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FI792058A - Nya 2,6-dimetyl-4,2,3-disubstituerade fenyl-1,4-dihydropyridin-3,5-dikarboxylsyra-3,5-asymmetriska diestrar med blodtryckssaenkande egenskaper samt foerfarande foer framstaellning av dem och farmaceutiska preparat innehaollande desamma - Google Patents

Nya 2,6-dimetyl-4,2,3-disubstituerade fenyl-1,4-dihydropyridin-3,5-dikarboxylsyra-3,5-asymmetriska diestrar med blodtryckssaenkande egenskaper samt foerfarande foer framstaellning av dem och farmaceutiska preparat innehaollande desamma

Info

Publication number
FI792058A
FI792058A FI792058A FI792058A FI792058A FI 792058 A FI792058 A FI 792058A FI 792058 A FI792058 A FI 792058A FI 792058 A FI792058 A FI 792058A FI 792058 A FI792058 A FI 792058A
Authority
FI
Finland
Prior art keywords
sub
disubstituerade
diestrar
dicarboxylsyra
nya
Prior art date
Application number
FI792058A
Other languages
English (en)
Other versions
FI70573C (fi
FI70573B (fi
Inventor
Peder Bernhard Berntsson
Stig Aoke Ingemar Carlsson
Jan Oernulf Gaarder
Bengt Richard Ljung
Original Assignee
Haessle Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20335348&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI792058(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Haessle Ab filed Critical Haessle Ab
Publication of FI792058A publication Critical patent/FI792058A/fi
Application granted granted Critical
Publication of FI70573B publication Critical patent/FI70573B/fi
Publication of FI70573C publication Critical patent/FI70573C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/80—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D211/84—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen directly attached to ring carbon atoms
    • C07D211/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Steroid Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Peptides Or Proteins (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI792058A 1978-06-30 1979-06-29 Analogifoerfarande foer framstaellning av terapeutiskt aktiv 2,6-dimetyl-4-(2,3-diklorfenyl)-1,4-dihydro- pyridin-3,5-dikarboxylsyra-3-metylester-5-etylester FI70573C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE7807404A SE429652B (sv) 1978-06-30 1978-06-30 2.6-dimetyl-4-(2.3-diklorfenyl)-1.4-dihydropyridin-3.5-dikarboxylsyra-3-metylester-5-etylester
SE7807404 1978-06-30

Publications (3)

Publication Number Publication Date
FI792058A true FI792058A (fi) 1979-12-31
FI70573B FI70573B (fi) 1986-06-06
FI70573C FI70573C (fi) 1986-09-24

Family

ID=20335348

Family Applications (1)

Application Number Title Priority Date Filing Date
FI792058A FI70573C (fi) 1978-06-30 1979-06-29 Analogifoerfarande foer framstaellning av terapeutiskt aktiv 2,6-dimetyl-4-(2,3-diklorfenyl)-1,4-dihydro- pyridin-3,5-dikarboxylsyra-3-metylester-5-etylester

Country Status (24)

Country Link
US (1) US4264611A (fi)
EP (1) EP0007293B1 (fi)
JP (1) JPS559083A (fi)
AT (1) ATE1237T1 (fi)
AU (1) AU529116B2 (fi)
BG (1) BG61420B2 (fi)
CA (1) CA1117530A (fi)
CS (1) CS241021B2 (fi)
CY (1) CY1299A (fi)
DD (1) DD144667A5 (fi)
DE (1) DE2963150D1 (fi)
DK (1) DK148978C (fi)
FI (1) FI70573C (fi)
HK (1) HK60585A (fi)
HU (1) HU178568B (fi)
IE (1) IE48650B1 (fi)
LU (2) LU88666I2 (fi)
NL (2) NL930054I2 (fi)
NO (3) NO151965C (fi)
NZ (1) NZ190809A (fi)
SE (1) SE429652B (fi)
SG (1) SG26085G (fi)
SU (2) SU856380A3 (fi)
ZA (1) ZA792804B (fi)

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CN103906508A (zh) 2011-08-26 2014-07-02 沃克哈特有限公司 治疗心血管疾病的方法
AU2014255381A1 (en) 2013-04-17 2015-10-08 Pfizer Inc. N-piperidin-3-ylbenzamide derivatives for treating cardiovascular diseases
CN104177286A (zh) * 2014-08-11 2014-12-03 广东东阳光药业有限公司 一种地平类药物的制备方法
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KR101824982B1 (ko) 2015-10-07 2018-02-02 엘지전자 주식회사 차량 및 그 제어방법
CN107952483B (zh) * 2017-12-18 2020-07-28 万华化学集团股份有限公司 一种催化剂，使用该催化剂的反应器，以及一种制备β-苯乙醇的方法
CN108840819B (zh) * 2018-04-02 2021-07-30 常州瑞明药业有限公司 一种非洛地平的制备方法
JP7470647B2 (ja) 2018-06-14 2024-04-18 アストラゼネカ・ユーケイ・リミテッド ジヒドロピリジン型カルシウムチャネル遮断薬医薬組成物を用いて血圧を低下させるための方法
BR112021013807A2 (pt) 2019-01-18 2021-11-30 Astrazeneca Ab Inibidores de pcsk9 e seus métodos de uso

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GB1552911A (en) * 1975-07-02 1979-09-19 Fujisawa Pharmaceutical Co 1,4 dihydropyridine derivatives and the preparation thereof

Also Published As

Publication number Publication date
CY1299A (en) 1985-10-18
CA1117530A (en) 1982-02-02
NO151965B (no) 1985-04-01
NO792112L (no) 1980-01-03
EP0007293A1 (en) 1980-01-23
JPS559083A (en) 1980-01-22
JPS6121550B2 (fi) 1986-05-27
ATE1237T1 (de) 1982-07-15
FI70573C (fi) 1986-09-24
DK148978C (da) 1986-08-18
NO151965C (no) 1985-07-10
DK275079A (da) 1979-12-31
IE48650B1 (en) 1985-04-03
LU88666I2 (fr) 1996-02-01
NO1996006I1 (no) 1996-06-24
US4264611B1 (fi) 1984-07-17
NL930054I2 (nl) 1994-02-16
NL930054I1 (nl) 1993-09-01
FI70573B (fi) 1986-06-06
SG26085G (en) 1986-01-24
EP0007293B1 (en) 1982-06-23
DD144667A5 (de) 1980-10-29
BG61420B2 (bg) 1997-07-31
AU529116B2 (en) 1983-05-26
SE7807404L (sv) 1979-12-31
SU856380A3 (ru) 1981-08-15
CS241021B2 (en) 1986-03-13
SU915799A3 (en) 1982-03-23
LU88306I2 (fr) 1994-05-04
AU4831679A (en) 1980-02-07
ZA792804B (en) 1980-06-25
SE429652B (sv) 1983-09-19
DK148978B (da) 1985-12-09
DE2963150D1 (en) 1982-08-12
US4264611A (en) 1981-04-28
IE791217L (en) 1979-12-30
HK60585A (en) 1985-08-23
NO1994026I1 (no) 1994-12-21
HU178568B (en) 1982-05-28
NL940012I1 (nl) 1994-08-01
NZ190809A (en) 1982-03-09

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Owner name: AKTIEBOLAGET HAESSLE