceutical compositions containing them HUP0200580A3 (en)

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PT1404300E (pt) 2001-06-22 2009-11-09 Bend Res Inc Composições farmacêuticas de dispersões de fármacos e polímeros neutros
WO2004026235A2 (en) * 2002-09-20 2004-04-01 Transform Pharmaceuticals, Inc. Pharmaceutical compositions with improved dissolution
US7446107B2 (en) 2002-02-15 2008-11-04 Transform Pharmaceuticals, Inc. Crystalline forms of conazoles and methods of making and using the same
WO2003101392A2 (en) 2002-05-31 2003-12-11 Transform Pharmaceuticals, Inc. Novel conazole crystalline forms and related processes, pharmaceutical compositions and methods
US7927613B2 (en) 2002-02-15 2011-04-19 University Of South Florida Pharmaceutical co-crystal compositions
US7790905B2 (en) 2002-02-15 2010-09-07 Mcneil-Ppc, Inc. Pharmaceutical propylene glycol solvate compositions
US20030224006A1 (en) 2002-03-01 2003-12-04 Zaworotko Michael J. Multiple-component solid phases containing at least one active pharmaceutical ingredient
US20050025791A1 (en) * 2002-06-21 2005-02-03 Julius Remenar Pharmaceutical compositions with improved dissolution
WO2004061433A1 (en) * 2002-12-30 2004-07-22 Transform Pharmaceuticals, Inc. Pharmaceutical compositions with improved dissolution
MXPA04011323A (es) * 2002-05-13 2005-02-14 Pharmacia Corp Compuestos de celecoxib amorfo estable y su proceso de obtencion.
CA2511881C (en) * 2002-12-30 2013-06-25 Transform Pharmaceuticals, Inc. Pharmaceutical compositions comprising a sodium salt of celecoxib with improved dissolution
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BRPI0508063A (pt) * 2004-06-29 2007-07-17 Nycomed Danmark Aps processo para a manufatura de uma composição farmacêutica, nsaid, e, composição farmacêutica
GB0423103D0 (en) * 2004-10-19 2004-11-17 Boots Healthcare Int Ltd Therapeutic agents
AU2006224623A1 (en) * 2005-03-14 2006-09-21 Nycomed Gmbh Method for preventing cardiovascular diseases
CN103462920A (zh) * 2012-06-06 2013-12-25 南京亿华药业有限公司 一种口服环加氧酶-2抑制剂塞来昔布的组合物
CN103524416B (zh) * 2013-10-29 2016-08-17 湖北华世通生物医药科技有限公司 一种塞来昔布新晶型a及其制备方法
CN103539739B (zh) * 2013-10-30 2016-02-10 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型b及其制备方法
CN103508958A (zh) * 2013-10-30 2014-01-15 中美华世通生物医药科技（武汉）有限公司 一种塞来昔布新晶型c及其制备方法
KR101476096B1 (ko) * 2014-03-28 2014-12-24 대원제약주식회사 용해도가 향상된 쎄레콕시브의 약제학적 조성물

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TWI276435B (en) 2007-03-21
PT1150960E (pt) 2005-06-30
KR20020002386A (ko) 2002-01-09
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BG65239B1 (bg) 2007-09-28
OA11831A (en) 2005-08-23
ECSP003807A (es) 2005-07-06
MY128971A (en) 2007-03-30
AU2041201A (en) 2001-06-18
PT1150959E (pt) 2008-04-21
WO2001041536A2 (en) 2001-06-14
ES2236011T3 (es) 2005-07-16
AR030039A1 (es) 2003-08-13
PE20010911A1 (es) 2001-09-10
CO5251445A1 (es) 2003-02-28
EA200401397A1 (ru) 2005-08-25
YU57801A (sh) 2005-07-19
SV2002000235A (es) 2002-06-13
CZ20012875A3 (cs) 2002-02-13
HUP0200580A3 (en) 2002-12-28
NZ529933A (en) 2005-06-24
MY128366A (en) 2007-01-31
CN1411447A (zh) 2003-04-16
KR100717570B1 (ko) 2007-05-15
CN1216869C (zh) 2005-08-31
AR027897A1 (es) 2003-04-16
ZA200107146B (en) 2002-08-29

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