FI840968A - Nya azoler, deras framstaellningsprocesser och deras anvaendning. - Google Patents

Nya azoler, deras framstaellningsprocesser och deras anvaendning. Download PDF

Info

Publication number: FI840968A
Authority: FI; Finland
Prior art keywords: deras; framstaellningsprocesser; azoler; nya; anvaendning
Prior art date: 1983-03-11

Application number

FI840968A

Other languages

English (en)

Other versions

FI840968A0 (fi

Inventor

Anton Stuetz

Helmut Egger

Original Assignee

Sandoz Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-03-11

Filing date

1984-03-09

Publication date

1984-09-12

1984-03-09 Application filed by Sandoz Ag filed Critical Sandoz Ag

1984-03-09 Publication of FI840968A0 publication Critical patent/FI840968A0/fi

1984-09-12 Publication of FI840968A publication Critical patent/FI840968A/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/62—Oxygen or sulfur atoms
- C07D213/70—Sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
- C07C45/63—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/14—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D295/155—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with the ring nitrogen atoms and the carbon atoms with three bonds to hetero atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/192—Radicals derived from carboxylic acids from aromatic carboxylic acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
- C07D295/215—Radicals derived from nitrogen analogues of carbonic acid

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Plural Heterocyclic Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

FI840968A 1983-03-11 1984-03-09 Nya azoler, deras framstaellningsprocesser och deras anvaendning. FI840968A (fi)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
CH1332/83A CH655103A5 (de)	1983-03-11	1983-03-11	Azolderivate, verfahren zu ihrer herstellung und ihre verwendung.

Publications (2)

Publication Number	Publication Date
FI840968A0 FI840968A0 (fi)	1984-03-09
FI840968A true FI840968A (fi)	1984-09-12

Family

ID=4207992

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI840968A FI840968A (fi)	1983-03-11	1984-03-09	Nya azoler, deras framstaellningsprocesser och deras anvaendning.

Country Status (24)

Country	Link
JP (1)	JPS59175472A (fi)
KR (1)	KR890000377B1 (fi)
AU (1)	AU571494B2 (fi)
BE (1)	BE899073A (fi)
CA (1)	CA1242723A (fi)
CH (1)	CH655103A5 (fi)
DE (1)	DE3408127A1 (fi)
DK (1)	DK149784A (fi)
ES (1)	ES8506639A1 (fi)
FI (1)	FI840968A (fi)
FR (1)	FR2542315B1 (fi)
GB (1)	GB2136801B (fi)
GR (1)	GR81869B (fi)
HU (1)	HUT36098A (fi)
IL (1)	IL71203A (fi)
IT (1)	IT1199085B (fi)
LU (1)	LU85245A1 (fi)
NL (1)	NL8400730A (fi)
NZ (1)	NZ207453A (fi)
PH (1)	PH24667A (fi)
PL (1)	PL146072B1 (fi)
PT (1)	PT78226B (fi)
SE (1)	SE8401321L (fi)
ZA (1)	ZA841782B (fi)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8618188D0 (en) *	1986-07-25	1986-09-03	Ici Plc	Diamine compounds
DE3644615A1 (de) *	1986-12-29	1988-07-07	Lentia Gmbh	Imidazol- und triazolderivate zur verwendung als antimykotische mittel
DE3644616A1 (de) *	1986-12-29	1988-07-07	Lentia Gmbh	Imidazolderivate, verfahren zur herstellung und deren verwendung
US5252594A (en) *	1992-06-17	1993-10-12	Rohm And Haas Company	Fungicidal (2-aryl-2-substituted)ethyl-1,2,4-triazoles
US5358939A (en) *	1992-06-25	1994-10-25	Rohm And Haas Company	Fungicidal 2-aryl-2,2-disubstituted ethyl-1,2,4-triazoles
DE4412358A1 (de) *	1994-04-11	1995-10-12	Bayer Ag	Cyclopropyl-ethyl-azole
GB9409882D0 (en) *	1994-05-18	1994-07-06	Sandoz Ltd	Organic compounds
JP3214987B2 (ja) *	1994-09-05	2001-10-02	日本碍子株式会社	半導体装置およびその製造方法
WO2004058713A1 (en) *	2002-12-20	2004-07-15	Irm Llc	Differential tumor cytotoxocity compounds and compositions
WO2004056744A1 (en) *	2002-12-23	2004-07-08	Janssen Pharmaceutica N.V.	Adamantyl acetamides as hydroxysteroid dehydrogenase inhibitors
NZ551077A (en)	2004-05-07	2009-05-31	Janssen Pharmaceutica Nv	Pyrrolidin-2-one and piperidin-2-one derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors
CN101300005B (zh)	2004-08-30	2013-05-01	詹森药业有限公司	作为11-β羟类固醇脱氢酶抑制剂的N-2金刚烷基-2-苯氧基-乙酰胺衍生物
DE602005017159D1 (de)	2004-08-30	2009-11-26	Janssen Pharmaceutica Nv	Oxysteroid-dehydrogenase-inhibitoren
US8563591B2 (en)	2004-08-30	2013-10-22	Janssen Pharmaceutica N.V.	Tricyclic lactam derivatives as 11-beta hydroxysteroid dehydrogenase inhibitors
US8071603B2 (en)	2004-09-20	2011-12-06	Xenon Pharmaceuticals Inc.	Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors
EP1814551A2 (en)	2004-09-20	2007-08-08	Xenon Pharmaceuticals Inc.	Pyridazine derivatives for inhibiting human stearoyl-coa-desaturase
WO2006034315A2 (en)	2004-09-20	2006-03-30	Xenon Pharmaceuticals Inc.	Heterocyclic derivatives for the treatment of diseases mediated by stearoyl-coa desaturase enzymes
US7951805B2 (en)	2004-09-20	2011-05-31	Xenon Pharmaceuticals Inc.	Heterocyclic derivatives and their use as mediators of stearoyl-CoA desaturase
BRPI0515505A (pt)	2004-09-20	2008-07-29	Xenon Pharmaceuticals Inc	derivados heterocìclicos e sua utilização como inibidores da estearoil-coa desaturase
JP5043668B2 (ja)	2004-09-20	2012-10-10	ゼノン・ファーマシューティカルズ・インコーポレイテッド	複素環誘導体および治療薬としてのそれらの使用
EP2269610A3 (en)	2004-09-20	2011-03-09	Xenon Pharmaceuticals Inc.	Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
US8541457B2 (en)	2005-06-03	2013-09-24	Xenon Pharmaceuticals Inc.	Aminothiazole derivatives as human stearoyl-CoA desaturase inhibitors
CN104530038A (zh) *	2014-12-10	2015-04-22	沈阳药科大学	酰胺咪唑类衍生物及其用途
CN112142673B (zh) *	2020-09-18	2023-06-30	聊城大学	芳基烯烃唑类衍生物及其制备方法和用途

