[go: up one dir, main page]
More Web Proxy on the site http://driver.im/

ES8802317A1 - Un procedimiento para preparar derivados de acido (2-aminosustituido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico - Google Patents

Un procedimiento para preparar derivados de acido (2-aminosustituido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico

Info

Publication number
ES8802317A1
ES8802317A1 ES554495A ES554495A ES8802317A1 ES 8802317 A1 ES8802317 A1 ES 8802317A1 ES 554495 A ES554495 A ES 554495A ES 554495 A ES554495 A ES 554495A ES 8802317 A1 ES8802317 A1 ES 8802317A1
Authority
ES
Spain
Prior art keywords
stands
hydrogen
production
organic residue
antibiotic derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES554495A
Other languages
English (en)
Other versions
ES554495A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Chemical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/JP1985/000247 external-priority patent/WO1986006380A1/ja
Priority claimed from PCT/JP1985/000394 external-priority patent/WO1987000527A1/ja
Priority claimed from JP61063735A external-priority patent/JPS62228075A/ja
Application filed by Takeda Chemical Industries Ltd filed Critical Takeda Chemical Industries Ltd
Publication of ES554495A0 publication Critical patent/ES554495A0/es
Publication of ES8802317A1 publication Critical patent/ES8802317A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

LOS DERIVADOS DEL ACIDO (2-AMINO-SUSTITUIDO-3-OXO-2-ISOXAZOLIDINIL)-5-OXO-2-TETRAHIDROFURANCARBOXILICO (I), DONDE NO EXCLUSIVAMENTE, R1 ES AMINO O RESTO UNIDO POR NITROGENO, R2 CARBOXILO O GRUPO DERIVABLE, Y R3, R4, R5, R6, R7 Y R8 SON HIDROGENO O RESIDUO ORGANICO Y X ES HIDROGENO, METOXI O FORMILAMINO; SE OBTIENEN HACIENDO REACCIONAR (II) CON (III), EN UN DISOLVENTE TAL COMO LA N,N-DIMETILFORMANIDA EN PRESENCIA DE UN AGENTE DE CONDENSACION O ACIDO DE LEWIS, A UNA TEMPERATURA ENTRE C10 Y 100JC DURANTE 5 MINUTOS A 30 HORAS. ES UN ANTIBACTERIANO GRAM-POSITIVO Y GRAM-NEGATIVO DE BAJA TOXICIDAD, POR LO QUE ES APLICABLE EN EL TRATAMIENTO DE INFECCIONES DE TRACTO RESPIRATORIO, URINARIO, DE LOS CONDUCTOS BILIARES, ETC.
ES554495A 1985-04-30 1986-04-29 Un procedimiento para preparar derivados de acido (2-aminosustituido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico Expired ES8802317A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
PCT/JP1985/000247 WO1986006380A1 (en) 1985-04-30 1985-04-30 Antibacterial compounds, use and preparation thereof
PCT/JP1985/000394 WO1987000527A1 (en) 1985-07-12 1985-07-12 Antibacterial compounds, their use, and process for their preparation
JP28415485 1985-12-16
JP61063735A JPS62228075A (ja) 1985-04-30 1986-03-20 抗菌性化合物，その製造法および用途

Publications (2)

Publication Number Publication Date
ES554495A0 ES554495A0 (es) 1988-05-01
ES8802317A1 true ES8802317A1 (es) 1988-05-01

Family

ID=27464357

Family Applications (2)

Application Number Title Priority Date Filing Date
ES554495A Expired ES8802317A1 (es) 1985-04-30 1986-04-29 Un procedimiento para preparar derivados de acido (2-aminosustituido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico
ES557661A Expired ES8801650A1 (es) 1985-04-30 1987-08-13 Un metodo para preparar derivados de acido (2-amino sustutuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico.

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES557661A Expired ES8801650A1 (es) 1985-04-30 1987-08-13 Un metodo para preparar derivados de acido (2-amino sustutuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico.

Country Status (6)

Country Link
US (1) US4851422A (es)
EP (1) EP0219923B1 (es)
CN (1) CN86102923A (es)
CA (1) CA1285950C (es)
DE (1) DE3686632T2 (es)
ES (2) ES8802317A1 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4882434A (en) * 1986-10-29 1989-11-21 Takeda Chemical Industries, Ltd. Gamma-lactonecarboxylic acid derivatives and their use as antibacterial agents or intermediates
WO1999019295A1 (en) 1997-10-10 1999-04-22 Trustees Of The University Of Pennsylvania Compositions and methods for inhibiting arginase activity
WO2000041473A2 (de) * 1999-01-13 2000-07-20 Jomaa Pharmaka Gmbh Verwendung von 3-isoxazolidinonen und hydroxylaminsäuren zur behandlung von infektionen
NZ564743A (en) * 2005-07-11 2010-03-26 Mitsubishi Tanabe Pharma Corp An oxime derivative as a glucokinase activating agent and preparations thereof
US11780832B2 (en) * 2021-03-31 2023-10-10 Fedora Pharmaceuticals Inc. Lactivicin compounds, their preparation and use as antibacterial agents

