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HRP20120656T1 - Derivati indazolil amida za liječenje poremećaja posredovanih glukokortikoidnim receptorom - Google Patents

Derivati indazolil amida za liječenje poremećaja posredovanih glukokortikoidnim receptorom Download PDF

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Publication number
HRP20120656T1
HRP20120656T1 HRP20120656TT HRP20120656T HRP20120656T1 HR P20120656 T1 HRP20120656 T1 HR P20120656T1 HR P20120656T T HRP20120656T T HR P20120656TT HR P20120656 T HRP20120656 T HR P20120656T HR P20120656 T1 HRP20120656 T1 HR P20120656T1
Authority
HR
Croatia
Prior art keywords
fluorophenyl
oxy
indazol
propan
phenyl
Prior art date
Application number
HRP20120656TT
Other languages
English (en)
Croatian (hr)
Inventor
Berger Markus
Dahm�n Jan
Eriksson Anders
Gabos Balint
Hansson Thomas
Hemmerling Martin
Henriksson Krister
Ivanova Svetlana
Lepist Matti
Mckerrecher Darren
Munck Af Rosenschld Magnus
Nilsson Stinabritt
Rehwinkel Hartmut
Taflin Camilla
Edman Karl
Original Assignee
Bayer Pharma Aktiengesellschaft
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Pharma Aktiengesellschaft, Astrazeneca Ab filed Critical Bayer Pharma Aktiengesellschaft
Publication of HRP20120656T1 publication Critical patent/HRP20120656T1/hr

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    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
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HRP20120656TT 2006-12-21 2007-12-20 Derivati indazolil amida za liječenje poremećaja posredovanih glukokortikoidnim receptorom HRP20120656T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US87118406P 2006-12-21 2006-12-21
US94174507P 2007-06-04 2007-06-04
US97852607P 2007-10-09 2007-10-09
PCT/SE2007/001136 WO2008076048A1 (en) 2006-12-21 2007-12-20 Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disorders

Publications (1)

Publication Number Publication Date
HRP20120656T1 true HRP20120656T1 (hr) 2012-09-30

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HRP20120656TT HRP20120656T1 (hr) 2006-12-21 2007-12-20 Derivati indazolil amida za liječenje poremećaja posredovanih glukokortikoidnim receptorom

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US (4) US7728030B2 (ko)
EP (1) EP2102169B1 (ko)
JP (2) JP5119267B2 (ko)
KR (1) KR20090091354A (ko)
CN (1) CN101611015B (ko)
AR (1) AR064505A1 (ko)
AU (1) AU2007334659B2 (ko)
CA (1) CA2673277A1 (ko)
CL (1) CL2007003804A1 (ko)
CR (1) CR10875A (ko)
CY (1) CY1113269T1 (ko)
DK (1) DK2102169T3 (ko)
DO (1) DOP2009000148A (ko)
EA (1) EA016895B1 (ko)
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