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FI954614A0 - Imidatsolokinoksalinonijohdannaiset EAA-antagonisteina - Google Patents

Imidatsolokinoksalinonijohdannaiset EAA-antagonisteina

Info

Publication number
FI954614A0
FI954614A0 FI954614A FI954614A FI954614A0 FI 954614 A0 FI954614 A0 FI 954614A0 FI 954614 A FI954614 A FI 954614A FI 954614 A FI954614 A FI 954614A FI 954614 A0 FI954614 A0 FI 954614A0
Authority
FI
Finland
Prior art keywords
imidazoloquinoxalinone
derivatives
preparation
eaa antagonists
eaa
Prior art date
Application number
FI954614A
Other languages
English (en)
Swedish (sv)
Other versions
FI954614A7 (fi
FI954614L (fi
Inventor
Hans-Joerg Treiber
Berthold Behl
Hans-Peter Hofmann
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE4329970A external-priority patent/DE4329970A1/de
Application filed by Basf Ag filed Critical Basf Ag
Publication of FI954614A7 publication Critical patent/FI954614A7/fi
Publication of FI954614A0 publication Critical patent/FI954614A0/fi
Publication of FI954614L publication Critical patent/FI954614L/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI954614A 1993-03-31 1994-03-19 Imidatsolokinoksalinonijohdannaiset EAA-antagonisteina FI954614L (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE4310521 1993-03-31
DE4329970A DE4329970A1 (de) 1993-03-31 1993-09-04 Neue Imidazolo-chinoxalinone, ihre Hestellung und Verwendung
PCT/EP1994/000871 WO1994022865A1 (de) 1993-03-31 1994-03-19 Imidazolochinoxalinonderivate als eaa antagonisten

Publications (3)

Publication Number Publication Date
FI954614A7 FI954614A7 (fi) 1995-09-28
FI954614A0 true FI954614A0 (fi) 1995-09-28
FI954614L FI954614L (fi) 1995-09-28

Family

ID=25924528

Family Applications (1)

Application Number Title Priority Date Filing Date
FI954614A FI954614L (fi) 1993-03-31 1994-03-19 Imidatsolokinoksalinonijohdannaiset EAA-antagonisteina

Country Status (17)

Country Link
EP (1) EP0691970B1 (fi)
JP (1) JPH08508271A (fi)
CN (1) CN1041928C (fi)
AT (1) ATE173263T1 (fi)
AU (1) AU6428294A (fi)
BR (1) BR9406034A (fi)
CA (1) CA2158167A1 (fi)
CZ (1) CZ246495A3 (fi)
FI (1) FI954614L (fi)
HR (1) HRP940210A2 (fi)
HU (1) HUT73970A (fi)
IL (1) IL109076A (fi)
NO (1) NO953892L (fi)
NZ (1) NZ263552A (fi)
PL (1) PL310950A1 (fi)
SI (1) SI9420023A (fi)
WO (1) WO1994022865A1 (fi)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1045964C (zh) * 1994-02-11 1999-10-27 诺沃-诺迪斯克有限公司 杂环化合物及其制备和应用
FR2722789B1 (fr) * 1994-07-20 1996-08-23 Rhone Poulenc Rorer Sa Derives d'acide imidazo (1,2-a)indeno(1,2-e) pyrazine-2-carboxylique, leur preparation et les medicaments les contenant
IT1276167B1 (it) * 1995-11-24 1997-10-27 Foscama Biomed Chim Farma Imidazo(1,2-alfa)chinossalin-4-ammine attivi come antagonisti adenosinici,procedimento per la loro preparazione e loro composizioni
FR2743363A1 (fr) * 1996-01-10 1997-07-11 Rhone Poulenc Rorer Sa 5h,10h-imidazo(1,2-a)indeno(1,2-e)pyrazine-a-ones substituees en position 2, leur preparation et les medicaments les contenant
US6271418B1 (en) * 2000-02-22 2001-08-07 Nippon Kayaku Co., Ltd. Process for preparing (hetero) aromatic substituted benzene derivatives
GB0017518D0 (en) 2000-07-17 2000-08-30 Merck Sharp & Dohme Therapeutic agents
GB0018473D0 (en) * 2000-07-27 2000-09-13 Merck Sharp & Dohme Therapeutic agents
CN100386326C (zh) * 2003-10-22 2008-05-07 中国人民解放军军事医学科学院毒物药物研究所 1-羟甲基咪唑并[1,2-a]喹喔啉化合物及其应用
JP5578786B2 (ja) 2006-12-13 2014-08-27 あすか製薬株式会社 キノキサリン誘導体
FR2921927B1 (fr) * 2007-10-03 2012-10-12 Univ De Montpellier 1 Imidazo°1,2-a!quinoxalines et derives pour le traitement des cancers

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2043064B (en) * 1979-02-09 1983-04-13 Roussel Lab Ltd Oximidazoquinoxaline derivatives
US5153196A (en) * 1991-06-05 1992-10-06 Eli Lilly And Company Excitatory amino acid receptor antagonists and methods for the use thereof
US5182386A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain imidazoquinoxalinones; a new class of gaba brain receptor ligands

Also Published As

Publication number Publication date
IL109076A (en) 1997-06-10
AU6428294A (en) 1994-10-24
CA2158167A1 (en) 1994-10-13
FI954614A7 (fi) 1995-09-28
HUT73970A (en) 1996-10-28
IL109076A0 (en) 1994-06-24
NO953892D0 (no) 1995-09-29
NO953892L (no) 1995-09-29
BR9406034A (pt) 1996-01-02
EP0691970A1 (de) 1996-01-17
ATE173263T1 (de) 1998-11-15
EP0691970B1 (de) 1998-11-11
CN1041928C (zh) 1999-02-03
CZ246495A3 (en) 1996-03-13
NZ263552A (en) 1997-06-24
PL310950A1 (en) 1996-01-08
CN1120336A (zh) 1996-04-10
HU9502848D0 (en) 1995-11-28
JPH08508271A (ja) 1996-09-03
FI954614L (fi) 1995-09-28
SI9420023A (en) 1996-04-30
WO1994022865A1 (de) 1994-10-13
HRP940210A2 (en) 1996-12-31

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Legal Events

Date Code Title Description
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