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SU557755A3 (ru) *	1968-08-19	1977-05-05	Янссен Фармасьютика Н.В. (Фирма)	Способ получени производных имидазола
CA1189857A (en) *	1981-03-27	1985-07-02	Janssen Pharmaceutica Naamloze Vennootschap	Antimicrobial triazole derivatives
AU8314482A (en) *	1981-05-19	1982-11-25	Imperial Chemical Industries Plc	3-triazolyl(imidazolyl)-2,2 bis phenyl-propionamides
EP0117462A3 (en) *	1983-02-28	1986-08-20	American Cyanamid Company	N-(2-4-(1h-imidazol-1-yl)alkyl)arylamides

1983
- 1983-03-11 CH CH1332/83A patent/CH655103A5/de not_active IP Right Cessation
1984
- 1984-02-27 HU HU84780A patent/HUT36098A/hu unknown
- 1984-02-29 DK DK149784A patent/DK149784A/da not_active Application Discontinuation
- 1984-03-05 FR FR8403733A patent/FR2542315B1/fr not_active Expired
- 1984-03-05 BE BE1/10974A patent/BE899073A/fr not_active IP Right Cessation
- 1984-03-06 DE DE19843408127 patent/DE3408127A1/de not_active Withdrawn
- 1984-03-07 GB GB08405900A patent/GB2136801B/en not_active Expired
- 1984-03-07 NL NL8400730A patent/NL8400730A/nl not_active Application Discontinuation
- 1984-03-08 IT IT47817/84A patent/IT1199085B/it active
- 1984-03-09 NZ NZ207453A patent/NZ207453A/en unknown
- 1984-03-09 FI FI840968A patent/FI840968A/fi not_active Application Discontinuation
- 1984-03-09 ES ES530461A patent/ES8506639A1/es not_active Expired
- 1984-03-09 PH PH30375A patent/PH24667A/en unknown
- 1984-03-09 PT PT78226A patent/PT78226B/pt not_active IP Right Cessation
- 1984-03-09 SE SE8401321A patent/SE8401321L/xx not_active Application Discontinuation
- 1984-03-09 CA CA000449330A patent/CA1242723A/en not_active Expired
- 1984-03-09 IL IL71203A patent/IL71203A/xx unknown
- 1984-03-09 AU AU25475/84A patent/AU571494B2/en not_active Ceased
- 1984-03-09 PL PL1984246600A patent/PL146072B1/pl unknown
- 1984-03-09 ZA ZA841782A patent/ZA841782B/xx unknown
- 1984-03-09 LU LU85245A patent/LU85245A1/fr unknown
- 1984-03-10 JP JP59046384A patent/JPS59175472A/ja active Pending
- 1984-03-10 KR KR1019840001218A patent/KR890000377B1/ko not_active IP Right Cessation
- 1984-03-12 GR GR74070A patent/GR81869B/el unknown

