GB1334628A - Thiazolino-pyrimidinone derivatives their preparation and appli cations - Google Patents
Thiazolino-pyrimidinone derivatives their preparation and appli cationsInfo
- Publication number
- GB1334628A GB1334628A GB1334628DA GB1334628A GB 1334628 A GB1334628 A GB 1334628A GB 1334628D A GB1334628D A GB 1334628DA GB 1334628 A GB1334628 A GB 1334628A
- Authority
- GB
- United Kingdom
- Prior art keywords
- pyrimidin
- thiazolo
- dihydro
- thiazolino
- dihydrothiazolo
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
1334628 Some thiazolino-pyrimidinene derivatives SEPERIC 2 Feb 1972 4878/72 Addition to 1306558 Heading C2C The novel compounds 7-methyl-2,3-dihydrothiazolo [3,2-a] pyrimidin-5-one; 7-n-pentyl-2,3- dihydrothiazolo[3,2-a]pyrimidin- 5 - one; 7-phenethyl-2,3-dihydrothiazolo[3, 2- a] - pyrimidin-5-one; 7-ethyl-2,3-dihydro-thiazolo[3,2-a]- pyrimidin-5-one; 7-cyclopropyl-2,3-dihydro-2,3 thiazolo[3,2-a]-pyrimidin-5-one; 3,7-dimethyl- 2,3-dihydro-thiazolo[3,2-a]pyrimidin-5-one; 3- methyl - 7 - benzyl - 2,3 - dihydro-thiazolo- [3,2-a]pyrimidin-5-one may be prepared by cyclizing the appropriate 2-imino-thiazolidine with the appropriate #-substituted #-keto propionic ester. Pharmaceutical compositions of the novel compounds above show analgesic activity when administered orally, parenterally or rectally with the usual excipients.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB487872 | 1972-02-02 |
Publications (1)
Publication Number | Publication Date |
---|---|
GB1334628A true GB1334628A (en) | 1973-10-24 |
Family
ID=9785536
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
GB1334628D Expired GB1334628A (en) | 1972-02-02 | 1972-02-02 | Thiazolino-pyrimidinone derivatives their preparation and appli cations |
Country Status (1)
Country | Link |
---|---|
GB (1) | GB1334628A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4609660A (en) * | 1983-01-12 | 1986-09-02 | Farmitalia Carlo Erba, S.P.A. | Substituted carboxy-thiazolo[3,2-a]pyrimidine derivatives |
-
1972
- 1972-02-02 GB GB1334628D patent/GB1334628A/en not_active Expired
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4609660A (en) * | 1983-01-12 | 1986-09-02 | Farmitalia Carlo Erba, S.P.A. | Substituted carboxy-thiazolo[3,2-a]pyrimidine derivatives |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PS | Patent sealed | ||
435 | Patent endorsed 'licences of right' on the date specified (sect. 35/1949) | ||
PCNP | Patent ceased through non-payment of renewal fee |