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FI51189B - - Google Patents

Info

Publication number
FI51189B
FI51189B FI2460/69A FI246069A FI51189B FI 51189 B FI51189 B FI 51189B FI 2460/69 A FI2460/69 A FI 2460/69A FI 246069 A FI246069 A FI 246069A FI 51189 B FI51189 B FI 51189B
Authority
FI
Finland
Application number
FI2460/69A
Other languages
Finnish (fi)
Other versions
FI51189C (fi
Inventor
Joseph George Lombardino
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Application granted granted Critical
Publication of FI51189B publication Critical patent/FI51189B/fi
Publication of FI51189C publication Critical patent/FI51189C/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D279/00Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/021,2-Thiazines; Hydrogenated 1,2-thiazines

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
FI692460A 1968-08-27 1969-08-25 Menetelmä tulehduksenvastaisina aineina käytettävien 3,4-dihydro-2H-1, 2-bentsotiatsiini-1,1-dioksidien valmistamiseksi. FI51189C (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76759468A 1968-08-27 1968-08-27

Publications (2)

Publication Number Publication Date
FI51189B true FI51189B (pt) 1976-08-02
FI51189C FI51189C (fi) 1976-11-10

Family

ID=25079964

Family Applications (1)

Application Number Title Priority Date Filing Date
FI692460A FI51189C (fi) 1968-08-27 1969-08-25 Menetelmä tulehduksenvastaisina aineina käytettävien 3,4-dihydro-2H-1, 2-bentsotiatsiini-1,1-dioksidien valmistamiseksi.

Country Status (18)

Country Link
US (1) US3591584A (pt)
JP (2) JPS50677B1 (pt)
AT (2) AT298503B (pt)
BE (1) BE737962A (pt)
BR (1) BR6911817D0 (pt)
CH (1) CH520705A (pt)
DE (2) DE1967325C2 (pt)
DK (1) DK145297C (pt)
ES (1) ES370861A1 (pt)
FI (1) FI51189C (pt)
FR (1) FR2016455B1 (pt)
GB (1) GB1257180A (pt)
IL (1) IL32836A (pt)
MY (1) MY7300310A (pt)
NL (1) NL157013B (pt)
NO (1) NO129746B (pt)
PH (1) PH10029A (pt)
SE (2) SE373854B (pt)