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1768114A1 (de) * 1968-04-02 1971-10-07 Bayer Ag Verfahren zur Herstellung von alpha-Ketoglutarsaeure
JPS57179133A (en) * 1981-04-27 1982-11-04 Mitsui Toatsu Chem Inc Synthesis of gamma-ketocarboxylic acid and its ester
IL67451A (en) * 1981-12-25 1987-10-20 Takeda Chemical Industries Ltd 4-cyano-2-azetidinones and production thereof and process for the preparation of 4-carbamoyl-2-azetidinones using them
US4546101A (en) * 1982-09-10 1985-10-08 Fujisawa Pharmaceutical Co., Ltd. New cephem compounds useful for treating infectious diseases in human being and animals and processes for preparation thereof
US4595532A (en) * 1983-02-02 1986-06-17 University Of Notre Dame Du Lac N-(substituted-methyl)-azetidin-2-ones
EP0146735A1 (de) * 1983-11-23 1985-07-03 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Optisch einheitliche beta-Lactame
US4656288A (en) * 1984-03-29 1987-04-07 Takeda Chemical Industries, Ltd. Antibiotics, their production and use
JPH0473775A (ja) * 1990-07-13 1992-03-09 Mutoh Ind Ltd 電子写真装置
JPH0473772A (ja) * 1990-07-13 1992-03-09 Toshiba Corp 画像形成装置

Also Published As

Publication number Publication date
US4851422A (en) 1989-07-25
CA1285950C (en) 1991-07-09
DE3686632T2 (de) 1993-01-21
CN86102923A (zh) 1986-11-12
ES554495A0 (es) 1988-05-01
DE3686632D1 (de) 1992-10-08
EP0219923A1 (en) 1987-04-29
ES557661A0 (es) 1988-02-16
EP0219923B1 (en) 1992-09-02
ES8801650A1 (es) 1988-02-16

Similar Documents

Publication Publication Date Title
CA2290709A1 (en) 2,6-diaminopyridine compounds as intermediates for producing antibacterial dihydropyridone carboxylic acid derivatives
MY108967A (en) Triazolopyridazine compounds, their production and use
ES468173A1 (es) Un procedimiento para la preparacion de derivados de morfina
HUT50345A (en) Process for production of cefem-derivatives and their intermediers
MX9203548A (es) Compuestos de penem, su produccion y uso.
NZ333991A (en) method of preparing cyclohexene carboxylate derivatives
ES2001794A6 (es) Un procedimiento para la preparacion de derivados de quinolina
ES8301915A1 (es) Procedimiento para preparar derivados de 2-oxoazetidina .
CA2014490A1 (en) Diaminoethylene compounds
CA2036163A1 (en) Novel beta-lactam compounds and their production
ES8802317A1 (es) Un procedimiento para preparar derivados de acido (2-aminosustituido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carboxilico
JPS57134485A (en) Trisubstituted pyrimidopyrimidine
ES2004079A6 (es) Procedimiento para la preparacion de derivados aminicos antimicoticos y agrofungicidas
TW238304B (en) A process for the preparation of 1-substituted-5(4H)-tetrazolinones
ES468170A1 (es) Un procedimiento para la preparacion de un nuevo derivado demorfina
EP0601191A4 (en) Novel tetracyclic compound.
ES8705431A1 (es) Un metodo para producir derivados de acido 2-(4-amino susti-tuido-3-oxo-2-isoxazolidinil)-5-oxo-2-tetrahidrofuran-carbo-xilico
CA2208520A1 (en) Diclavulanate salt with a diamino ether and process of preparation
ES473182A1 (es) Procedimiento para la preparacion de compuestos triciclicos con cabeza de puente de nitrogeno
JPS6450880A (en) 7-(2-methyl-4-aminopyrrolidinyl)naphthylidine and quinoline compound
EP1227081A4 (en) PROCESS FOR THE PREPARATION OF OXYMINOALKANOIC ACID DERIVATIVES
ES8101646A1 (es) Un procedimiento para producir un compuesto opticamente ac- tivo
CA2053705A1 (en) Piperazine derivatives
ES8200142A1 (es) Un procedimiento para la produccion de analogos de cefalosporina.
EP0271586A4 (en) COMPOUNDS OF -g (b) -LACTAM AND THEIR PREPARATION PROCESS.

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19990201