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FR2804682B1 - Procede de preparation diastereoselective de piperidines fonctionnalisees en positions 2 et 4 utilisables comme intermediaires de synthese - Google Patents

Procede de preparation diastereoselective de piperidines fonctionnalisees en positions 2 et 4 utilisables comme intermediaires de synthese

Info

Publication number
FR2804682B1
FR2804682B1 FR0001605A FR0001605A FR2804682B1 FR 2804682 B1 FR2804682 B1 FR 2804682B1 FR 0001605 A FR0001605 A FR 0001605A FR 0001605 A FR0001605 A FR 0001605A FR 2804682 B1 FR2804682 B1 FR 2804682B1
Authority
FR
France
Prior art keywords
piperidines
functionalized
positions
synthesis intermediates
diastereoselective preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
FR0001605A
Other languages
English (en)
Other versions
FR2804682A1 (fr
Inventor
Janine Cossy
Damien Belotti
Jean Roger Desmurs
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rhodia Chimie SAS
Original Assignee
Rhodia Chimie SAS
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Rhodia Chimie SAS filed Critical Rhodia Chimie SAS
Priority to FR0001605A priority Critical patent/FR2804682B1/fr
Priority to PCT/FR2001/000370 priority patent/WO2001058872A1/fr
Priority to AU2001235633A priority patent/AU2001235633A1/en
Publication of FR2804682A1 publication Critical patent/FR2804682A1/fr
Application granted granted Critical
Publication of FR2804682B1 publication Critical patent/FR2804682B1/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/60—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Hematology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
FR0001605A 2000-02-09 2000-02-09 Procede de preparation diastereoselective de piperidines fonctionnalisees en positions 2 et 4 utilisables comme intermediaires de synthese Expired - Fee Related FR2804682B1 (fr)

Priority Applications (3)

Application Number Priority Date Filing Date Title
FR0001605A FR2804682B1 (fr) 2000-02-09 2000-02-09 Procede de preparation diastereoselective de piperidines fonctionnalisees en positions 2 et 4 utilisables comme intermediaires de synthese
PCT/FR2001/000370 WO2001058872A1 (fr) 2000-02-09 2001-02-08 Procede de preparation diastereoselective de piperidines fonctionnalisees en positions 2 et 4 utilisables comme intermediaires de synthese
AU2001235633A AU2001235633A1 (en) 2000-02-09 2001-02-08 Method for diastereoselective preparation of piperidines functionalised in positions 2 and 4 for use as synthesis intermediates

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0001605A FR2804682B1 (fr) 2000-02-09 2000-02-09 Procede de preparation diastereoselective de piperidines fonctionnalisees en positions 2 et 4 utilisables comme intermediaires de synthese

Publications (2)

Publication Number Publication Date
FR2804682A1 FR2804682A1 (fr) 2001-08-10
FR2804682B1 true FR2804682B1 (fr) 2002-05-03

Family

ID=8846809

Family Applications (1)

Application Number Title Priority Date Filing Date
FR0001605A Expired - Fee Related FR2804682B1 (fr) 2000-02-09 2000-02-09 Procede de preparation diastereoselective de piperidines fonctionnalisees en positions 2 et 4 utilisables comme intermediaires de synthese

Country Status (3)

Country Link
AU (1) AU2001235633A1 (fr)
FR (1) FR2804682B1 (fr)
WO (1) WO2001058872A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2305646A1 (fr) 2009-10-02 2011-04-06 Enantia, S.L. Procédé pour la préparation d'acides trans-(2R)-4-substitués-pipécoliques et de leurs esters, et des composés intermédiaires

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE48623B1 (en) * 1978-08-31 1985-03-20 Mitsubishi Chem Ind Alpha-(n-arylsulfonyl-l-argininamides,processes for their preparation and pharmaceutical compositions containing these substances
FR2702220B1 (fr) * 1993-03-03 1995-05-12 Synthelabo Dédoublement enzymatique de dérivés de 4-alkyl-2-pipéridine-carboxylate et utilisation des composés obtenus, comme intermédiaires de synthèse.
DE19616049A1 (de) * 1996-04-23 1997-10-30 Wolfgang Dr Grell Neues Verfahren zur Herstellung von 2,4-trans-disubstituierten Piperidin-Derivaten

Also Published As

Publication number Publication date
FR2804682A1 (fr) 2001-08-10
WO2001058872A1 (fr) 2001-08-16
AU2001235633A1 (en) 2001-08-20

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Legal Events

Date Code Title Description
ST Notification of lapse