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US3927002A (en) * 1973-04-23 1975-12-16 Pfizer N-(pyridyl)-N{40 -alkyl-N{40 -(2-alkoxycarbonylbenzenesulfonyl)-glycineamides and derivatives
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US4474955A (en) * 1981-06-17 1984-10-02 Vincenzo Iannella Process for preparing 4-hydroxy-2-methyl-2H-1,2-benzothiazine-3-[N-(2-pyridinyl)carboxamide]-1,1-dioxide, and its phosphoric ester
GT198276334A (es) * 1981-08-03 1984-01-10 Procedimiento e inter-medios para la produccion de carboxamidas de benzotiazina.
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CA1197244A (en) * 1982-04-16 1985-11-26 Medichem, S.A. Process for the preparation of 4-hydroxy-2-methyl-2h- 1,2-benzothiazine-3-carboxamide-1,1-dioxides
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IT1153293B (it) * 1982-10-22 1987-01-14 Francia Famaceutici S R L Derivati del 4-idrossi-2-metil-2h-1, 2-benzotiazina-3-carbossamide 1, 1-biossido e procedimento per la loro preparazione
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JPS59179683U (ja) * 1983-05-19 1984-11-30 寺田毛織株式会社 貼り合わせふとん
GR80576B (en) * 1983-10-17 1984-11-29 Fujisawa Pharmaceutical Co Thiazine derivatives, process for preparation thereof and pharmaceutical composition comprising the same
US4551452A (en) * 1983-12-21 1985-11-05 Pfizer Inc. Anti-inflammatory 2-methyl-2H-1,2-benzo-(or -thieno-)thiazine-3-carboxamide 1,1-dioxide derivatives, compositions, and method of use therefor
US4656265A (en) * 1984-06-21 1987-04-07 Pfizer Inc. Cyclic prodrugs of antiinflammatory oxicams
DE3437232A1 (de) * 1984-10-10 1986-04-17 Mack Chem Pharm Stabilisierte injektionsloesungen von piroxicam
US4582831A (en) 1984-11-16 1986-04-15 Pfizer Inc. Anti-inflammatory polymorphic monoethanolamine salt of N-(2-pyridyl)-2-methyl-4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide compound, composition, and method of use therefor
CH663899A5 (fr) * 1985-03-20 1988-01-29 Nestle Sa Procede pour la preparation d'une composition a base d'un principe actif de faible hydrosolubilite finement divise.
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EP0259085B1 (en) * 1986-08-29 1991-08-21 Pfizer Inc. 2-guanidino-4-arylthiazoles for treatment of peptic ulcers
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MX174093B (es) * 1987-06-10 1994-04-21 Pfizer 1,1-DIOXIDOS DE 3,4-DIHIDRO-2-ALQUIL-3-OXO-N-ARIL-2H[1] BENZOTIENO[3,2-e]-1,2-TIAZINO-4-CARBOXIAMIDA
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JPH0717589B2 (ja) * 1990-01-22 1995-03-01 ファイザー製薬株式会社 新規1,3―ジカルボニル化合物およびその組成物
JP2988739B2 (ja) * 1990-04-16 1999-12-13 協和醗酵工業株式会社 1,8−ナフチリジン−2−オン誘導体
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JP2964195B2 (ja) * 1992-04-28 1999-10-18 エスエス製薬株式会社 ピロキシカム錠及びその製造法
US5362758A (en) * 1992-09-18 1994-11-08 Pfizer Inc. Ophthalmic piroxicam solution
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US5436241A (en) * 1994-01-14 1995-07-25 Bristol-Myers Squibb Company Topical anti-inflammatory compositions containing piroxicam
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US5952328A (en) * 1997-11-12 1999-09-14 Cephalon, Inc. Benzothiazo and related heterocyclic group-containing cysteine and serine protease inhibitors
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US20050222227A1 (en) * 2004-04-01 2005-10-06 Pfizer Inc Oxazole-amine compounds for the treatment of neurodegenerative disorders
JP2009529057A (ja) 2006-03-08 2009-08-13 コートリア・コーポレーシヨン Cox−関連胃損傷を予防するための非−選択的cox阻害剤との組み合わせ療法
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Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1302858B (pt) * 1962-09-21 1972-05-04

Also Published As

Publication number Publication date
SE373854B (pt) 1975-02-17
BR6911817D0 (pt) 1973-02-13
DE1943265B2 (de) 1981-05-14
FR2016455A1 (pt) 1970-05-08
CH520705A (fr) 1972-03-31
DE1943265C3 (de) 1982-02-04
DE1967325B2 (de) 1981-08-13
PH10029A (en) 1976-07-13
NO129746B (pt) 1974-05-20
FR2016455B1 (pt) 1974-02-01
IL32836A (en) 1972-08-30
MY7300310A (en) 1973-12-31
GB1257180A (pt) 1971-12-15
NL6912981A (pt) 1970-03-03
BE737962A (pt) 1970-02-26
DE1967325C2 (de) 1982-03-18
ES370861A1 (es) 1971-07-01
AT298503B (de) 1972-05-10
IL32836A0 (en) 1969-11-12
AT294113B (de) 1971-11-10
JPS5142114B1 (pt) 1976-11-13
NL157013B (nl) 1978-06-15
JPS50677B1 (pt) 1975-01-10
FI51189C (fi) 1976-11-10
DK145297B (da) 1982-10-25
DE1943265A1 (de) 1970-08-13
US3591584A (en) 1971-07-06
DK145297C (da) 1983-03-14
SE402459B (sv) 1978-07-03

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