Also Published As

Publication number	Publication date
FR2542315B1 (fr)	1986-02-07
IL71203A (en)	1988-10-31
ES530461A0 (es)	1985-07-16
KR890000377B1 (ko)	1989-03-15
ES8506639A1 (es)	1985-07-16
GB2136801A (en)	1984-09-26
PT78226B (en)	1986-07-15
JPS59175472A (ja)	1984-10-04
BE899073A (fr)	1984-09-05
PH24667A (en)	1990-09-07
CA1242723A (en)	1988-10-04
AU2547584A (en)	1984-09-13
PT78226A (en)	1984-04-01
SE8401321L (sv)	1984-09-12
DK149784A (da)	1984-09-12
DE3408127A1 (de)	1984-09-13
NL8400730A (nl)	1984-10-01
NZ207453A (en)	1987-09-30
KR850006386A (ko)	1985-10-05
ZA841782B (en)	1985-10-30
FR2542315A1 (fr)	1984-09-14
AU571494B2 (en)	1988-04-21
GB8405900D0 (en)	1984-04-11
LU85245A1 (fr)	1984-11-14
DK149784D0 (da)	1984-02-29
PL146072B1 (en)	1988-12-31
IT8447817A0 (it)	1984-03-08
PL246600A1 (en)	1985-03-12
IT1199085B (it)	1988-12-30
GB2136801B (en)	1987-03-04
IL71203A0 (en)	1984-06-29
FI840968A0 (fi)	1984-03-09
HUT36098A (en)	1985-08-28
GR81869B (fi)	1984-12-12
CH655103A5 (de)	1986-03-27
SE8401321D0 (sv)	1984-03-09

Publication	Publication Date	Title
FI843594L (fi)	1985-03-17	Trihalogenmetylgrupper innehaollande karbonylmetylenheterocykler, foerfarande foer deras framstaellning och ljuskaenslig blandning vilken innehaoller dessa foereningar.
FI840968A (fi)	1984-09-12	Nya azoler, deras framstaellningsprocesser och deras anvaendning.
FI845117L (fi)	1985-06-29	Nya fenyl-imidazoler, deras framstaellning och dessa foereningar innehaollande laekemdel.
FI841128A0 (fi)	1984-03-21	Pyrimidinderivat, deras framstaellning och deras anvaendning.
FI842666A (fi)	1985-01-06	Nya imidazoler, deras framstaellning och dessa foereningar innehaollande laekemedel.
FI855080A0 (fi)	1985-12-19	Nya imidazoderivat, deras framstaellning och dessa foereningar innehaollande laekemedel.
FI852796L (fi)	1986-01-20	Nya pyrimidinderivat, foerfarande foer deras framstaellning och dessa innehaollande kompositioner.
FI843672L (fi)	1985-03-22	Nya pyridoindolderivat, deras framstaellningsfoerfarande och deras anvaendning.
FI841841A0 (fi)	1984-05-08	1-pyrimidinyloxi-3-hetarylalkylamino-2- propanoler, deras framstaellning och anvaendning.
FI855081A (fi)	1986-06-22	Nya imidazoderivat, deras framstaellning och dessa foereningar innehaollande laekemedel.
FI840206A (fi)	1984-07-23	Aminosyraderivat, foerfarande foer deras framstaellning och anvaendning.
FI840675A (fi)	1984-08-23	Nya immunoglobulin producerande hybridcelllinjer, deras anvaendning och foerfarande foer deras framstaellning.
FI841594A0 (fi)	1984-04-19	Nya fenylalkansyraderivat, deras framstaellning och anvaendning.
FI840428A (fi)	1984-08-04	Biologiskt aktivt ketonderivat, framstaellning och anvaendning.
FI845084L (fi)	1985-06-24	Nya benzimidazoler, deras framstaellning och dessa foereningar innehaollande laekemedel.
FI854863A (fi)	1986-06-13	Nya imidazoderivat, dessa foereningar innehaollande laekemedel och foerfarande foer deras framstaellning.
FI842210A0 (fi)	1984-06-01	Kefalosporinester-derivat, deras framstaellning och anvaendning.
FI845086A0 (fi)	1984-12-21	Nya imidazolderivat, deras framstaellning och dessa foereningar innehaollande laekemedel.
FI841615A (fi)	1984-10-28	4-fenyl-tetrahydro-furano-pyridiner, foerfarande foer deras framstaellning och farmaceutiska blandningar.
FI844480L (fi)	1985-05-31	Nya azabicykliska foereningar och foerfarande foer deras framstaellning.
FI853651L (fi)	1986-03-26	Nya hydroxitiaalkener, deras framstaellning och anvaendning.
FI851612A0 (fi)	1985-04-24	Nya apovinkaminolderivat, foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska foereningar.
FI842884A0 (fi)	1984-07-18	Nya tioamider, deras framstaellning och anvaendning.
FI842853A0 (fi)	1984-07-16	Nya 1-fenylimidazolidin-2-on-derivat, deras framstaellning och anvaendning.
FI842300A0 (fi)	1984-06-07	Mono- och ditioestrar, deras framstaellning och anvaendning.

Legal Events

Date	Code	Title	Description
2004-08-31	FD	Application lapsed	Owner name: SANDOZ AG